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Page 1
Discovery of selective 2,4-diaminoquinazoline toll-like receptor 7 (TLR 7) agonists.
Pieters S, McGowan D, Herschke F, Pauwels F, Stoops B, Last S, Embrechts W, Scholliers A, Mostmans W, Van Dijck K, Van Schoubroeck B, Thoné T, De Pooter D, Fanning G, Rosauro ML, Khamlichi MD, Houpis I, Arnoult E, Jonckers THM, Raboisson P. Pieters S, et al. Among authors: houpis i. Bioorg Med Chem Lett. 2018 Feb 15;28(4):711-719. doi: 10.1016/j.bmcl.2018.01.014. Epub 2018 Jan 16. Bioorg Med Chem Lett. 2018. PMID: 29366653
Stereoselective C-glycosylation reactions with arylzinc reagents.
Lemaire S, Houpis IN, Xiao T, Li J, Digard E, Gozlan C, Liu R, Gavryushin A, Diène C, Wang Y, Farina V, Knochel P. Lemaire S, et al. Among authors: houpis in. Org Lett. 2012 Mar 16;14(6):1480-3. doi: 10.1021/ol300220p. Epub 2012 Mar 2. Org Lett. 2012. PMID: 22385274
Synthesis of a muscarinic receptor antagonist via a diastereoselective Michael reaction, selective deoxyfluorination and aromatic metal-halogen exchange reaction.
Mase T, Houpis IN, Akao A, Dorziotis I, Emerson K, Hoang T, Iida T, Itoh T, Kamei K, Kato S, Kato Y, Kawasaki M, Lang F, Lee J, Lynch J, Maligres P, Molina A, Nemoto T, Okada S, Reamer R, Song JZ, Tschaen D, Wada T, Zewge D, Volante RP, Reider PJ, Tomimoto K. Mase T, et al. Among authors: houpis in. J Org Chem. 2001 Oct 5;66(20):6775-86. doi: 10.1021/jo0157425. J Org Chem. 2001. PMID: 11578234
Synthesis of (1R,2S)-1-amino-2-vinylcyclopropanecarboxylic acid vinyl-ACCA) derivatives: key intermediates for the preparation of inhibitors of the hepatitis C virus NS3 protease.
Beaulieu PL, Gillard J, Bailey MD, Boucher C, Duceppe JS, Simoneau B, Wang XJ, Zhang L, Grozinger K, Houpis I, Farina V, Heimroth H, Krueger T, Schnaubelt J. Beaulieu PL, et al. Among authors: houpis i. J Org Chem. 2005 Jul 22;70(15):5869-79. doi: 10.1021/jo050468q. J Org Chem. 2005. PMID: 16018680
Efficient large-scale synthesis of BILN 2061, a potent HCV protease inhibitor, by a convergent approach based on ring-closing metathesis.
Yee NK, Farina V, Houpis IN, Haddad N, Frutos RP, Gallou F, Wang XJ, Wei X, Simpson RD, Feng X, Fuchs V, Xu Y, Tan J, Zhang L, Xu J, Smith-Keenan LL, Vitous J, Ridges MD, Spinelli EM, Johnson M, Donsbach K, Nicola T, Brenner M, Winter E, Kreye P, Samstag W. Yee NK, et al. Among authors: houpis in. J Org Chem. 2006 Sep 15;71(19):7133-45. doi: 10.1021/jo060285j. J Org Chem. 2006. PMID: 16958506
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