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Indoloxytriazines as binding molecules for the JAK2 JH2 pseudokinase domain and its V617F variant.
Tetrahedron Lett. 2021 Aug 3;77:153248. doi: 10.1016/j.tetlet.2021.153248. Epub 2021 Jul 2.
Tetrahedron Lett. 2021.
PMID: 34393283
Free PMC article.
Selective Janus Kinase 2 (JAK2) Pseudokinase Ligands with a Diaminotriazole Core.
Liosi ME, Krimmer SG, Newton AS, Dawson TK, Puleo DE, Cutrona KJ, Suzuki Y, Schlessinger J, Jorgensen WL.
Liosi ME, et al.
J Med Chem. 2020 May 28;63(10):5324-5340. doi: 10.1021/acs.jmedchem.0c00192. Epub 2020 May 8.
J Med Chem. 2020.
PMID: 32329617
Free PMC article.
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Identification of 14 Known Drugs as Inhibitors of the Main Protease of SARS-CoV-2.
Ghahremanpour MM, Tirado-Rives J, Deshmukh M, Ippolito JA, Zhang CH, de Vaca IC, Liosi ME, Anderson KS, Jorgensen WL.
Ghahremanpour MM, et al. Among authors: liosi me.
bioRxiv [Preprint]. 2020 Aug 28:2020.08.28.271957. doi: 10.1101/2020.08.28.271957.
bioRxiv. 2020.
PMID: 32869018
Free PMC article.
Updated.
Preprint.
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Identification of 14 Known Drugs as Inhibitors of the Main Protease of SARS-CoV-2.
Ghahremanpour MM, Tirado-Rives J, Deshmukh M, Ippolito JA, Zhang CH, Cabeza de Vaca I, Liosi ME, Anderson KS, Jorgensen WL.
Ghahremanpour MM, et al. Among authors: liosi me.
ACS Med Chem Lett. 2020 Oct 25;11(12):2526-2533. doi: 10.1021/acsmedchemlett.0c00521. eCollection 2020 Dec 10.
ACS Med Chem Lett. 2020.
PMID: 33324471
Free PMC article.
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Optimization of Triarylpyridinone Inhibitors of the Main Protease of SARS-CoV-2 to Low-Nanomolar Antiviral Potency.
Zhang CH, Spasov KA, Reilly RA, Hollander K, Stone EA, Ippolito JA, Liosi ME, Deshmukh MG, Tirado-Rives J, Zhang S, Liang Z, Miller SJ, Isaacs F, Lindenbach BD, Anderson KS, Jorgensen WL.
Zhang CH, et al. Among authors: liosi me.
ACS Med Chem Lett. 2021 Jul 14;12(8):1325-1332. doi: 10.1021/acsmedchemlett.1c00326. eCollection 2021 Aug 12.
ACS Med Chem Lett. 2021.
PMID: 34408808
Free PMC article.
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Conversion of a False Virtual Screen Hit into Selective JAK2 JH2 Domain Binders Using Convergent Design Strategies.
Henry SP, Liosi ME, Ippolito JA, Cutrona KJ, Krimmer SG, Newton AS, Schlessinger J, Jorgensen WL.
Henry SP, et al. Among authors: liosi me.
ACS Med Chem Lett. 2022 Apr 21;13(5):819-826. doi: 10.1021/acsmedchemlett.2c00051. eCollection 2022 May 12.
ACS Med Chem Lett. 2022.
PMID: 35586418
Free PMC article.
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Insights on JAK2 Modulation by Potent, Selective, and Cell-Permeable Pseudokinase-Domain Ligands.
Liosi ME, Ippolito JA, Henry SP, Krimmer SG, Newton AS, Cutrona KJ, Olivarez RA, Mohanty J, Schlessinger J, Jorgensen WL.
Liosi ME, et al.
J Med Chem. 2022 Jun 23;65(12):8380-8400. doi: 10.1021/acs.jmedchem.2c00283. Epub 2022 Jun 2.
J Med Chem. 2022.
PMID: 35653642
Free PMC article.
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Covalent Modification of the JH2 Domain of Janus Kinase 2.
Henry SP, Liosi ME, Ippolito JA, Menges F, Newton AS, Schlessinger J, Jorgensen WL.
Henry SP, et al. Among authors: liosi me.
ACS Med Chem Lett. 2022 Oct 24;13(11):1819-1826. doi: 10.1021/acsmedchemlett.2c00414. eCollection 2022 Nov 10.
ACS Med Chem Lett. 2022.
PMID: 36385940
Free PMC article.
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