Ruchaud S - Search Results

1

Kinase-Based Screening of Marine Natural Extracts Leads to the Identification of a Cytotoxic High Molecular Weight Metabolite from the Mediterranean Sponge Crambe tailliezi.

Nguyen TN, Feizbakhsh O, Sfecci E, Baratte B, Delehouzé C, Garcia A, Moulin C, Colas P, Ruchaud S, Mehiri M, Bach S. Nguyen TN, et al. Among authors: ruchaud s. Mar Drugs. 2019 Oct 9;17(10):569. doi: 10.3390/md17100569. Mar Drugs. 2019. PMID: 31600933 Free PMC article.

2

Neurymenolide A, a Novel Mitotic Spindle Poison from the New Caledonian Rhodophyta Phacelocarpus neurymenioides.

Motuhi SE, Feizbakhsh O, Foll-Josselin B, Baratte B, Delehouzé C, Cousseau A, Fant X, Bulinski JC, Payri CE, Ruchaud S, Mehiri M, Bach S. Motuhi SE, et al. Among authors: ruchaud s. Mar Drugs. 2019 Feb 1;17(2):93. doi: 10.3390/md17020093. Mar Drugs. 2019. PMID: 30717235 Free PMC article.

3

Discovery of simplified benzazole fragments derived from the marine benzosceptrin B as necroptosis inhibitors involving the receptor interacting protein Kinase-1.

Benchekroun M, Ermolenko L, Tran MQ, Vagneux A, Nedev H, Delehouzé C, Souab M, Baratte B, Josselin B, Iorga BI, Ruchaud S, Bach S, Al-Mourabit A. Benchekroun M, et al. Among authors: ruchaud s. Eur J Med Chem. 2020 Sep 1;201:112337. doi: 10.1016/j.ejmech.2020.112337. Epub 2020 Jun 25. Eur J Med Chem. 2020. PMID: 32659605

4

Design of new disubstituted imidazo[1,2-b]pyridazine derivatives as selective Haspin inhibitors. Synthesis, binding mode and anticancer biological evaluation.

Elie J, Feizbakhsh O, Desban N, Josselin B, Baratte B, Bescond A, Duez J, Fant X, Bach S, Marie D, Place M, Ben Salah S, Chartier A, Berteina-Raboin S, Chaikuad A, Knapp S, Carles F, Bonnet P, Buron F, Routier S, Ruchaud S. Elie J, et al. Among authors: ruchaud s. J Enzyme Inhib Med Chem. 2020 Dec;35(1):1840-1853. doi: 10.1080/14756366.2020.1825408. J Enzyme Inhib Med Chem. 2020. PMID: 33040634 Free PMC article.

5

From Synthetic Simplified Marine Metabolite Analogues to New Selective Allosteric Inhibitor of Aurora B Kinase.

Juillet C, Ermolenko L, Boyarskaya D, Baratte B, Josselin B, Nedev H, Bach S, Iorga BI, Bignon J, Ruchaud S, Al-Mourabit A. Juillet C, et al. Among authors: ruchaud s. J Med Chem. 2021 Jan 28;64(2):1197-1219. doi: 10.1021/acs.jmedchem.0c02064. Epub 2021 Jan 8. J Med Chem. 2021. PMID: 33417773

6

Bioactive Metabolites from the Deep Subseafloor Fungus Oidiodendron griseum UBOCC-A-114129.

Navarri M, Jégou C, Bondon A, Pottier S, Bach S, Baratte B, Ruchaud S, Barbier G, Burgaud G, Fleury Y. Navarri M, et al. Among authors: ruchaud s. Mar Drugs. 2017 Apr 7;15(4):111. doi: 10.3390/md15040111. Mar Drugs. 2017. PMID: 28387732 Free PMC article.

7

Structure Activity Relationship Studies around DB18, a Potent and Selective Inhibitor of CLK Kinases.

Brahmaiah D, Bhavani AKD, Aparna P, Kumar NS, Solhi H, Le Guevel R, Baratte B, Robert T, Ruchaud S, Bach S, Jadav SS, Reddy CR, Mosset P, Gouault N, Levoin N, Grée R. Brahmaiah D, et al. Among authors: ruchaud s. Molecules. 2022 Sep 20;27(19):6149. doi: 10.3390/molecules27196149. Molecules. 2022. PMID: 36234686 Free PMC article.

8

Discovery of DB18, a potent inhibitor of CLK kinases with a high selectivity against DYRK1A kinase.

Brahmaiah D, Kanaka Durga Bhavani A, Aparna P, Sampath Kumar N, Solhi H, Le Guevel R, Baratte B, Ruchaud S, Bach S, Singh Jadav S, Raji Reddy C, Roisnel T, Mosset P, Levoin N, Grée R. Brahmaiah D, et al. Among authors: ruchaud s. Bioorg Med Chem. 2021 Feb 1;31:115962. doi: 10.1016/j.bmc.2020.115962. Epub 2020 Dec 31. Bioorg Med Chem. 2021. PMID: 33422908

9

Exploration of 7-azaindole-coumaranone hybrids and their analogues as protein kinase inhibitors.

Qhobosheane MA, Beteck RM, Baratte B, Robert T, Ruchaud S, Bach S, Legoabe LJ. Qhobosheane MA, et al. Among authors: ruchaud s. Chem Biol Interact. 2021 Jul 1;343:109478. doi: 10.1016/j.cbi.2021.109478. Epub 2021 Apr 25. Chem Biol Interact. 2021. PMID: 33905741

10

Synthesis, biological evaluation and molecular modeling studies of imidazo[1,2-a]pyridines derivatives as protein kinase inhibitors.

Lawson M, Rodrigo J, Baratte B, Robert T, Delehouzé C, Lozach O, Ruchaud S, Bach S, Brion JD, Alami M, Hamze A. Lawson M, et al. Among authors: ruchaud s. Eur J Med Chem. 2016 Nov 10;123:105-114. doi: 10.1016/j.ejmech.2016.07.040. Epub 2016 Jul 21. Eur J Med Chem. 2016. PMID: 27474927

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