Krasavin M - Search Results

1

Panel docking of small-molecule libraries - Prospects to improve efficiency of lead compound discovery.

Sarnpitak P, Mujumdar P, Taylor P, Cross M, Coster MJ, Gorse AD, Krasavin M, Hofmann A. Sarnpitak P, et al. Among authors: krasavin m. Biotechnol Adv. 2015 Nov 1;33(6 Pt 1):941-7. doi: 10.1016/j.biotechadv.2015.05.006. Epub 2015 May 27. Biotechnol Adv. 2015. PMID: 26025037 Free article. Review.

2

Potent, orally available, selective COX-2 inhibitors based on 2-imidazoline core.

Sarnpitak P, Mujumdar P, Morisseau C, Hwang SH, Hammock B, Iurchenko V, Zozulya S, Gavalas A, Geronikaki A, Ivanenkov Y, Krasavin M. Sarnpitak P, et al. Among authors: krasavin m. Eur J Med Chem. 2014 Sep 12;84:160-72. doi: 10.1016/j.ejmech.2014.07.023. Epub 2014 Jul 8. Eur J Med Chem. 2014. PMID: 25016374

3

Library of diversely substituted 2-(quinolin-4-yl)imidazolines delivers novel non-cytotoxic antitubercular leads.

Krasavin M, Mujumdar P, Parchinsky V, Vinogradova T, Manicheva O, Dogonadze M. Krasavin M, et al. J Enzyme Inhib Med Chem. 2016 Dec;31(6):1146-55. doi: 10.3109/14756366.2015.1101094. Epub 2015 Nov 2. J Enzyme Inhib Med Chem. 2016. PMID: 26526717

4

Isoform-selective inhibitory profile of 2-imidazoline-substituted benzene sulfonamides against a panel of human carbonic anhydrases.

Supuran CT, Kalinin S, Tanç M, Sarnpitak P, Mujumdar P, Poulsen SA, Krasavin M. Supuran CT, et al. Among authors: krasavin m. J Enzyme Inhib Med Chem. 2016;31(sup1):197-202. doi: 10.1080/14756366.2016.1178248. Epub 2016 May 10. J Enzyme Inhib Med Chem. 2016. PMID: 27160030

5

Design, in silico prioritization and biological profiling of apoptosis-inducing lactams amenable by the Castagnoli-Cushman reaction.

Krasavin M, Gureyev MA, Dar'in D, Bakulina O, Chizhova M, Lepikhina A, Novikova D, Grigoreva T, Ivanov G, Zhumagalieva A, Garabadzhiu AV, Tribulovich VG. Krasavin M, et al. Bioorg Med Chem. 2018 May 15;26(9):2651-2673. doi: 10.1016/j.bmc.2018.04.036. Epub 2018 Apr 18. Bioorg Med Chem. 2018. PMID: 29691156

6

Novel free fatty acid receptor 1 (GPR40) agonists based on 1,3,4-thiadiazole-2-carboxamide scaffold.

Krasavin M, Lukin A, Zhurilo N, Kovalenko A, Zahanich I, Zozulya S, Moore D, Tikhonova IG. Krasavin M, et al. Bioorg Med Chem. 2016 Jul 1;24(13):2954-2963. doi: 10.1016/j.bmc.2016.04.065. Epub 2016 May 5. Bioorg Med Chem. 2016. PMID: 27229618

7

Continued SAR exploration of 1,2,4-thiadiazole-containing scaffolds in the design of free fatty acid receptor 1 (GPR40) agonists.

Krasavin M, Lukin A, Bakholdina A, Zhurilo N, Onopchenko O, Borysko P, Zozulya S, Moore D, Tikhonova IG. Krasavin M, et al. Eur J Med Chem. 2017 Nov 10;140:229-238. doi: 10.1016/j.ejmech.2017.09.019. Epub 2017 Sep 13. Eur J Med Chem. 2017. PMID: 28938138

8

Heterocyclic periphery in the design of carbonic anhydrase inhibitors: 1,2,4-Oxadiazol-5-yl benzenesulfonamides as potent and selective inhibitors of cytosolic hCA II and membrane-bound hCA IX isoforms.

Krasavin M, Shetnev A, Sharonova T, Baykov S, Tuccinardi T, Kalinin S, Angeli A, Supuran CT. Krasavin M, et al. Bioorg Chem. 2018 Feb;76:88-97. doi: 10.1016/j.bioorg.2017.10.005. Epub 2017 Oct 16. Bioorg Chem. 2018. PMID: 29153590

9

Non-chelating p-phenylidene-linked bis-imidazoline analogs of known influenza virus endonuclease inhibitors: Synthesis and anti-influenza activity.

Dar'in D, Zarubaev V, Galochkina A, Gureev M, Krasavin M. Dar'in D, et al. Among authors: krasavin m. Eur J Med Chem. 2019 Jan 1;161:526-532. doi: 10.1016/j.ejmech.2018.10.063. Epub 2018 Oct 29. Eur J Med Chem. 2019. PMID: 30390440

10

Novel electrophilic amides amenable by the Ugi reaction perturb thioredoxin system via thioredoxin reductase 1 (TrxR1) inhibition: Identification of DVD-445 as a new lead compound for anticancer therapy.

Jovanović M, Zhukovsky D, Podolski-Renić A, Domračeva I, Žalubovskis R, Senćanski M, Glišić S, Sharoyko V, Tennikova T, Dar'in D, Pešić M, Krasavin M. Jovanović M, et al. Among authors: krasavin m. Eur J Med Chem. 2019 Nov 1;181:111580. doi: 10.1016/j.ejmech.2019.111580. Epub 2019 Aug 1. Eur J Med Chem. 2019. PMID: 31400708

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