Köse M - Search Results

1

8-Benzyltetrahydropyrazino[2,1-f]purinediones: water-soluble tricyclic xanthine derivatives as multitarget drugs for neurodegenerative diseases.

Brunschweiger A, Koch P, Schlenk M, Pineda F, Küppers P, Hinz S, Köse M, Ullrich S, Hockemeyer J, Wiese M, Heer J, Müller CE. Brunschweiger A, et al. Among authors: kose m. ChemMedChem. 2014 Aug;9(8):1704-24. doi: 10.1002/cmdc.201402082. Epub 2014 May 9. ChemMedChem. 2014. PMID: 24817533

2

1,3-Dialkyl-substituted tetrahydropyrimido[1,2-f]purine-2,4-diones as multiple target drugs for the potential treatment of neurodegenerative diseases.

Koch P, Akkari R, Brunschweiger A, Borrmann T, Schlenk M, Küppers P, Köse M, Radjainia H, Hockemeyer J, Drabczyńska A, Kieć-Kononowicz K, Müller CE. Koch P, et al. Among authors: kose m. Bioorg Med Chem. 2013 Dec 1;21(23):7435-52. doi: 10.1016/j.bmc.2013.09.044. Epub 2013 Sep 25. Bioorg Med Chem. 2013. PMID: 24139167

3

2-Amino[1,2,4]triazolo[1,5-c]quinazolines and Derived Novel Heterocycles: Syntheses and Structure-Activity Relationships of Potent Adenosine Receptor Antagonists.

Burbiel JC, Ghattas W, Küppers P, Köse M, Lacher S, Herzner AM, Kombu RS, Akkinepally RR, Hockemeyer J, Müller CE. Burbiel JC, et al. Among authors: kose m. ChemMedChem. 2016 Oct 19;11(20):2272-2286. doi: 10.1002/cmdc.201600255. Epub 2016 Aug 17. ChemMedChem. 2016. PMID: 27531666

4

Szymańska E, Drabczyńska A, Karcz T, Müller CE, Köse M, Karolak-Wojciechowska J, Fruziński A, Schabikowski J, Doroz-Płonka A, Handzlik J, Kieć-Kononowicz K. Szymańska E, et al. Among authors: kose m. Bioorg Med Chem. 2016 Sep 15;24(18):4347-4362. doi: 10.1016/j.bmc.2016.07.028. Epub 2016 Jul 18. Bioorg Med Chem. 2016. PMID: 27485602

5

Focused screening to identify new adenosine kinase inhibitors.

Köse M, Schiedel AC, Bauer AA, Poschenrieder H, Burbiel JC, Akkinepally RR, Stachel HD, Müller CE. Köse M, et al. Bioorg Med Chem. 2016 Nov 1;24(21):5127-5133. doi: 10.1016/j.bmc.2016.08.026. Epub 2016 Aug 21. Bioorg Med Chem. 2016. PMID: 27595538

6

High-affinity, non-nucleotide-derived competitive antagonists of platelet P2Y12 receptors.

Baqi Y, Atzler K, Köse M, Glänzel M, Müller CE. Baqi Y, et al. Among authors: kose m. J Med Chem. 2009 Jun 25;52(12):3784-93. doi: 10.1021/jm9003297. J Med Chem. 2009. PMID: 19463000

7

Characterization of P2X4 receptor agonists and antagonists by calcium influx and radioligand binding studies.

Abdelrahman A, Namasivayam V, Hinz S, Schiedel AC, Köse M, Burton M, El-Tayeb A, Gillard M, Bajorath J, de Ryck M, Müller CE. Abdelrahman A, et al. Among authors: kose m. Biochem Pharmacol. 2017 Feb 1;125:41-54. doi: 10.1016/j.bcp.2016.11.016. Epub 2016 Nov 17. Biochem Pharmacol. 2017. PMID: 27867013

8

Development of [(3)H]2-Carboxy-4,6-dichloro-1H-indole-3-propionic Acid ([(3)H]PSB-12150): A Useful Tool for Studying GPR17.

Köse M, Ritter K, Thiemke K, Gillard M, Kostenis E, Müller CE. Köse M, et al. ACS Med Chem Lett. 2014 Jan 16;5(4):326-30. doi: 10.1021/ml400399f. eCollection 2014 Apr 10. ACS Med Chem Lett. 2014. PMID: 24900835 Free PMC article.

9

Synthesis and Analgesic Activity of Annelated Xanthine Derivatives in Experimental Models in Rodents.

Zygmunt M, Sapa J, Drabczyńska A, Karcz T, Müller C, Köse M, Latacz G, Schabikowski J, Bednarski M, Kieć-Kononowicz K. Zygmunt M, et al. Among authors: kose m. Arch Pharm (Weinheim). 2015 Oct;348(10):704-14. doi: 10.1002/ardp.201500169. Epub 2015 Aug 6. Arch Pharm (Weinheim). 2015. PMID: 26248713

10

Fluorescent-Labeled Selective Adenosine A_2B Receptor Antagonist Enables Competition Binding Assay by Flow Cytometry.

Köse M, Gollos S, Karcz T, Fiene A, Heisig F, Behrenswerth A, Kieć-Kononowicz K, Namasivayam V, Müller CE. Köse M, et al. J Med Chem. 2018 May 24;61(10):4301-4316. doi: 10.1021/acs.jmedchem.7b01627. Epub 2018 May 15. J Med Chem. 2018. PMID: 29681156

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

452 results

Search Page