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Novel N-aryl nicotinamide derivatives: Taking stock on 3,6-diazabicyclo[3.1.1]heptanes as ligands for neuronal acetylcholine receptors.
Eur J Med Chem. 2019 Oct 15;180:51-61. doi: 10.1016/j.ejmech.2019.06.079. Epub 2019 Jul 5.
Eur J Med Chem. 2019.
PMID: 31299587
Free article.
From pyrrolidinyl-benzodioxane to pyrrolidinyl-pyridodioxanes, or from unselective antagonism to selective partial agonism at α4β2 nicotinic acetylcholine receptor.
Bolchi C, Bavo F, Gotti C, Fumagalli L, Fasoli F, Binda M, Mucchietto V, Sciaccaluga M, Plutino S, Fucile S, Pallavicini M.
Bolchi C, et al. Among authors: plutino s.
Eur J Med Chem. 2017 Jan 5;125:1132-1144. doi: 10.1016/j.ejmech.2016.10.048. Epub 2016 Oct 21.
Eur J Med Chem. 2017.
PMID: 27810599
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Pyridinyl- and pyridazinyl-3,6-diazabicyclo[3.1.1]heptane-anilines: Novel selective ligands with subnanomolar affinity for α4β2 nACh receptors.
Deligia F, Murineddu G, Gotti C, Ragusa G, Fasoli F, Sciaccaluga M, Plutino S, Fucile S, Loriga G, Asproni B, Pinna GA.
Deligia F, et al. Among authors: plutino s.
Eur J Med Chem. 2018 May 25;152:401-416. doi: 10.1016/j.ejmech.2018.04.026. Epub 2018 Apr 17.
Eur J Med Chem. 2018.
PMID: 29751234
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The fifth subunit in α3β4 nicotinic receptor is more than an accessory subunit.
Crespi A, Plutino S, Sciaccaluga M, Righi M, Borgese N, Fucile S, Gotti C, Colombo SF.
Crespi A, et al. Among authors: plutino s.
FASEB J. 2018 Aug;32(8):4190-4202. doi: 10.1096/fj.201701377R. Epub 2018 Mar 5.
FASEB J. 2018.
PMID: 29505300
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Extracellular mild acidosis decreases the Ca2+ permeability of the human NMDA receptors.
Plutino S, Sciaccaluga M, Fucile S.
Plutino S, et al.
Cell Calcium. 2019 Jun;80:63-70. doi: 10.1016/j.ceca.2019.04.001. Epub 2019 Apr 4.
Cell Calcium. 2019.
PMID: 30978540
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Barrel cortex development lacks a key stage of hyperconnectivity from deep to superficial layers in a rat model of Absence Epilepsy.
Plutino S, Laghouati E, Jarre G, Depaulis A, Guillemain I, Bureau I.
Plutino S, et al.
Prog Neurobiol. 2024 Mar;234:102564. doi: 10.1016/j.pneurobio.2023.102564. Epub 2024 Jan 19.
Prog Neurobiol. 2024.
PMID: 38244975
Free article.
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