Klochkov VG - Search Results

1

Towards multi-target antidiabetic agents: In vitro and in vivo evaluation of 3,5-disubstituted indolin-2-one derivatives as novel α-glucosidase inhibitors.

Klochkov VG, Bezsonova EN, Dubar M, Melekhina DD, Temnov VV, Zaryanova EV, Lozinskaya NA, Babkov DA, Spasov AA. Klochkov VG, et al. Bioorg Med Chem Lett. 2022 Jan 1;55:128449. doi: 10.1016/j.bmcl.2021.128449. Epub 2021 Nov 12. Bioorg Med Chem Lett. 2022. PMID: 34780899

2

Synthesis, in vitro and in vivo evaluation of 2-aryl-4H-chromene and 3-aryl-1H-benzo[f]chromene derivatives as novel α-glucosidase inhibitors.

Spasov AA, Babkov DA, Osipov DV, Klochkov VG, Prilepskaya DR, Demidov MR, Osyanin VA, Klimochkin YN. Spasov AA, et al. Among authors: klochkov vg. Bioorg Med Chem Lett. 2019 Jan 1;29(1):119-123. doi: 10.1016/j.bmcl.2018.10.018. Epub 2018 Oct 12. Bioorg Med Chem Lett. 2019. PMID: 30340897

3

[Neural network modeling of multitarget RAGE inhibitory activity].

Vassiliev PM, Spasov AA, Yanaliyeva LR, Kochetkov AN, Vorfolomeyeva VV, Klochkov VG, Appazova DT. Vassiliev PM, et al. Among authors: klochkov vg. Biomed Khim. 2019 Feb;65(2):91-98. doi: 10.18097/PBMC20196502091. Biomed Khim. 2019. PMID: 30950813 Russian.

4

Synthesis and multifaceted pharmacological activity of novel quinazoline NHE-1 inhibitors.

Spasov A, Ozerov A, Vassiliev P, Kosolapov V, Gurova N, Kucheryavenko A, Naumenko L, Babkov D, Sirotenko V, Taran A, Litvinov R, Borisov A, Klochkov V, Merezhkina D, Miroshnikov M, Uskov G, Ovsyankina N. Spasov A, et al. Sci Rep. 2021 Dec 21;11(1):24380. doi: 10.1038/s41598-021-03722-w. Sci Rep. 2021. PMID: 34934125 Free PMC article.

5

Discovery of Nitro-azolo[1,5-a]pyrimidines with Anti-Inflammatory and Protective Activity against LPS-Induced Acute Lung Injury.

Spasov A, Kosolapov V, Babkov D, Klochkov V, Sokolova E, Miroshnikov M, Borisov A, Velikorodnaya Y, Smirnov A, Savateev K, Fedotov V, Kotovskaya S, Rusinov V. Spasov A, et al. Pharmaceuticals (Basel). 2022 Apr 27;15(5):537. doi: 10.3390/ph15050537. Pharmaceuticals (Basel). 2022. PMID: 35631365 Free PMC article.

6

Guanidine Derivatives of Quinazoline-2,4(1H,3H)-Dione as NHE-1 Inhibitors and Anti-Inflammatory Agents.

Spasov A, Ozerov A, Kosolapov V, Gurova N, Kucheryavenko A, Naumenko L, Babkov D, Sirotenko V, Taran A, Borisov A, Sokolova E, Klochkov V, Merezhkina D, Miroshnikov M, Ovsyankina N, Smirnov A, Velikorodnaya Y. Spasov A, et al. Life (Basel). 2022 Oct 20;12(10):1647. doi: 10.3390/life12101647. Life (Basel). 2022. PMID: 36295082 Free PMC article.

7

Design, Synthesis and Pharmacological Evaluation of Novel C²,C³-Quinoxaline Derivatives as Promising Anxiolytic Agents.

Maltsev DV, Skripka MO, Spasov AA, Vassiliev PM, Perfiliev MA, Divaeva LN, Zubenko AA, Morkovnik AS, Klimenko AI, Miroshnikov MV, Klochkov VG, Ianalieva LR. Maltsev DV, et al. Among authors: klochkov vg. Int J Mol Sci. 2022 Nov 19;23(22):14401. doi: 10.3390/ijms232214401. Int J Mol Sci. 2022. PMID: 36430878 Free PMC article.

8

Amino Derivatives of Diaryl Pyrimidines and Azolopyrimidines as Protective Agents against LPS-Induced Acute Lung Injury.

Spasov A, Ovchinnikova I, Fedorova O, Titova Y, Babkov D, Kosolapov V, Borisov A, Sokolova E, Klochkov V, Skripka M, Velikorodnaya Y, Smirnov A, Rusinov G, Charushin V. Spasov A, et al. Molecules. 2023 Jan 11;28(2):741. doi: 10.3390/molecules28020741. Molecules. 2023. PMID: 36677799 Free PMC article.

9

3-Arylidene-2-oxindoles as Potent NRH:Quinone Oxidoreductase 2 Inhibitors.

Lozinskaya NA, Bezsonova EN, Dubar M, Melekhina DD, Bazanov DR, Bunev AS, Grigor'eva OB, Klochkov VG, Sokolova EV, Babkov DA, Spasov AA, Sosonyuk SE. Lozinskaya NA, et al. Among authors: klochkov vg. Molecules. 2023 Jan 25;28(3):1174. doi: 10.3390/molecules28031174. Molecules. 2023. PMID: 36770840 Free PMC article.

10

3-Arylidene-2-oxindoles as GSK3β inhibitors and anti-thrombotic agents.

Babkov D, Bezsonova E, Sirotenko V, Othman E, Klochkov V, Sosonyuk S, Lozinskaya N, Spasov A. Babkov D, et al. Bioorg Med Chem Lett. 2023 May 1;87:129283. doi: 10.1016/j.bmcl.2023.129283. Epub 2023 Apr 11. Bioorg Med Chem Lett. 2023. PMID: 37054760 Free PMC article.

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