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PLBD: protein-ligand binding database of thermodynamic and kinetic intrinsic parameters.
Lingė D, Gedgaudas M, Merkys A, Petrauskas V, Vaitkus A, Grybauskas A, Paketurytė V, Zubrienė A, Zakšauskas A, Mickevičiūtė A, Smirnovienė J, Baranauskienė L, Čapkauskaitė E, Dudutienė V, Urniežius E, Konovalovas A, Kazlauskas E, Shubin K, Schiöth HB, Chen WY, Ladbury JE, Gražulis S, Matulis D. Lingė D, et al. Among authors: grazulis s. Database (Oxford). 2023 Jun 8;2023:baad040. doi: 10.1093/database/baad040. Database (Oxford). 2023. PMID: 37290059 Free PMC article.
Inhibition and binding studies of carbonic anhydrase isozymes I, II and IX with benzimidazo[1,2-c][1,2,3]thiadiazole-7-sulphonamides.
Baranauskienė L, Hilvo M, Matulienė J, Golovenko D, Manakova E, Dudutienė V, Michailovienė V, Torresan J, Jachno J, Parkkila S, Maresca A, Supuran CT, Gražulis S, Matulis D. Baranauskienė L, et al. Among authors: grazulis s. J Enzyme Inhib Med Chem. 2010 Dec;25(6):863-70. doi: 10.3109/14756360903571685. Epub 2010 Feb 18. J Enzyme Inhib Med Chem. 2010. PMID: 20166809
4-[N-(substituted 4-pyrimidinyl)amino]benzenesulfonamides as inhibitors of carbonic anhydrase isozymes I, II, VII, and XIII.
Sūdžius J, Baranauskienė L, Golovenko D, Matulienė J, Michailovienė V, Torresan J, Jachno J, Sukackaitė R, Manakova E, Gražulis S, Tumkevičius S, Matulis D. Sūdžius J, et al. Among authors: grazulis s. Bioorg Med Chem. 2010 Nov 1;18(21):7413-21. doi: 10.1016/j.bmc.2010.09.011. Epub 2010 Sep 8. Bioorg Med Chem. 2010. PMID: 20889345
Benzenesulfonamides with pyrimidine moiety as inhibitors of human carbonic anhydrases I, II, VI, VII, XII, and XIII.
Čapkauskaitė E, Zubrienė A, Smirnov A, Torresan J, Kišonaitė M, Kazokaitė J, Gylytė J, Michailovienė V, Jogaitė V, Manakova E, Gražulis S, Tumkevičius S, Matulis D. Čapkauskaitė E, et al. Among authors: grazulis s. Bioorg Med Chem. 2013 Nov 15;21(22):6937-47. doi: 10.1016/j.bmc.2013.09.029. Epub 2013 Sep 20. Bioorg Med Chem. 2013. PMID: 24103428
4-amino-substituted benzenesulfonamides as inhibitors of human carbonic anhydrases.
Rutkauskas K, Zubrienė A, Tumosienė I, Kantminienė K, Kažemėkaitė M, Smirnov A, Kazokaitė J, Morkūnaitė V, Čapkauskaitė E, Manakova E, Gražulis S, Beresnevičius ZJ, Matulis D. Rutkauskas K, et al. Among authors: grazulis s. Molecules. 2014 Oct 28;19(11):17356-80. doi: 10.3390/molecules191117356. Molecules. 2014. PMID: 25353386 Free PMC article.
Discovery and characterization of novel selective inhibitors of carbonic anhydrase IX.
Dudutienė V, Matulienė J, Smirnov A, Timm DD, Zubrienė A, Baranauskienė L, Morkūnaite V, Smirnovienė J, Michailovienė V, Juozapaitienė V, Mickevičiūtė A, Kazokaitė J, Bakšytė S, Kasiliauskaitė A, Jachno J, Revuckienė J, Kišonaitė M, Pilipuitytė V, Ivanauskaitė E, Milinavičiūtė G, Smirnovas V, Petrikaitė V, Kairys V, Petrauskas V, Norvaišas P, Lingė D, Gibieža P, Capkauskaitė E, Zakšauskas A, Kazlauskas E, Manakova E, Gražulis S, Ladbury JE, Matulis D. Dudutienė V, et al. Among authors: grazulis s. J Med Chem. 2014 Nov 26;57(22):9435-46. doi: 10.1021/jm501003k. Epub 2014 Nov 10. J Med Chem. 2014. PMID: 25358084
Intrinsic Thermodynamics and Structure Correlation of Benzenesulfonamides with a Pyrimidine Moiety Binding to Carbonic Anhydrases I, II, VII, XII, and XIII.
Kišonaitė M, Zubrienė A, Capkauskaitė E, Smirnov A, Smirnovienė J, Kairys V, Michailovienė V, Manakova E, Gražulis S, Matulis D. Kišonaitė M, et al. Among authors: grazulis s. PLoS One. 2014 Dec 10;9(12):e114106. doi: 10.1371/journal.pone.0114106. eCollection 2014. PLoS One. 2014. PMID: 25493428 Free PMC article.
69 results