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Intratumoral delivery of TransCon™ TLR7/8 Agonist promotes sustained anti-tumor activity and local immune cell activation while minimizing systemic cytokine induction.
Cancer Cell Int. 2022 Sep 19;22(1):286. doi: 10.1186/s12935-022-02708-6.
Cancer Cell Int. 2022.
PMID: 36123697
Free PMC article.
Degradable Hydrogel for Sustained Localized Delivery of Anti-Tumor Drugs.
Lessmann T, Jones SA, Voigt T, Weisbrod S, Kracker O, Winter S, Zúñiga LA, Stark S, Bisek N, Sprogøe K.
Lessmann T, et al. Among authors: kracker o.
J Pharm Sci. 2023 Nov;112(11):2843-2852. doi: 10.1016/j.xphs.2023.05.018. Epub 2023 Jun 4.
J Pharm Sci. 2023.
PMID: 37279836
Free article.
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Peptidotriazolamers Inhibit Aβ(1-42) Oligomerization and Cross a Blood-Brain-Barrier Model.
Tonali N, Hericks L, Schröder DC, Kracker O, Krzemieniecki R, Kaffy J, Le Joncour V, Laakkonen P, Marion A, Ongeri S, Dodero VI, Sewald N.
Tonali N, et al. Among authors: kracker o.
Chempluschem. 2021 Jun;86(6):840-851. doi: 10.1002/cplu.202000814. Epub 2021 May 6.
Chempluschem. 2021.
PMID: 33905181
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1,4-Disubstituted 1H-1,2,3-Triazole Containing Peptidotriazolamers: A New Class of Peptidomimetics With Interesting Foldamer Properties.
Schröder DC, Kracker O, Fröhr T, Góra J, Jewginski M, Nieß A, Antes I, Latajka R, Marion A, Sewald N.
Schröder DC, et al. Among authors: kracker o.
Front Chem. 2019 Mar 26;7:155. doi: 10.3389/fchem.2019.00155. eCollection 2019.
Front Chem. 2019.
PMID: 30972322
Free PMC article.
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1,5-Disubstituted 1,2,3-Triazole-Containing Peptidotriazolamers: Design Principles for a Class of Versatile Peptidomimetics.
Kracker O, Góra J, Krzciuk-Gula J, Marion A, Neumann B, Stammler HG, Nieß A, Antes I, Latajka R, Sewald N.
Kracker O, et al.
Chemistry. 2018 Jan 19;24(4):953-961. doi: 10.1002/chem.201704583. Epub 2017 Dec 13.
Chemistry. 2018.
PMID: 29160605
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Amber-Compatible Parametrization Procedure for Peptide-like Compounds: Application to 1,4- and 1,5-Substituted Triazole-Based Peptidomimetics.
Marion A, Góra J, Kracker O, Fröhr T, Latajka R, Sewald N, Antes I.
Marion A, et al. Among authors: kracker o.
J Chem Inf Model. 2018 Jan 22;58(1):90-110. doi: 10.1021/acs.jcim.7b00305. Epub 2017 Dec 21.
J Chem Inf Model. 2018.
PMID: 29112399
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