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A G358S mutation in the Plasmodium falciparum Na+ pump PfATP4 confers clinically-relevant resistance to cipargamin.
Nat Commun. 2022 Sep 30;13(1):5746. doi: 10.1038/s41467-022-33403-9.
Nat Commun. 2022.
PMID: 36180431
Free PMC article.
Diverse antimalarials from whole-cell phenotypic screens disrupt malaria parasite ion and volume homeostasis.
Dennis ASM, Rosling JEO, Lehane AM, Kirk K.
Dennis ASM, et al. Among authors: rosling jeo.
Sci Rep. 2018 Jun 11;8(1):8795. doi: 10.1038/s41598-018-26819-1.
Sci Rep. 2018.
PMID: 29892073
Free PMC article.
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Biochemical characterization and chemical inhibition of PfATP4-associated Na+-ATPase activity in Plasmodium falciparum membranes.
Rosling JEO, Ridgway MC, Summers RL, Kirk K, Lehane AM.
Rosling JEO, et al.
J Biol Chem. 2018 Aug 24;293(34):13327-13337. doi: 10.1074/jbc.RA118.003640. Epub 2018 Jul 9.
J Biol Chem. 2018.
PMID: 29986883
Free PMC article.
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