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Pharmacophore-Based Virtual Screening to Discover New Active Compounds for Human Choline Kinase α1.
Mol Inform. 2015 Jun;34(6-7):458-66. doi: 10.1002/minf.201400140. Epub 2015 Jun 18.
Mol Inform. 2015.
PMID: 27490389
Design, synthesis, crystallization and biological evaluation of new symmetrical biscationic compounds as selective inhibitors of human Choline Kinase α1 (ChoKα1).
Schiaffino-Ortega S, Baglioni E, Mariotto E, Bortolozzi R, Serrán-Aguilera L, Ríos-Marco P, Carrasco-Jimenez MP, Gallo MA, Hurtado-Guerrero R, Marco C, Basso G, Viola G, Entrena A, López-Cara LC.
Schiaffino-Ortega S, et al. Among authors: serran aguilera l.
Sci Rep. 2016 Mar 31;6:23793. doi: 10.1038/srep23793.
Sci Rep. 2016.
PMID: 27029499
Free PMC article.
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Choline kinase active site provides features for designing versatile inhibitors.
Serran-Aguilera L, Nuti R, López-Cara LC, Ríos-Marco P, Carrasco MP, Marco C, Entrena A, Macchiarulo A, Hurtado-Guerrero R.
Serran-Aguilera L, et al.
Curr Top Med Chem. 2014;14(23):2684-93. doi: 10.2174/1568026614666141216093337.
Curr Top Med Chem. 2014.
PMID: 25515750
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Plasmodium falciparum Choline Kinase Inhibition Leads to a Major Decrease in Phosphatidylethanolamine Causing Parasite Death.
Serrán-Aguilera L, Denton H, Rubio-Ruiz B, López-Gutiérrez B, Entrena A, Izquierdo L, Smith TK, Conejo-García A, Hurtado-Guerrero R.
Serrán-Aguilera L, et al.
Sci Rep. 2016 Sep 12;6:33189. doi: 10.1038/srep33189.
Sci Rep. 2016.
PMID: 27616047
Free PMC article.
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Synthesis, biological evaluation, in silico modeling and crystallization of novel small monocationic molecules with potent antiproliferative activity by dual mechanism.
Serrán-Aguilera L, Mariotto E, Rubbini G, Castro Navas FF, Marco C, Carrasco-Jiménez MP, Ballarotto M, Macchiarulo A, Hurtado-Guerrero R, Viola G, Lopez-Cara LC.
Serrán-Aguilera L, et al.
Eur J Med Chem. 2020 Dec 1;207:112797. doi: 10.1016/j.ejmech.2020.112797. Epub 2020 Sep 6.
Eur J Med Chem. 2020.
PMID: 32977218
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Recent advances in the design of choline kinase α inhibitors and the molecular basis of their inhibition.
Rubio-Ruiz B, Serrán-Aguilera L, Hurtado-Guerrero R, Conejo-García A.
Rubio-Ruiz B, et al. Among authors: serran aguilera l.
Med Res Rev. 2021 Mar;41(2):902-927. doi: 10.1002/med.21746. Epub 2020 Oct 25.
Med Res Rev. 2021.
PMID: 33103259
Free article.
Review.
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