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Fusion with Promiscuous Gα16 Subunit Reveals Signaling Bias at Muscarinic Receptors.
Int J Mol Sci. 2021 Sep 18;22(18):10089. doi: 10.3390/ijms221810089.
Int J Mol Sci. 2021.
PMID: 34576254
Free PMC article.
Novel M2 -selective, Gi -biased agonists of muscarinic acetylcholine receptors.
Randáková A, Nelic D, Ungerová D, Nwokoye P, Su Q, Doležal V, El-Fakahany EE, Boulos J, Jakubík J.
Randáková A, et al. Among authors: nelic d.
Br J Pharmacol. 2020 May;177(9):2073-2089. doi: 10.1111/bph.14970. Epub 2020 Feb 15.
Br J Pharmacol. 2020.
PMID: 31910288
Free PMC article.
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Agonist-Specific Conformations of the M2 Muscarinic Acetylcholine Receptor Assessed by Molecular Dynamics.
Randáková A, Nelic D, Doležal V, El-Fakahany EE, Boulos J, Jakubík J.
Randáková A, et al. Among authors: nelic d.
J Chem Inf Model. 2020 Apr 27;60(4):2325-2338. doi: 10.1021/acs.jcim.0c00041. Epub 2020 Mar 13.
J Chem Inf Model. 2020.
PMID: 32130001
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Neuroactive steroids, WIN-compounds and cholesterol share a common binding site on muscarinic acetylcholine receptors.
Dolejší E, Chetverikov N, Szánti-Pintér E, Nelic D, Randáková A, Doležal V, El-Fakahany EE, Kudová E, Jakubík J.
Dolejší E, et al. Among authors: nelic d.
Biochem Pharmacol. 2021 Oct;192:114699. doi: 10.1016/j.bcp.2021.114699. Epub 2021 Jul 26.
Biochem Pharmacol. 2021.
PMID: 34324870
Free article.
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Neurosteroids and steroid hormones are allosteric modulators of muscarinic receptors.
Dolejší E, Szánti-Pintér E, Chetverikov N, Nelic D, Randáková A, Doležal V, Kudová E, Jakubík J.
Dolejší E, et al. Among authors: nelic d.
Neuropharmacology. 2021 Nov 1;199:108798. doi: 10.1016/j.neuropharm.2021.108798. Epub 2021 Sep 22.
Neuropharmacology. 2021.
PMID: 34555368
Free article.
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Guanidine Derivatives: How Simple Structural Modification of Histamine H3R Antagonists Has Led to the Discovery of Potent Muscarinic M2R/M4R Antagonists.
Staszewski M, Nelic D, Jończyk J, Dubiel M, Frank A, Stark H, Bajda M, Jakubik J, Walczyński K.
Staszewski M, et al. Among authors: nelic d.
ACS Chem Neurosci. 2021 Jul 7;12(13):2503-2519. doi: 10.1021/acschemneuro.1c00237. Epub 2021 Jun 8.
ACS Chem Neurosci. 2021.
PMID: 34100603
Free PMC article.
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Agonist-selective activation of individual G-proteins by muscarinic receptors.
Nelic D, Chetverikov N, Hochmalová M, Diaz C, Doležal V, Boulos J, Jakubík J, Martemyanov K, Janoušková-Randáková A.
Nelic D, et al.
Sci Rep. 2024 Apr 26;14(1):9652. doi: 10.1038/s41598-024-60259-4.
Sci Rep. 2024.
PMID: 38671143
Free PMC article.
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A critical re-evaluation of the slope factor of the operational model of agonism: When to exponentiate operational efficacy.
Randáková A, Nelic D, Jakubík J.
Randáková A, et al. Among authors: nelic d.
Sci Rep. 2023 Oct 16;13(1):17587. doi: 10.1038/s41598-023-45004-7.
Sci Rep. 2023.
PMID: 37845324
Free PMC article.
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