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Discovery and selection of TMC114, a next generation HIV-1 protease inhibitor.
J Med Chem. 2005 Mar 24;48(6):1813-22. doi: 10.1021/jm049560p.
J Med Chem. 2005.
PMID: 15771427
Structure-activity relationship study on a novel series of cyclopentane-containing macrocyclic inhibitors of the hepatitis C virus NS3/4A protease leading to the discovery of TMC435350.
Raboisson P, de Kock H, Rosenquist A, Nilsson M, Salvador-Oden L, Lin TI, Roue N, Ivanov V, Wähling H, Wickström K, Hamelink E, Edlund M, Vrang L, Vendeville S, Van de Vreken W, McGowan D, Tahri A, Hu L, Boutton C, Lenz O, Delouvroy F, Pille G, Surleraux D, Wigerinck P, Samuelsson B, Simmen K.
Raboisson P, et al.
Bioorg Med Chem Lett. 2008 Sep 1;18(17):4853-8. doi: 10.1016/j.bmcl.2008.07.088. Epub 2008 Jul 24.
Bioorg Med Chem Lett. 2008.
PMID: 18678486
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Design and optimization of tricyclic phtalimide analogues as novel inhibitors of HIV-1 integrase.
Verschueren WG, Dierynck I, Amssoms KI, Hu L, Boonants PM, Pille GM, Daeyaert FF, Hertogs K, Surleraux DL, Wigerinck PB.
Verschueren WG, et al. Among authors: pille gm.
J Med Chem. 2005 Mar 24;48(6):1930-40. doi: 10.1021/jm049559q.
J Med Chem. 2005.
PMID: 15771437
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Design of HIV-1 protease inhibitors active on multidrug-resistant virus.
Surleraux DL, de Kock HA, Verschueren WG, Pille GM, Maes LJ, Peeters A, Vendeville S, De Meyer S, Azijn H, Pauwels R, de Bethune MP, King NM, Prabu-Jeyabalan M, Schiffer CA, Wigerinck PB.
Surleraux DL, et al. Among authors: pille gm.
J Med Chem. 2005 Mar 24;48(6):1965-73. doi: 10.1021/jm049454n.
J Med Chem. 2005.
PMID: 15771440
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1,5-Benzodiazepine inhibitors of HCV NS5B polymerase.
McGowan D, Nyanguile O, Cummings MD, Vendeville S, Vandyck K, Van den Broeck W, Boutton CW, De Bondt H, Quirynen L, Amssoms K, Bonfanti JF, Last S, Rombauts K, Tahri A, Hu L, Delouvroy F, Vermeiren K, Vandercruyssen G, Van der Helm L, Cleiren E, Mostmans W, Lory P, Pille G, Van Emelen K, Fanning G, Pauwels F, Lin TI, Simmen K, Raboisson P.
McGowan D, et al.
Bioorg Med Chem Lett. 2009 May 1;19(9):2492-6. doi: 10.1016/j.bmcl.2009.03.035. Epub 2009 Mar 14.
Bioorg Med Chem Lett. 2009.
PMID: 19342234
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2,4-Diaminoquinazolines as Dual Toll-like Receptor (TLR) 7/8 Modulators for the Treatment of Hepatitis B Virus.
Embrechts W, Herschke F, Pauwels F, Stoops B, Last S, Pieters S, Pande V, Pille G, Amssoms K, Smyej I, Dhuyvetter D, Scholliers A, Mostmans W, Van Dijck K, Van Schoubroeck B, Thone T, De Pooter D, Fanning G, Jonckers THM, Horton H, Raboisson P, McGowan D.
Embrechts W, et al.
J Med Chem. 2018 Jul 26;61(14):6236-6246. doi: 10.1021/acs.jmedchem.8b00643. Epub 2018 Jul 17.
J Med Chem. 2018.
PMID: 29965759
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Sustained release of the candidate antiretroviral peptides T-1249 and JNJ54310516-AFP from a rod insert vaginal ring.
Murphy DJ, Amssoms K, Pille G, Clarke A, O'Hara M, van Roey J, Malcolm RK.
Murphy DJ, et al.
Drug Deliv Transl Res. 2016 Jun;6(3):234-42. doi: 10.1007/s13346-015-0273-8.
Drug Deliv Transl Res. 2016.
PMID: 26787615
Free PMC article.
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