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Mode of action of p-quinone derivatives with trypanocidal activity studied by experimental and in silico models.
Eur J Med Chem. 2023 Jan 15;246:114926. doi: 10.1016/j.ejmech.2022.114926. Epub 2022 Nov 17.
Eur J Med Chem. 2023.
PMID: 36508970
Design, Synthesis, In Silico Studies and Inhibitory Activity towards Bcr-Abl, BTK and FLT3-ITD of New 2,6,9-Trisubstituted Purine Derivatives as Potential Agents for the Treatment of Leukaemia.
Bertrand J, Dostálová H, Kryštof V, Jorda R, Delgado T, Castro-Alvarez A, Mella J, Cabezas D, Faúndez M, Espinosa-Bustos C, Salas CO.
Bertrand J, et al.
Pharmaceutics. 2022 Jun 17;14(6):1294. doi: 10.3390/pharmaceutics14061294.
Pharmaceutics. 2022.
PMID: 35745866
Free PMC article.
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New 2,6,9-trisubstituted purine derivatives as Bcr-Abl and Btk inhibitors and as promising agents against leukemia.
Bertrand J, Dostálová H, Krystof V, Jorda R, Castro A, Mella J, Espinosa-Bustos C, María Zarate A, Salas CO.
Bertrand J, et al.
Bioorg Chem. 2020 Jan;94:103361. doi: 10.1016/j.bioorg.2019.103361. Epub 2019 Oct 17.
Bioorg Chem. 2020.
PMID: 31699386
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