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5-Substituted Pyridine-2,4-dicarboxylate Derivatives Have Potential for Selective Inhibition of Human Jumonji-C Domain-Containing Protein 5.
J Med Chem. 2023 Aug 10;66(15):10849-10865. doi: 10.1021/acs.jmedchem.3c01114. Epub 2023 Aug 1.
J Med Chem. 2023.
PMID: 37527664
Free PMC article.
Arginase 1/2 Inhibitor OATD-02: From Discovery to First-in-man Setup in Cancer Immunotherapy.
Borek B, Nowicka J, Gzik A, Dziegielewski M, Jedrzejczak K, Brzezinska J, Grzybowski M, Stanczak P, Pomper P, Zagozdzon A, Rejczak T, Matyszewski K, Golebiowski A, Olczak J, Lisiecki K, Tyszkiewicz M, Kania M, Piasecka S, Cabaj A, Dera P, Mulewski K, Chrzanowski J, Kusmirek D, Sobolewska E, Magdycz M, Mucha L, Masnyk M, Golab J, Nowotny M, Nowak E, Napiorkowska-Gromadzka A, Pikul S, Jazwiec R, Dzwonek K, Dobrzanski P, Meyring M, Skowronek K, Iwanowski P, Zaslona Z, Blaszczyk R.
Borek B, et al. Among authors: piasecka s.
Mol Cancer Ther. 2023 Jul 5;22(7):807-817. doi: 10.1158/1535-7163.MCT-22-0721.
Mol Cancer Ther. 2023.
PMID: 36939275
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Impaired protein hydroxylase activity causes replication stress and developmental abnormalities in humans.
Fletcher SC, Hall C, Kennedy TJ, Pajusalu S, Wojcik MH, Boora U, Li C, Oja KT, Hendrix E, Westrip CA, Andrijes R, Piasecka SK, Singh M, El-Asrag ME, Ptasinska A, Tillmann V, Higgs MR, Carere DA, Beggs AD, Pappas J, Rabin R, Smerdon SJ, Stewart GS, Õunap K, Coleman ML.
Fletcher SC, et al. Among authors: piasecka sk.
J Clin Invest. 2023 Apr 3;133(7):e152784. doi: 10.1172/JCI152784.
J Clin Invest. 2023.
PMID: 36795492
Free PMC article.
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Discovery of OATD-01, a First-in-Class Chitinase Inhibitor as Potential New Therapeutics for Idiopathic Pulmonary Fibrosis.
Koralewski R, Dymek B, Mazur M, Sklepkiewicz P, Olejniczak S, Czestkowski W, Matyszewski K, Andryianau G, Niedziejko P, Kowalski M, Gruza M, Borek B, Jedrzejczak K, Bartoszewicz A, Pluta E, Rymaszewska A, Kania M, Rejczak T, Piasecka S, Mlacki M, Mazurkiewicz M, Piotrowicz M, Salamon M, Zagozdzon A, Napiorkowska-Gromadzka A, Bartlomiejczak A, Mozga W, Dobrzański P, Dzwonek K, Golab J, Nowotny M, Olczak J, Golebiowski A.
Koralewski R, et al. Among authors: piasecka s.
J Med Chem. 2020 Dec 24;63(24):15527-15540. doi: 10.1021/acs.jmedchem.0c01179. Epub 2020 Oct 20.
J Med Chem. 2020.
PMID: 33078933
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Building expanded structures from tetrahedral DNA branching elements, RNA and TMV protein.
Wenz NL, Piasecka S, Kalinowski M, Schneider A, Richert C, Wege C.
Wenz NL, et al. Among authors: piasecka s.
Nanoscale. 2018 Apr 5;10(14):6496-6510. doi: 10.1039/C7NR07743B.
Nanoscale. 2018.
PMID: 29569670
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Phosphoramidate Ligation of Oligonucleotides in Nanoscale Structures.
Kalinowski M, Haug R, Said H, Piasecka S, Kramer M, Richert C.
Kalinowski M, et al. Among authors: piasecka s.
Chembiochem. 2016 Jun 16;17(12):1150-5. doi: 10.1002/cbic.201600061. Epub 2016 May 25.
Chembiochem. 2016.
PMID: 27225865
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