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Combretastatin A-4 sulfur-containing heterocyclic derivatives: Synthesis, antiproliferative activities and molecular docking studies.
Faouzi A, Arnaud A, Bancet A, Barette C, Preto J, Do CV, Jordheim LP, Bousfiha Z, Nguyen TTB, Verrière M, Farce A, Fauvarque MO, Barret R, Lomberget T. Faouzi A, et al. Among authors: lomberget t. Eur J Med Chem. 2021 Apr 5;215:113275. doi: 10.1016/j.ejmech.2021.113275. Epub 2021 Feb 8. Eur J Med Chem. 2021. PMID: 33618157
Synthesis and biological evaluation of thiophene and benzo[b]thiophene analogs of combretastatin A-4 and isocombretastatin A-4: A comparison between the linkage positions of the 3,4,5-trimethoxystyrene unit.
Do CV, Faouzi A, Barette C, Farce A, Fauvarque MO, Colomb E, Catry L, Berthier-Vergnes O, Haftek M, Barret R, Lomberget T. Do CV, et al. Among authors: lomberget t. Bioorg Med Chem Lett. 2016 Jan 1;26(1):174-80. doi: 10.1016/j.bmcl.2015.11.010. Epub 2015 Nov 10. Bioorg Med Chem Lett. 2016. PMID: 26602281
Fragment Linking Strategies for Structure-Based Drug Design.
Bancet A, Raingeval C, Lomberget T, Le Borgne M, Guichou JF, Krimm I. Bancet A, et al. Among authors: lomberget t. J Med Chem. 2020 Oct 22;63(20):11420-11435. doi: 10.1021/acs.jmedchem.0c00242. Epub 2020 Jun 23. J Med Chem. 2020. PMID: 32539387 Review.
Synthesis of new steroidal inhibitors of P-glycoprotein-mediated multidrug resistance and biological evaluation on K562/R7 erythroleukemia cells.
de Ravel MR, Alameh G, Melikian M, Mahiout Z, Emptoz-Bonneton A, Matera EL, Lomberget T, Barret R, Rocheblave L, Walchshofer N, Beltran S, El Jawad L, Mappus E, Grenot C, Pugeat M, Dumontet C, Le Borgne M, Cuilleron CY. de Ravel MR, et al. Among authors: lomberget t. J Med Chem. 2015 Feb 26;58(4):1832-45. doi: 10.1021/jm501676v. Epub 2015 Feb 11. J Med Chem. 2015. PMID: 25634041
2-Aminothiazole Derivatives as Selective Allosteric Modulators of the Protein Kinase CK2. 2. Structure-Based Optimization and Investigation of Effects Specific to the Allosteric Mode of Action.
Bestgen B, Kufareva I, Seetoh W, Abell C, Hartmann RW, Abagyan R, Le Borgne M, Filhol O, Cochet C, Lomberget T, Engel M. Bestgen B, et al. Among authors: lomberget t. J Med Chem. 2019 Feb 28;62(4):1817-1836. doi: 10.1021/acs.jmedchem.8b01765. Epub 2019 Feb 13. J Med Chem. 2019. PMID: 30689946 Free PMC article.
2-Aminothiazole Derivatives as Selective Allosteric Modulators of the Protein Kinase CK2. 1. Identification of an Allosteric Binding Site.
Bestgen B, Krimm I, Kufareva I, Kamal AAM, Seetoh WG, Abell C, Hartmann RW, Abagyan R, Cochet C, Le Borgne M, Engel M, Lomberget T. Bestgen B, et al. Among authors: lomberget t. J Med Chem. 2019 Feb 28;62(4):1803-1816. doi: 10.1021/acs.jmedchem.8b01766. Epub 2019 Feb 18. J Med Chem. 2019. PMID: 30689953 Free PMC article.
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