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The pharmacology of tacrine at N-methyl-d-aspartate receptors.
Horak M, Holubova K, Nepovimova E, Krusek J, Kaniakova M, Korabecny J, Vyklicky L, Kuca K, Stuchlik A, Ricny J, Vales K, Soukup O. Horak M, et al. Among authors: krusek j. Prog Neuropsychopharmacol Biol Psychiatry. 2017 Apr 3;75:54-62. doi: 10.1016/j.pnpbp.2017.01.003. Epub 2017 Jan 13. Prog Neuropsychopharmacol Biol Psychiatry. 2017. PMID: 28089695 Review.
A resurrection of 7-MEOTA: a comparison with tacrine.
Soukup O, Jun D, Zdarova-Karasova J, Patocka J, Musilek K, Korabecny J, Krusek J, Kaniakova M, Sepsova V, Mandikova J, Trejtnar F, Pohanka M, Drtinova L, Pavlik M, Tobin G, Kuca K. Soukup O, et al. Among authors: krusek j. Curr Alzheimer Res. 2013 Oct;10(8):893-906. doi: 10.2174/1567205011310080011. Curr Alzheimer Res. 2013. PMID: 24093535
7-Methoxyderivative of tacrine is a 'foot-in-the-door' open-channel blocker of GluN1/GluN2 and GluN1/GluN3 NMDA receptors with neuroprotective activity in vivo.
Kaniakova M, Kleteckova L, Lichnerova K, Holubova K, Skrenkova K, Korinek M, Krusek J, Smejkalova T, Korabecny J, Vales K, Soukup O, Horak M. Kaniakova M, et al. Among authors: krusek j. Neuropharmacology. 2018 Sep 15;140:217-232. doi: 10.1016/j.neuropharm.2018.08.010. Epub 2018 Aug 9. Neuropharmacology. 2018. PMID: 30099049
Cholesterol modulates open probability and desensitization of NMDA receptors.
Korinek M, Vyklicky V, Borovska J, Lichnerova K, Kaniakova M, Krausova B, Krusek J, Balik A, Smejkalova T, Horak M, Vyklicky L. Korinek M, et al. Among authors: krusek j. J Physiol. 2015 May 15;593(10):2279-93. doi: 10.1113/jphysiol.2014.288209. Epub 2015 Mar 24. J Physiol. 2015. PMID: 25651798 Free PMC article.
Structure, function, and pharmacology of NMDA receptor channels.
Vyklicky V, Korinek M, Smejkalova T, Balik A, Krausova B, Kaniakova M, Lichnerova K, Cerny J, Krusek J, Dittert I, Horak M, Vyklicky L. Vyklicky V, et al. Among authors: krusek j. Physiol Res. 2014;63(Suppl 1):S191-203. doi: 10.33549/physiolres.932678. Physiol Res. 2014. PMID: 24564659 Free article. Review.
Dual effect of lobeline on α4β2 rat neuronal nicotinic receptors.
Kaniaková M, Lindovský J, Krůšek J, Adámek S, Vyskočil F. Kaniaková M, et al. Among authors: krusek j. Eur J Pharmacol. 2011 May 11;658(2-3):108-13. doi: 10.1016/j.ejphar.2011.02.012. Epub 2011 Mar 1. Eur J Pharmacol. 2011. PMID: 21371469
50 results