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Structural Investigations on Novel Non-Nucleoside Inhibitors of Human Norovirus Polymerase.
Viruses. 2022 Dec 27;15(1):74. doi: 10.3390/v15010074.
Viruses. 2022.
PMID: 36680114
Free PMC article.
Small Molecule Inhibitors of KDM5 Histone Demethylases Increase the Radiosensitivity of Breast Cancer Cells Overexpressing JARID1B.
Pippa S, Mannironi C, Licursi V, Bombardi L, Colotti G, Cundari E, Mollica A, Coluccia A, Naccarato V, La Regina G, Silvestri R, Negri R.
Pippa S, et al. Among authors: naccarato v.
Molecules. 2019 May 4;24(9):1739. doi: 10.3390/molecules24091739.
Molecules. 2019.
PMID: 31060229
Free PMC article.
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Drug Design and Synthesis of First in Class PDZ1 Targeting NHERF1 Inhibitors as Anticancer Agents.
Coluccia A, La Regina G, Naccarato V, Nalli M, Orlando V, Biagioni S, De Angelis ML, Baiocchi M, Gautier C, Gianni S, Di Pastena F, Di Magno L, Canettieri G, Coluccia AML, Silvestri R.
Coluccia A, et al. Among authors: naccarato v.
ACS Med Chem Lett. 2019 Jan 14;10(4):499-503. doi: 10.1021/acsmedchemlett.8b00532. eCollection 2019 Apr 11.
ACS Med Chem Lett. 2019.
PMID: 30996786
Free PMC article.
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Towards modern anticancer agents that interact with tubulin.
La Regina G, Coluccia A, Naccarato V, Silvestri R.
La Regina G, et al. Among authors: naccarato v.
Eur J Pharm Sci. 2019 Apr 1;131:58-68. doi: 10.1016/j.ejps.2019.01.028. Epub 2019 Jan 25.
Eur J Pharm Sci. 2019.
PMID: 30690185
Review.
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New 6- and 7-heterocyclyl-1H-indole derivatives as potent tubulin assembly and cancer cell growth inhibitors.
La Regina G, Bai R, Coluccia A, Naccarato V, Famiglini V, Nalli M, Masci D, Verrico A, Rovella P, Mazzoccoli C, Da Pozzo E, Cavallini C, Martini C, Vultaggio S, Dondio G, Varasi M, Mercurio C, Hamel E, Lavia P, Silvestri R.
La Regina G, et al. Among authors: naccarato v.
Eur J Med Chem. 2018 May 25;152:283-297. doi: 10.1016/j.ejmech.2018.04.042. Epub 2018 Apr 25.
Eur J Med Chem. 2018.
PMID: 29730191
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β-catenin knockdown promotes NHERF1-mediated survival of colorectal cancer cells: implications for a double-targeted therapy.
Saponaro C, Sergio S, Coluccia A, De Luca M, La Regina G, Mologni L, Famiglini V, Naccarato V, Bonetti D, Gautier C, Gianni S, Vergara D, Salzet M, Fournier I, Bucci C, Silvestri R, Passerini CG, Maffia M, Coluccia AML.
Saponaro C, et al. Among authors: naccarato v.
Oncogene. 2018 Jun;37(24):3301-3316. doi: 10.1038/s41388-018-0170-y. Epub 2018 Mar 19.
Oncogene. 2018.
PMID: 29551770
Free PMC article.
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3-Aroyl-1,4-diarylpyrroles Inhibit Chronic Myeloid Leukemia Cell Growth through an Interaction with Tubulin.
La Regina G, Bai R, Coluccia A, Famiglini V, Passacantilli S, Naccarato V, Ortar G, Mazzoccoli C, Ruggieri V, Agriesti F, Piccoli C, Tataranni T, Nalli M, Brancale A, Vultaggio S, Mercurio C, Varasi M, Saponaro C, Sergio S, Maffia M, Coluccia AML, Hamel E, Silvestri R.
La Regina G, et al. Among authors: naccarato v.
ACS Med Chem Lett. 2017 Apr 26;8(5):521-526. doi: 10.1021/acsmedchemlett.7b00022. eCollection 2017 May 11.
ACS Med Chem Lett. 2017.
PMID: 28523104
Free PMC article.
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