Marco-Contelles J - Search Results

1

Exploring the Potential of Sulfonamide-Dihydropyridine Hybrids as Multitargeted Ligands for Alzheimer's Disease Treatment.

Dakhlaoui I, Bernard PJ, Pietrzak D, Simakov A, Maj M, Refouvelet B, Béduneau A, Cornu R, Jozwiak K, Chabchoub F, Iriepa I, Martin H, Marco-Contelles J, Ismaili L. Dakhlaoui I, et al. Among authors: marco contelles j. Int J Mol Sci. 2023 Jun 4;24(11):9742. doi: 10.3390/ijms24119742. Int J Mol Sci. 2023. PMID: 37298693 Free PMC article.

2

Novel multipotent tacrine-dihydropyridine hybrids with improved acetylcholinesterase inhibitory and neuroprotective activities as potential drugs for the treatment of Alzheimer's disease.

Marco-Contelles J, León R, de Los Ríos C, Guglietta A, Terencio J, López MG, García AG, Villarroya M. Marco-Contelles J, et al. J Med Chem. 2006 Dec 28;49(26):7607-10. doi: 10.1021/jm061047j. J Med Chem. 2006. PMID: 17181144

3

New tacrine-dihydropyridine hybrids that inhibit acetylcholinesterase, calcium entry, and exhibit neuroprotection properties.

León R, de los Ríos C, Marco-Contelles J, Huertas O, Barril X, Luque FJ, López MG, García AG, Villarroya M. León R, et al. Bioorg Med Chem. 2008 Aug 15;16(16):7759-69. doi: 10.1016/j.bmc.2008.07.005. Epub 2008 Jul 8. Bioorg Med Chem. 2008. PMID: 18640842

4

Tacripyrines, the first tacrine-dihydropyridine hybrids, as multitarget-directed ligands for the treatment of Alzheimer's disease.

Marco-Contelles J, León R, de los Ríos C, Samadi A, Bartolini M, Andrisano V, Huertas O, Barril X, Luque FJ, Rodríguez-Franco MI, López B, López MG, García AG, Carreiras Mdo C, Villarroya M. Marco-Contelles J, et al. J Med Chem. 2009 May 14;52(9):2724-32. doi: 10.1021/jm801292b. J Med Chem. 2009. PMID: 19374444

5

Synthesis, inhibitory activity of cholinesterases, and neuroprotective profile of novel 1,8-naphthyridine derivatives.

de Los Ríos C, Egea J, Marco-Contelles J, León R, Samadi A, Iriepa I, Moraleda I, Gálvez E, García AG, López MG, Villarroya M, Romero A. de Los Ríos C, et al. J Med Chem. 2010 Jul 22;53(14):5129-43. doi: 10.1021/jm901902w. J Med Chem. 2010. PMID: 20575555

6

Synthesis, biological assessment and molecular modeling of new dihydroquinoline-3-carboxamides and dihydroquinoline-3-carbohydrazide derivatives as cholinesterase inhibitors, and Ca channel antagonists.

Tomassoli I, Ismaili L, Pudlo M, de Los Ríos C, Soriano E, Colmena I, Gandía L, Rivas L, Samadi A, Marco-Contelles J, Refouvelet B. Tomassoli I, et al. Eur J Med Chem. 2011 Jan;46(1):1-10. doi: 10.1016/j.ejmech.2010.08.054. Epub 2010 Dec 15. Eur J Med Chem. 2011. PMID: 21111515

7

Synthesis, biological assessment and molecular modeling of 14-aryl-10,11,12,14-tetrahydro-9H-benzo[5,6]chromeno[2,3-b]quinolin-13-amines.

Maalej E, Chabchoub F, Samadi A, de los Ríos C, Perona A, Morreale A, Marco-Contelles J. Maalej E, et al. Bioorg Med Chem Lett. 2011 Apr 15;21(8):2384-8. doi: 10.1016/j.bmcl.2011.02.094. Epub 2011 Mar 14. Bioorg Med Chem Lett. 2011. PMID: 21411323

8

Synthesis, biological assessment and molecular modeling of new multipotent MAO and cholinesterase inhibitors as potential drugs for the treatment of Alzheimer's disease.

Samadi A, Chioua M, Bolea I, de Los Ríos C, Iriepa I, Moraleda I, Bastida A, Esteban G, Unzeta M, Gálvez E, Marco-Contelles J. Samadi A, et al. Eur J Med Chem. 2011 Sep;46(9):4665-8. doi: 10.1016/j.ejmech.2011.05.048. Epub 2011 May 26. Eur J Med Chem. 2011. PMID: 21669479

9

Chemical and pharmacological studies on enantiomerically pure p-methoxytacripyrines, promising multi-target-directed ligands for the treatment of Alzheimer's disease.

Bartolini M, Pistolozzi M, Andrisano V, Egea J, López MG, Iriepa I, Moraleda I, Gálvez E, Marco-Contelles J, Samadi A. Bartolini M, et al. ChemMedChem. 2011 Nov 4;6(11):1990-7. doi: 10.1002/cmdc.201100239. Epub 2011 Aug 24. ChemMedChem. 2011. PMID: 21990269 No abstract available.

10

Synthesis and biological assessment of diversely substituted furo[2,3-b]quinolin-4-amine and pyrrolo[2,3-b]quinolin-4-amine derivatives, as novel tacrine analogues.

Martins C, Carreiras MC, León R, de los Ríos C, Bartolini M, Andrisano V, Iriepa I, Moraleda I, Gálvez E, García M, Egea J, Samadi A, Chioua M, Marco-Contelles J. Martins C, et al. Eur J Med Chem. 2011 Dec;46(12):6119-30. doi: 10.1016/j.ejmech.2011.09.038. Epub 2011 Sep 29. Eur J Med Chem. 2011. PMID: 22000936

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