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Synthesis and in vitro antimycobacterial activity of 3-substituted 5-hydroxy-5-trifluoro[chloro]methyl-4,5-dihydro-1H-1-(isonicotinoyl) pyrazoles.
Almeida da Silva PE, Ramos DF, Bonacorso HG, de la Iglesia AI, Oliveira MR, Coelho T, Navarini J, Morbidoni HR, Zanatta N, Martins MA. Almeida da Silva PE, et al. Among authors: ramos df. Int J Antimicrob Agents. 2008 Aug;32(2):139-44. doi: 10.1016/j.ijantimicag.2008.03.019. Epub 2008 Jun 20. Int J Antimicrob Agents. 2008. PMID: 18571384
In vitro and in silico analysis of the efficiency of tetrahydropyridines as drug efflux inhibitors in Escherichia coli.
Silva L Jr, Carrion LL, von Groll A, Costa SS, Junqueira E, Ramos DF, Cantos J, Seus VR, Couto I, Fernandes LD, Bonacorso HG, Martins MA, Zanatta N, Viveiros M, Machado KS, Almeida da Silva PE. Silva L Jr, et al. Among authors: ramos df. Int J Antimicrob Agents. 2017 Mar;49(3):308-314. doi: 10.1016/j.ijantimicag.2016.11.024. Epub 2017 Jan 30. Int J Antimicrob Agents. 2017. PMID: 28153476 Free article.
Alternative Pharmaceutical Formulation for Oral Administration of Rifampicin.
Halicki PCB, Hädrich G, Boschero R, Ferreira LA, von Groll A, da Silva PEA, Dora CL, Ramos DF. Halicki PCB, et al. Among authors: ramos df. Assay Drug Dev Technol. 2018 Dec;16(8):456-461. doi: 10.1089/adt.2018.874. Epub 2018 Oct 16. Assay Drug Dev Technol. 2018. PMID: 30325673
Tetrahydropyridine derivative as efflux inhibitor in Mycobacterium abscessus.
Vianna JS, Ramis IB, Bierhals D, von Groll A, Ramos DF, Zanatta N, Lourenço MC, Viveiros M, Almeida da Silva PE. Vianna JS, et al. Among authors: ramos df. J Glob Antimicrob Resist. 2019 Jun;17:296-299. doi: 10.1016/j.jgar.2018.12.020. Epub 2019 Jan 7. J Glob Antimicrob Resist. 2019. PMID: 30630106
Design of hybrid molecules as antimycobacterial compounds: Synthesis of isoniazid-naphthoquinone derivatives and their activity against susceptible and resistant strains of Mycobacterium tuberculosis.
Reis WJ, Bozzi ÍAO, Ribeiro MF, Halicki PCB, Ferreira LA, Almeida da Silva PE, Ramos DF, de Simone CA, da Silva Júnior EN. Reis WJ, et al. Among authors: ramos df. Bioorg Med Chem. 2019 Sep 15;27(18):4143-4150. doi: 10.1016/j.bmc.2019.07.045. Epub 2019 Jul 27. Bioorg Med Chem. 2019. PMID: 31378595 Free article.
Development of Lipid Nanocarriers for Tuberculosis Treatment: Evaluation of Suitable Excipients and Nanocarriers.
Hädrich G, Vaz GR, Boschero R, Appel AS, Ramos C, Halicki PCB, Bidone J, Teixeira HF, Muccillo-Baisch AL, Dal-Bó A, Silva Pinto L, Dailey LA, Da Silva PEA, Ramos DF, Dora CL. Hädrich G, et al. Among authors: ramos df, ramos c. Curr Drug Deliv. 2021;18(6):770-778. doi: 10.2174/1567201818666210212092112. Curr Drug Deliv. 2021. PMID: 33583376
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