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Pyrrolyl and Indolyl α-γ-Diketo Acid Derivatives Acting as Selective Inhibitors of Human Carbonic Anhydrases IX and XII.
Ialongo D, Messore A, Madia VN, Tudino V, Nocentini A, Gratteri P, Giovannuzzi S, Supuran CT, Nicolai A, Scarpa S, Taurone S, Camarda M, Artico M, Papa V, Saccoliti F, Scipione L, Di Santo R, Costi R. Ialongo D, et al. Among authors: saccoliti f. Pharmaceuticals (Basel). 2023 Jan 27;16(2):188. doi: 10.3390/ph16020188. Pharmaceuticals (Basel). 2023. PMID: 37259337 Free PMC article.
Analytical Characterization of an Inulin-Type Fructooligosaccharide from Root-Tubers of Asphodelusramosus L.
Madia VN, De Vita D, Messore A, Toniolo C, Tudino V, De Leo A, Pindinello I, Ialongo D, Saccoliti F, D'Ursi AM, Grimaldi M, Ceccobelli P, Scipione L, Di Santo R, Costi R. Madia VN, et al. Among authors: saccoliti f. Pharmaceuticals (Basel). 2021 Mar 19;14(3):278. doi: 10.3390/ph14030278. Pharmaceuticals (Basel). 2021. PMID: 33808608 Free PMC article.
Structure-activity relationship of pyrrolyl diketo acid derivatives as dual inhibitors of HIV-1 integrase and reverse transcriptase ribonuclease H domain.
Cuzzucoli Crucitti G, Métifiot M, Pescatori L, Messore A, Madia VN, Pupo G, Saccoliti F, Scipione L, Tortorella S, Esposito F, Corona A, Cadeddu M, Marchand C, Pommier Y, Tramontano E, Costi R, Di Santo R. Cuzzucoli Crucitti G, et al. Among authors: saccoliti f. J Med Chem. 2015 Feb 26;58(4):1915-28. doi: 10.1021/jm501799k. Epub 2015 Feb 11. J Med Chem. 2015. PMID: 25629256 Free PMC article.
N-Substituted Quinolinonyl Diketo Acid Derivatives as HIV Integrase Strand Transfer Inhibitors and Their Activity against RNase H Function of Reverse Transcriptase.
Pescatori L, Métifiot M, Chung S, Masoaka T, Cuzzucoli Crucitti G, Messore A, Pupo G, Madia VN, Saccoliti F, Scipione L, Tortorella S, Di Leva FS, Cosconati S, Marinelli L, Novellino E, Le Grice SF, Pommier Y, Marchand C, Costi R, Di Santo R. Pescatori L, et al. Among authors: saccoliti f. J Med Chem. 2015 Jun 11;58(11):4610-23. doi: 10.1021/acs.jmedchem.5b00159. Epub 2015 May 26. J Med Chem. 2015. PMID: 25961960 Free PMC article.
Structure-Activity Relationships on Cinnamoyl Derivatives as Inhibitors of p300 Histone Acetyltransferase.
Madia VN, Benedetti R, Barreca ML, Ngo L, Pescatori L, Messore A, Pupo G, Saccoliti F, Valente S, Mai A, Scipione L, Zheng YG, Tintori C, Botta M, Cecchetti V, Altucci L, Di Santo R, Costi R. Madia VN, et al. Among authors: saccoliti f. ChemMedChem. 2017 Aug 22;12(16):1359-1368. doi: 10.1002/cmdc.201700040. Epub 2017 Apr 12. ChemMedChem. 2017. PMID: 28346821
Novel Benzazole Derivatives Endowed with Potent Antiheparanase Activity.
Madia VN, Messore A, Pescatori L, Saccoliti F, Tudino V, De Leo A, Bortolami M, Scipione L, Costi R, Rivara S, Scalvini L, Mor M, Ferrara FF, Pavoni E, Roscilli G, Cassinelli G, Milazzo FM, Battistuzzi G, Di Santo R, Giannini G. Madia VN, et al. Among authors: saccoliti f. J Med Chem. 2018 Aug 9;61(15):6918-6936. doi: 10.1021/acs.jmedchem.8b00908. Epub 2018 Jul 30. J Med Chem. 2018. PMID: 30010344
In Vitro Antiviral Activity of New Oxazoline Derivatives as Potent Poliovirus Inhibitors.
Madia VN, Messore A, Pescatori L, Saccoliti F, Tudino V, De Leo A, Scipione L, Fiore L, Rhoden E, Manetti F, Oberste MS, Di Santo R, Costi R. Madia VN, et al. Among authors: saccoliti f. J Med Chem. 2019 Jan 24;62(2):798-810. doi: 10.1021/acs.jmedchem.8b01482. Epub 2018 Dec 18. J Med Chem. 2019. PMID: 30512950 Free PMC article.
Discovery of a pyrimidine compound endowed with antitumor activity.
Taglieri L, Saccoliti F, Nicolai A, Peruzzi G, Madia VN, Tudino V, Messore A, Di Santo R, Artico M, Taurone S, Salvati M, Costi R, Scarpa S. Taglieri L, et al. Among authors: saccoliti f. Invest New Drugs. 2020 Feb;38(1):39-49. doi: 10.1007/s10637-019-00762-y. Epub 2019 Mar 21. Invest New Drugs. 2020. PMID: 30900116
26 results