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Differential specificity of SARS-CoV-2 main protease variants on peptide versus protein-based substrates.
FEBS J. 2024 Jan;291(1):61-69. doi: 10.1111/febs.16970. Epub 2023 Nov 3.
FEBS J. 2024.
PMID: 37843490
Nitriles: an attractive approach to the development of covalent inhibitors.
Bonatto V, Lameiro RF, Rocho FR, Lameira J, Leitão A, Montanari CA.
Bonatto V, et al. Among authors: rocho fr.
RSC Med Chem. 2022 Nov 7;14(2):201-217. doi: 10.1039/d2md00204c. eCollection 2023 Feb 22.
RSC Med Chem. 2022.
PMID: 36846367
Free PMC article.
Review.
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A patent review on cathepsin K inhibitors to treat osteoporosis (2011 - 2021).
Rocho FR, Bonatto V, Lameiro RF, Lameira J, Leitão A, Montanari CA.
Rocho FR, et al.
Expert Opin Ther Pat. 2022 May;32(5):561-573. doi: 10.1080/13543776.2022.2040480. Epub 2022 Mar 10.
Expert Opin Ther Pat. 2022.
PMID: 35137661
Review.
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Nitrile-based peptoids as cysteine protease inhibitors.
Alves L, Santos DA, Cendron R, Rocho FR, Matos TKB, Leitão A, Montanari CA.
Alves L, et al. Among authors: rocho fr.
Bioorg Med Chem. 2021 Jul 1;41:116211. doi: 10.1016/j.bmc.2021.116211. Epub 2021 May 10.
Bioorg Med Chem. 2021.
PMID: 33991733
Free article.
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