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Ultrasound assisted one-pot synthesis of rosuvastatin based novel azaindole derivatives via coupling-cyclization strategy under Pd/Cu-catalysis: Their evaluation as potential cytotoxic agents.
Kumar JS, Reddy GS, Medishetti R, Amirul Hossain K, Thirupataiah B, Edelli J, Dilip Bele S, Kristina Edwin R, Joseph A, Shenoy GG, Mallikarjuna Rao C, Pal M. Kumar JS, et al. Bioorg Chem. 2022 Jul;124:105857. doi: 10.1016/j.bioorg.2022.105857. Epub 2022 May 10. Bioorg Chem. 2022. PMID: 35594765
Synthesis of 11,12-dihydro benzo[c]phenanthridines via a Pd-catalyzed unusual construction of isocoumarin ring/FeCl3-mediated intramolecular arene-allyl cyclization: First identification of a benzo[c]phenanthridine based PDE4 inhibitor.
Thirupataiah B, Reddy GS, Ghule SS, Kumar JS, Mounika G, Hossain KA, Mudgal J, Mathew JE, Shenoy GG, Parsa KVL, Pal M. Thirupataiah B, et al. Among authors: kumar js. Bioorg Chem. 2020 Apr;97:103691. doi: 10.1016/j.bioorg.2020.103691. Epub 2020 Feb 25. Bioorg Chem. 2020. PMID: 32143019
PdCl2-catalyzed synthesis of a new class of isocoumarin derivatives containing aminosulfonyl / aminocarboxamide moiety: First identification of a isocoumarin based PDE4 inhibitor.
Thirupataiah B, Mounika G, Reddy GS, Kumar JS, Hossain KA, Medishetti R, Samarpita S, Rasool M, Mudgal J, Mathew JE, Shenoy GG, Rao CM, Chatti K, Parsa KVL, Pal M. Thirupataiah B, et al. Among authors: kumar js. Eur J Med Chem. 2021 Oct 5;221:113514. doi: 10.1016/j.ejmech.2021.113514. Epub 2021 May 6. Eur J Med Chem. 2021. PMID: 33992926
Fe(III)-catalyzed regioselective and faster synthesis of isocoumarins with 3-oxoalkyl moiety at C-4: Identification of new inhibitors of PDE4.
Thirupataiah B, Bhuktar H, Mounika G, Reddy GS, Kumar JS, Shukla S, Hossain KA, Medishetti R, Samarpita S, Rasool M, Jagadish PC, Shenoy GG, Parsa KVL, Pal M. Thirupataiah B, et al. Among authors: kumar js. Bioorg Chem. 2022 Apr;121:105667. doi: 10.1016/j.bioorg.2022.105667. Epub 2022 Feb 9. Bioorg Chem. 2022. PMID: 35182886
InCl3 mediated heteroarylation of indoles and their derivatization via CH activation strategy: Discovery of 2-(1H-indol-3-yl)-quinoxaline derivatives as a new class of PDE4B selective inhibitors for arthritis and/or multiple sclerosis.
Sunke R, Bankala R, Thirupataiah B, Ramarao EVVS, Kumar JS, Doss HM, Medishetti R, Kulkarni P, Kapavarapu RK, Rasool M, Mudgal J, Mathew JE, Shenoy GG, Parsa KVL, Pal M. Sunke R, et al. Among authors: kumar js. Eur J Med Chem. 2019 Jul 15;174:198-215. doi: 10.1016/j.ejmech.2019.04.020. Epub 2019 Apr 16. Eur J Med Chem. 2019. PMID: 31035240
Novel isatin-indole derivatives as potential inhibitors of chorismate mutase (CM): their synthesis along with unexpected formation of 2-indolylmethylamino benzoate ester under Pd-Cu catalysis.
Reddy GS, Hossain KA, Kumar JS, Thirupataiah B, Edwin RK, Giliyaru VB, Chandrashekhar Hariharapura R, Shenoy GG, Misra P, Pal M. Reddy GS, et al. Among authors: kumar js. RSC Adv. 2020 Jan 2;10(1):289-297. doi: 10.1039/c9ra09236f. eCollection 2019 Dec 20. RSC Adv. 2020. PMID: 35492515 Free PMC article.
178 results