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Dual-Acting Small Molecules: Subtype-Selective Cannabinoid Receptor 2 Agonist/Butyrylcholinesterase Inhibitor Hybrids Show Neuroprotection in an Alzheimer's Disease Mouse Model.
J Med Chem. 2023 May 11;66(9):6414-6435. doi: 10.1021/acs.jmedchem.3c00541. Epub 2023 Apr 26.
J Med Chem. 2023.
PMID: 37127287
Free PMC article.
Convolamine, a tropane alkaloid extracted from Convolvulus plauricalis, is a potent sigma-1 receptor-positive modulator with cognitive and neuroprotective properties.
Crouzier L, Meunier J, Carles A, Morilleau A, Vrigneau C, Schmitt M, Bourguignon JJ, Delprat B, Maurice T.
Crouzier L, et al. Among authors: morilleau a.
Phytother Res. 2024 Feb;38(2):694-712. doi: 10.1002/ptr.8068. Epub 2023 Nov 27.
Phytother Res. 2024.
PMID: 38011416
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