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Rational Design of Bisubstrate-Type Analogues as Inhibitors of DNA Methyltransferases in Cancer Cells.
J Med Chem. 2017 Jun 8;60(11):4665-4679. doi: 10.1021/acs.jmedchem.7b00176. Epub 2017 May 23.
J Med Chem. 2017.
PMID: 28463515
Design and synthesis of new non nucleoside inhibitors of DNMT3A.
Erdmann A, Menon Y, Gros C, Molinier N, Novosad N, Samson A, Gregoire JM, Long C, Ausseil F, Halby L, Arimondo PB.
Erdmann A, et al. Among authors: novosad n.
Bioorg Med Chem. 2015 Sep 1;23(17):5946-53. doi: 10.1016/j.bmc.2015.06.066. Epub 2015 Jul 10.
Bioorg Med Chem. 2015.
PMID: 26220519
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Identification and optimization of hydrazone-gallate derivatives as specific inhibitors of DNA methyltransferase 3A.
Erdmann A, Menon Y, Gros C, Masson V, Aussagues Y, Ausseil F, Novosad N, Schambel P, Baltas M, Arimondo PB.
Erdmann A, et al. Among authors: novosad n.
Future Med Chem. 2016;8(4):373-80. doi: 10.4155/fmc.15.192. Epub 2016 Mar 15.
Future Med Chem. 2016.
PMID: 26976348
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Design, synthesis and biological evaluation of 4-amino-N- (4-aminophenyl)benzamide analogues of quinoline-based SGI-1027 as inhibitors of DNA methylation.
Rilova E, Erdmann A, Gros C, Masson V, Aussagues Y, Poughon-Cassabois V, Rajavelu A, Jeltsch A, Menon Y, Novosad N, Gregoire JM, Vispé S, Schambel P, Ausseil F, Sautel F, Arimondo PB, Cantagrel F.
Rilova E, et al. Among authors: novosad n.
ChemMedChem. 2014 Mar;9(3):590-601. doi: 10.1002/cmdc.201300420.
ChemMedChem. 2014.
PMID: 24678024
Free PMC article.
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Consequences of combining siRNA-mediated DNA methyltransferase 1 depletion with 5-aza-2'-deoxycytidine in human leukemic KG1 cells.
Vispé S, Deroide A, Davoine E, Desjobert C, Lestienne F, Fournier L, Novosad N, Bréand S, Besse J, Busato F, Tost J, De Vries L, Cussac D, Riond J, Arimondo PB.
Vispé S, et al. Among authors: novosad n.
Oncotarget. 2015 Jun 20;6(17):15265-82. doi: 10.18632/oncotarget.3317.
Oncotarget. 2015.
PMID: 25948775
Free PMC article.
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[The antimicrobial activity of thio-, thioxo- and oxo- derivatives of acridine].
Novosad NV.
Novosad NV.
Mikrobiol Z. 1996 Jul-Aug;58(4):55-8.
Mikrobiol Z. 1996.
PMID: 8991595
Russian.
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[Therapy of infected hematomas after trauma in hemophiliac patients].
Novosad NA, Kopystianskiĭ NR, Mel'nik AK, Loginskiĭ VE.
Novosad NA, et al.
Ortop Travmatol Protez. 1977 Nov;(11):50-3.
Ortop Travmatol Protez. 1977.
PMID: 609433
Russian.
No abstract available.
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[BLOOD COAGULATION SYSTEM AS A CLINICAL ASPECT OF THROMBOTIC COMPLICATIONS IN AMYLOID NEPHROSIS PATIENTS].
KOVALIV BM, NOVOSAD NA.
KOVALIV BM, et al. Among authors: novosad na.
Sov Med. 1964 Aug;27:21-5.
Sov Med. 1964.
PMID: 14239217
Russian.
No abstract available.
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