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β-Glucuronidase triggers extracellular MMAE release from an integrin-targeted conjugate.
Org Biomol Chem. 2019 May 15;17(19):4705-4710. doi: 10.1039/c9ob00617f.
Org Biomol Chem. 2019.
PMID: 31020985
Free article.
Tumor Targeting with an isoDGR-Drug Conjugate.
Zanella S, Angerani S, Pina A, López Rivas P, Giannini C, Panzeri S, Arosio D, Caruso M, Gasparri F, Fraietta I, Albanese C, Marsiglio A, Pignataro L, Belvisi L, Piarulli U, Gennari C.
Zanella S, et al. Among authors: lopez rivas p.
Chemistry. 2017 Jun 12;23(33):7910-7914. doi: 10.1002/chem.201701844. Epub 2017 May 26.
Chemistry. 2017.
PMID: 28449309
Free PMC article.
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Synthesis and biological evaluation of RGD and isoDGR peptidomimetic-α-amanitin conjugates for tumor-targeting.
Bodero L, López Rivas P, Korsak B, Hechler T, Pahl A, Müller C, Arosio D, Pignataro L, Gennari C, Piarulli U.
Bodero L, et al. Among authors: lopez rivas p.
Beilstein J Org Chem. 2018 Feb 14;14:407-415. doi: 10.3762/bjoc.14.29. eCollection 2018.
Beilstein J Org Chem. 2018.
PMID: 29520305
Free PMC article.
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Conjugates of Cryptophycin and RGD or isoDGR Peptidomimetics for Targeted Drug Delivery.
Borbély A, Figueras E, Martins A, Bodero L, Raposo Moreira Dias A, López Rivas P, Pina A, Arosio D, Gallinari P, Frese M, Steinkühler C, Gennari C, Piarulli U, Sewald N.
Borbély A, et al. Among authors: lopez rivas p.
ChemistryOpen. 2019 Jun 7;8(6):737-742. doi: 10.1002/open.201900110. eCollection 2019 Jun.
ChemistryOpen. 2019.
PMID: 31275795
Free PMC article.
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