Greene G - Search Results

1

Activating ESR1 Mutations Differentially Affect the Efficacy of ER Antagonists.

Toy W, Weir H, Razavi P, Lawson M, Goeppert AU, Mazzola AM, Smith A, Wilson J, Morrow C, Wong WL, De Stanchina E, Carlson KE, Martin TS, Uddin S, Li Z, Fanning S, Katzenellenbogen JA, Greene G, Baselga J, Chandarlapaty S. Toy W, et al. Among authors: greene g. Cancer Discov. 2017 Mar;7(3):277-287. doi: 10.1158/2159-8290.CD-15-1523. Epub 2016 Dec 16. Cancer Discov. 2017. PMID: 27986707 Free PMC article.

2

Identification of cysteine 530 as the covalent attachment site of an affinity-labeling estrogen (ketononestrol aziridine) and antiestrogen (tamoxifen aziridine) in the human estrogen receptor.

Harlow KW, Smith DN, Katzenellenbogen JA, Greene GL, Katzenellenbogen BS. Harlow KW, et al. Among authors: greene gl. J Biol Chem. 1989 Oct 15;264(29):17476-85. J Biol Chem. 1989. PMID: 2793867 Free article.

3

Analysis of the structural core of the human estrogen receptor ligand binding domain by selective proteolysis/mass spectrometric analysis.

Seielstad DA, Carlson KE, Kushner PJ, Greene GL, Katzenellenbogen JA. Seielstad DA, et al. Among authors: greene gl. Biochemistry. 1995 Oct 3;34(39):12605-15. doi: 10.1021/bi00039a016. Biochemistry. 1995. PMID: 7548010

4

Molecular characterization by mass spectrometry of the human estrogen receptor ligand-binding domain expressed in Escherichia coli.

Seielstad DA, Carlson KE, Katzenellenbogen JA, Kushner PJ, Greene GL. Seielstad DA, et al. Among authors: greene gl. Mol Endocrinol. 1995 Jun;9(6):647-58. doi: 10.1210/mend.9.6.8592511. Mol Endocrinol. 1995. PMID: 8592511

5

Allosteric control of ligand selectivity between estrogen receptors alpha and beta: implications for other nuclear receptors.

Nettles KW, Sun J, Radek JT, Sheng S, Rodriguez AL, Katzenellenbogen JA, Katzenellenbogen BS, Greene GL. Nettles KW, et al. Mol Cell. 2004 Feb 13;13(3):317-27. doi: 10.1016/s1097-2765(04)00054-1. Mol Cell. 2004. PMID: 14967140 Free article.

6

Structure-guided optimization of estrogen receptor binding affinity and antagonist potency of pyrazolopyrimidines with basic side chains.

Zhou HB, Sheng S, Compton DR, Kim Y, Joachimiak A, Sharma S, Carlson KE, Katzenellenbogen BS, Nettles KW, Greene GL, Katzenellenbogen JA. Zhou HB, et al. J Med Chem. 2007 Jan 25;50(2):399-403. doi: 10.1021/jm061035y. J Med Chem. 2007. PMID: 17228884

7

Elemental isomerism: a boron-nitrogen surrogate for a carbon-carbon double bond increases the chemical diversity of estrogen receptor ligands.

Zhou HB, Nettles KW, Bruning JB, Kim Y, Joachimiak A, Sharma S, Carlson KE, Stossi F, Katzenellenbogen BS, Greene GL, Katzenellenbogen JA. Zhou HB, et al. Chem Biol. 2007 Jun;14(6):659-69. doi: 10.1016/j.chembiol.2007.04.009. Chem Biol. 2007. PMID: 17584613

8

ESR1 ligand-binding domain mutations in hormone-resistant breast cancer.

Toy W, Shen Y, Won H, Green B, Sakr RA, Will M, Li Z, Gala K, Fanning S, King TA, Hudis C, Chen D, Taran T, Hortobagyi G, Greene G, Berger M, Baselga J, Chandarlapaty S. Toy W, et al. Among authors: greene g. Nat Genet. 2013 Dec;45(12):1439-45. doi: 10.1038/ng.2822. Epub 2013 Nov 3. Nat Genet. 2013. PMID: 24185512 Free PMC article.

9

The uterine and vascular actions of estetrol delineate a distinctive profile of estrogen receptor α modulation, uncoupling nuclear and membrane activation.

Abot A, Fontaine C, Buscato M, Solinhac R, Flouriot G, Fabre A, Drougard A, Rajan S, Laine M, Milon A, Muller I, Henrion D, Adlanmerini M, Valéra MC, Gompel A, Gerard C, Péqueux C, Mestdagt M, Raymond-Letron I, Knauf C, Ferriere F, Valet P, Gourdy P, Katzenellenbogen BS, Katzenellenbogen JA, Lenfant F, Greene GL, Foidart JM, Arnal JF. Abot A, et al. Among authors: greene gl. EMBO Mol Med. 2014 Oct;6(10):1328-46. doi: 10.15252/emmm.201404112. EMBO Mol Med. 2014. PMID: 25214462 Free PMC article.

10

Estrogen receptor alpha somatic mutations Y537S and D538G confer breast cancer endocrine resistance by stabilizing the activating function-2 binding conformation.

Fanning SW, Mayne CG, Dharmarajan V, Carlson KE, Martin TA, Novick SJ, Toy W, Green B, Panchamukhi S, Katzenellenbogen BS, Tajkhorshid E, Griffin PR, Shen Y, Chandarlapaty S, Katzenellenbogen JA, Greene GL. Fanning SW, et al. Among authors: greene gl. Elife. 2016 Feb 2;5:e12792. doi: 10.7554/eLife.12792. Elife. 2016. PMID: 26836308 Free PMC article.

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