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Page 1
Indole-2-carboxamides as novel NR2B selective NMDA receptor antagonists.
Borza I, Kolok S, Gere A, Agai-Csongor E, Agai B, Tárkányi G, Horváth C, Barta-Szalai G, Bozó E, Kiss C, Bielik A, Nagy J, Farkas S, Domány G. Borza I, et al. Among authors: kolok s. Bioorg Med Chem Lett. 2003 Nov 3;13(21):3859-61. doi: 10.1016/s0960-894x(03)00708-x. Bioorg Med Chem Lett. 2003. PMID: 14552795
Oxamides as novel NR2B selective NMDA receptor antagonists.
Barta-Szalai G, Borza I, Bozó E, Kiss C, Agai B, Proszenyák A, Keseru GM, Gere A, Kolok S, Galgóczy K, Horváth C, Farkas S, Domány G. Barta-Szalai G, et al. Among authors: kolok s. Bioorg Med Chem Lett. 2004 Aug 2;14(15):3953-6. doi: 10.1016/j.bmcl.2004.05.053. Bioorg Med Chem Lett. 2004. PMID: 15225705
Indole-2-carboxamidines as novel NR2B selective NMDA receptor antagonists.
Borza I, Kolok S, Ignácz-Szendrei G, Greiner I, Tárkányi G, Galgóczy K, Horváth C, Farkas S, Domány G. Borza I, et al. Among authors: kolok s. Bioorg Med Chem Lett. 2005 Dec 15;15(24):5439-41. doi: 10.1016/j.bmcl.2005.08.110. Epub 2005 Oct 5. Bioorg Med Chem Lett. 2005. PMID: 16213709
Benzimidazole-2-carboxamides as novel NR2B selective NMDA receptor antagonists.
Borza I, Kolok S, Gere A, Nagy J, Fodor L, Galgóczy K, Fetter J, Bertha F, Agai B, Horváth C, Farkas S, Domány G. Borza I, et al. Among authors: kolok s. Bioorg Med Chem Lett. 2006 Sep 1;16(17):4638-40. doi: 10.1016/j.bmcl.2006.06.002. Epub 2006 Jun 16. Bioorg Med Chem Lett. 2006. PMID: 16782335
Kynurenic acid amides as novel NR2B selective NMDA receptor antagonists.
Borza I, Kolok S, Galgóczy K, Gere A, Horváth C, Farkas S, Greiner I, Domány G. Borza I, et al. Among authors: kolok s. Bioorg Med Chem Lett. 2007 Jan 15;17(2):406-9. doi: 10.1016/j.bmcl.2006.10.033. Epub 2006 Oct 17. Bioorg Med Chem Lett. 2007. PMID: 17074483
Selective NR1/2B N-methyl-D-aspartate receptor antagonists among indole-2-carboxamides and benzimidazole-2-carboxamides.
Borza I, Bozó E, Barta-Szalai G, Kiss C, Tárkányi G, Demeter A, Gáti T, Háda V, Kolok S, Gere A, Fodor L, Nagy J, Galgóczy K, Magdó I, Agai B, Fetter J, Bertha F, Keserü GM, Horváth C, Farkas S, Greiner I, Domány G. Borza I, et al. Among authors: kolok s. J Med Chem. 2007 Mar 8;50(5):901-14. doi: 10.1021/jm060420k. Epub 2007 Feb 10. J Med Chem. 2007. PMID: 17290978
Hit-to-lead optimization of disubstituted oxadiazoles and tetrazoles as mGluR5 NAMs.
Wágner G, Wéber C, Nyéki O, Nógrádi K, Bielik A, Molnár L, Bobok A, Horváth A, Kiss B, Kolok S, Nagy J, Kurkó D, Gál K, Greiner I, Szombathelyi Z, Keseru GM, Domány G. Wágner G, et al. Among authors: kolok s. Bioorg Med Chem Lett. 2010 Jun 15;20(12):3737-41. doi: 10.1016/j.bmcl.2010.04.075. Epub 2010 Apr 22. Bioorg Med Chem Lett. 2010. PMID: 20483612
Carbamoyloximes as novel non-competitive mGlu5 receptor antagonists.
Galambos J, Wágner G, Nógrádi K, Bielik A, Molnár L, Bobok A, Horváth A, Kiss B, Kolok S, Nagy J, Kurkó D, Bakk ML, Vastag M, Sághy K, Gyertyán I, Gál K, Greiner I, Szombathelyi Z, Keseru GM, Domány G. Galambos J, et al. Among authors: kolok s. Bioorg Med Chem Lett. 2010 Aug 1;20(15):4371-5. doi: 10.1016/j.bmcl.2010.06.075. Epub 2010 Jun 17. Bioorg Med Chem Lett. 2010. PMID: 20615697
33 results