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Half-Sandwich Cyclopentadienylruthenium(II) Complexes: A New Antimalarial Chemotype.
Inorg Chem. 2020 Sep 8;59(17):12722-12732. doi: 10.1021/acs.inorgchem.0c01795. Epub 2020 Aug 24.
Inorg Chem. 2020.
PMID: 32838513
Identification of tetracyclic lactams as NMDA receptor antagonists with potential application in neurological disorders.
Espadinha M, Viejo L, Lopes RMRM, Herrera-Arozamena C, Molins E, Dos Santos DJVA, Gonçalves L, Rodríguez-Franco MI, Ríos CL, Santos MMM.
Espadinha M, et al. Among authors: lopes rmrm.
Eur J Med Chem. 2020 May 15;194:112242. doi: 10.1016/j.ejmech.2020.112242. Epub 2020 Mar 23.
Eur J Med Chem. 2020.
PMID: 32248004
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N,O-Iminoboronates: Reversible Iminoboronates with Improved Stability for Cancer Cells Targeted Delivery.
Lopes RMRM, Ventura AE, Silva LC, Faustino H, Gois PMP.
Lopes RMRM, et al.
Chemistry. 2018 Aug 27;24(48):12495-12499. doi: 10.1002/chem.201802515. Epub 2018 Jul 23.
Chemistry. 2018.
PMID: 29889332
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Diazaborines Are a Versatile Platform to Develop ROS-Responsive Antibody Drug Conjugates*.
António JPM, Carvalho JI, André AS, Dias JNR, Aguiar SI, Faustino H, Lopes RMRM, Veiros LF, Bernardes GJL, da Silva FA, Gois PMP.
António JPM, et al. Among authors: lopes rmrm.
Angew Chem Int Ed Engl. 2021 Dec 1;60(49):25914-25921. doi: 10.1002/anie.202109835. Epub 2021 Nov 5.
Angew Chem Int Ed Engl. 2021.
PMID: 34741376
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Selective Inhibition of Bruton's Tyrosine Kinase by a Designed Covalent Ligand Leads to Potent Therapeutic Efficacy in Blood Cancers Relative to Clinically Used Inhibitors.
Sousa BB, de Almeida CR, Barahona AF, Lopes R, Martins-Logrado A, Cavaco M, Neves V, Carvalho LAR, Labão-Almeida C, Coelho AR, Leal Bento M, Lopes RMRM, Oliveira BL, Castanho MARB, Neumeister P, Deutsch A, Vladimer GI, Krall N, João C, Corzana F, Seixas JD, Fior R, Bernardes GJL.
Sousa BB, et al. Among authors: lopes rmrm.
ACS Pharmacol Transl Sci. 2022 Nov 2;5(11):1156-1168. doi: 10.1021/acsptsci.2c00163. eCollection 2022 Nov 11.
ACS Pharmacol Transl Sci. 2022.
PMID: 36407952
Free PMC article.
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