Laura H. Heitman - Search Results

Year	Number of Results
2006	1
2007	2
2008	5
2009	3
2012	6
2013	5
2014	8
2015	14
2016	13
2017	16
2018	16
2019	10
2020	10
2021	14
2022	13
2023	12
2024	5

1

Pharmacological characterization of allosteric modulators: A case for chemokine receptors.

den Hollander LS, IJzerman AP, Heitman LH. den Hollander LS, et al. Among authors: heitman lh. Med Res Rev. 2024 Apr 18. doi: 10.1002/med.22043. Online ahead of print. Med Res Rev. 2024. PMID: 38634664 Review.

2

Computational Characterization of Membrane Proteins as Anticancer Targets: Current Challenges and Opportunities.

Gorostiola González M, Rakers PRJ, Jespers W, IJzerman AP, Heitman LH, van Westen GJP. Gorostiola González M, et al. Among authors: heitman lh. Int J Mol Sci. 2024 Mar 26;25(7):3698. doi: 10.3390/ijms25073698. Int J Mol Sci. 2024. PMID: 38612509 Free PMC article. Review.

3

Still in Search for an EAAT Activator: GT949 Does Not Activate EAAT2, nor EAAT3 in Impedance and Radioligand Uptake Assays.

van Veggel L, Mocking TAM, Sijben HJ, Liu R, Gorostiola González M, Dilweg MA, Royakkers J, Li A, Kumar V, Dong YY, Bullock A, Sauer DB, Diliën H, van Westen GJP, Schreiber R, Heitman LH, Vanmierlo T. van Veggel L, et al. Among authors: heitman lh. ACS Chem Neurosci. 2024 Apr 3;15(7):1424-1431. doi: 10.1021/acschemneuro.3c00731. Epub 2024 Mar 13. ACS Chem Neurosci. 2024. PMID: 38478848 Free PMC article.

4

Discovery of a Photoaffinity Probe that Captures the Active Conformation of the Cannabinoid CB₂ Receptor.

De Paus LV, An Y, Janssen APA, van den Berg RJBHN, Heitman LH, van der Stelt M. De Paus LV, et al. Among authors: heitman lh. Chembiochem. 2024 Apr 2;25(7):e202300785. doi: 10.1002/cbic.202300785. Epub 2024 Mar 1. Chembiochem. 2024. PMID: 38372466

5

Molecular insights into disease-associated glutamate transporter (EAAT1 / SLC1A3) variants using in silico and in vitro approaches.

Gorostiola González M, Sijben HJ, Dall' Acqua L, Liu R, IJzerman AP, Heitman LH, van Westen GJP. Gorostiola González M, et al. Among authors: heitman lh. Front Mol Biosci. 2023 Nov 23;10:1286673. doi: 10.3389/fmolb.2023.1286673. eCollection 2023. Front Mol Biosci. 2023. PMID: 38074092 Free PMC article.

6

A monoacylglycerol lipase inhibitor showing therapeutic efficacy in mice without central side effects or dependence.

Jiang M, Huizenga MCW, Wirt JL, Paloczi J, Amedi A, van den Berg RJBHN, Benz J, Collin L, Deng H, Di X, Driever WF, Florea BI, Grether U, Janssen APA, Hankemeier T, Heitman LH, Lam TW, Mohr F, Pavlovic A, Ruf I, van den Hurk H, Stevens AF, van der Vliet D, van der Wel T, Wittwer MB, van Boeckel CAA, Pacher P, Hohmann AG, van der Stelt M. Jiang M, et al. Among authors: heitman lh. Nat Commun. 2023 Dec 5;14(1):8039. doi: 10.1038/s41467-023-43606-3. Nat Commun. 2023. PMID: 38052772 Free PMC article.

7

Dual allosteric and orthosteric pharmacology of synthetic analog cannabidiol-dimethylheptyl, but not cannabidiol, on the cannabinoid CB₂ receptor.

Bouma J, Broekhuis JD, van der Horst C, Kumar P, Ligresti A, van der Stelt M, Heitman LH. Bouma J, et al. Among authors: heitman lh. Biochem Pharmacol. 2023 Dec;218:115924. doi: 10.1016/j.bcp.2023.115924. Epub 2023 Nov 14. Biochem Pharmacol. 2023. PMID: 37972874 Free article.

8

The 17^th EFMC Short Course on Medicinal Chemistry on Small Molecule Protein Degraders.

Ciulli A, O'Connor S, Chung CW, Hartung IV, Testa A, Daniels DL, Heitman LH. Ciulli A, et al. Among authors: heitman lh. ChemMedChem. 2023 Oct 17;18(20):e202300464. doi: 10.1002/cmdc.202300464. Epub 2023 Oct 10. ChemMedChem. 2023. PMID: 37817354

9

3DDPDs: describing protein dynamics for proteochemometric bioactivity prediction. A case for (mutant) G protein-coupled receptors.

Gorostiola González M, van den Broek RL, Braun TGM, Chatzopoulou M, Jespers W, IJzerman AP, Heitman LH, van Westen GJP. Gorostiola González M, et al. Among authors: heitman lh. J Cheminform. 2023 Aug 28;15(1):74. doi: 10.1186/s13321-023-00745-5. J Cheminform. 2023. PMID: 37641107 Free PMC article.

10

Development of an Affinity-Based Probe to Profile Endogenous Human Adenosine A₃ Receptor Expression.

Beerkens BLH, Snijders IM, Snoeck J, Liu R, Tool ATJ, Le Dévédec SE, Jespers W, Kuijpers TW, van Westen GJP, Heitman LH, IJzerman AP, van der Es D. Beerkens BLH, et al. Among authors: heitman lh. J Med Chem. 2023 Aug 24;66(16):11399-11413. doi: 10.1021/acs.jmedchem.3c00854. Epub 2023 Aug 2. J Med Chem. 2023. PMID: 37531576 Free PMC article.

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Results by year

Text availability

Article attribute

Article type

Publication date

134 results

Results by year

Search Page

Filters

My NCBI Filters

Results by year

Text availability

Article attribute

Article type

Publication date

Search Results

134 results

Results by year