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Discovery of non-boronic acid Arginase 1 inhibitors through virtual screening and biophysical methods.
Bioorg Med Chem Lett. 2023 Mar 15;84:129193. doi: 10.1016/j.bmcl.2023.129193. Epub 2023 Feb 21.
Bioorg Med Chem Lett. 2023.
PMID: 36822300
Discovery of IDO1 inhibitors containing a decahydroquinoline, decahydro-1,6-naphthyridine, or octahydro-1H-pyrrolo[3,2-c]pyridine scaffold.
Yu W, Deng Y, Sloman D, Li D, Liu K, Fradera X, Lesburg CA, Martinot T, Doty A, Ferguson H, Richard Miller J, Knemeyer I, Otte K, Vincent S, Sciammetta N, Jonathan Bennett D, Han Y.
Yu W, et al. Among authors: richard miller j.
Bioorg Med Chem Lett. 2021 Oct 1;49:128314. doi: 10.1016/j.bmcl.2021.128314. Epub 2021 Aug 13.
Bioorg Med Chem Lett. 2021.
PMID: 34391891
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