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Page 1
Novel Copper-Containing Cytotoxic Agents Based on 2-Thioxoimidazolones.
Krasnovskaya OO, Guk DA, Naumov AE, Nikitina VN, Semkina AS, Vlasova KY, Pokrovsky V, Ryabaya OO, Karshieva SS, Skvortsov DA, Zhirkina IV, Shafikov RR, Gorelkin PV, Vaneev AN, Erofeev AS, Mazur DM, Tafeenko VA, Pergushov VI, Melnikov MY, Soldatov MA, Shapovalov VV, Soldatov AV, Akasov RA, Gerasimov VM, Sakharov DA, Moiseeva AA, Zyk NV, Beloglazkina EK, Majouga AG. Krasnovskaya OO, et al. Among authors: gorelkin pv. J Med Chem. 2020 Nov 12;63(21):13031-13063. doi: 10.1021/acs.jmedchem.0c01196. Epub 2020 Oct 20. J Med Chem. 2020. PMID: 32985193
In Vitro and In Vivo Electrochemical Measurement of Reactive Oxygen Species After Treatment with Anticancer Drugs.
Vaneev AN, Gorelkin PV, Garanina AS, Lopatukhina HV, Vodopyanov SS, Alova AV, Ryabaya OO, Akasov RA, Zhang Y, Novak P, Salikhov SV, Abakumov MA, Takahashi Y, Edwards CRW, Klyachko NL, Majouga AG, Korchev YE, Erofeev AS. Vaneev AN, et al. Among authors: gorelkin pv. Anal Chem. 2020 Jun 16;92(12):8010-8014. doi: 10.1021/acs.analchem.0c01256. Epub 2020 May 28. Anal Chem. 2020. PMID: 32441506
New Small-Molecule Glycoconjugates of Docetaxel and GalNAc for Targeted Delivery to Hepatocellular Carcinoma.
Petrov RA, Mefedova SR, Yamansarov EY, Maklakova SY, Grishin DA, Lopatukhina EV, Burenina OY, Lopukhov AV, Kovalev SV, Timchenko YV, Ondar EE, Ivanenkov YA, Evteev SA, Vaneev AN, Timoshenko RV, Klyachko NL, Erofeev AS, Gorelkin PV, Beloglazkina EK, Majouga AG. Petrov RA, et al. Among authors: gorelkin pv. Mol Pharm. 2021 Jan 4;18(1):461-468. doi: 10.1021/acs.molpharmaceut.0c00980. Epub 2020 Dec 2. Mol Pharm. 2021. PMID: 33264010
Discovery of Bivalent GalNAc-Conjugated Betulin as a Potent ASGPR-Directed Agent against Hepatocellular Carcinoma.
Yamansarov EY, Lopatukhina EV, Evteev SA, Skvortsov DA, Lopukhov AV, Kovalev SV, Vaneev AN, Shkil' DO, Akasov RA, Lobov AN, Naumenko VA, Pavlova EN, Ryabaya OO, Burenina OY, Ivanenkov YA, Klyachko NL, Erofeev AS, Gorelkin PV, Beloglazkina EK, Majouga AG. Yamansarov EY, et al. Among authors: gorelkin pv. Bioconjug Chem. 2021 Apr 21;32(4):763-781. doi: 10.1021/acs.bioconjchem.1c00042. Epub 2021 Mar 10. Bioconjug Chem. 2021. PMID: 33691403
Dispirooxindoles Based on 2-Selenoxo-Imidazolidin-4-Ones: Synthesis, Cytotoxicity and ROS Generation Ability.
Novotortsev VK, Kukushkin ME, Tafeenko VA, Skvortsov DA, Kalinina MA, Timoshenko RV, Chmelyuk NS, Vasilyeva LA, Tarasevich BN, Gorelkin PV, Erofeev AS, Majouga AG, Zyk NV, Beloglazkina EK. Novotortsev VK, et al. Among authors: gorelkin pv. Int J Mol Sci. 2021 Mar 5;22(5):2613. doi: 10.3390/ijms22052613. Int J Mol Sci. 2021. PMID: 33807662 Free PMC article.
Synthesis and Biological Evaluation of PSMA Ligands with Aromatic Residues and Fluorescent Conjugates Based on Them.
Machulkin AE, Shafikov RR, Uspenskaya AA, Petrov SA, Ber AP, Skvortsov DA, Nimenko EA, Zyk NU, Smirnova GB, Pokrovsky VS, Abakumov MA, Saltykova IV, Akhmirov RT, Garanina AS, Polshakov VI, Saveliev OY, Ivanenkov YA, Aladinskaya AV, Finko AV, Yamansarov EU, Krasnovskaya OO, Erofeev AS, Gorelkin PV, Dontsova OA, Beloglazkina EK, Zyk NV, Khazanova ES, Majouga AG. Machulkin AE, et al. Among authors: gorelkin pv. J Med Chem. 2021 Apr 22;64(8):4532-4552. doi: 10.1021/acs.jmedchem.0c01935. Epub 2021 Apr 6. J Med Chem. 2021. PMID: 33822606
Mapping mechanical properties of living cells at nanoscale using intrinsic nanopipette-sample force interactions.
Kolmogorov VS , Erofeev AS , Woodcock E , Efremov YM , Iakovlev AP , Savin NA , Alova AV , Lavrushkina SV , Kireev II , Prelovskaya AO , Sviderskaya EV , Scaini D , Klyachko NL , Timashev PS , Takahashi Y , Salikhov SV , Parkhomenko YN , Majouga AG , Edwards CRW , Novak P , Korchev YE , Gorelkin PV . Kolmogorov VS , et al. Among authors: gorelkin pv. Nanoscale. 2021 Apr 7;13(13):6558-6568. doi: 10.1039/d0nr08349f. Epub 2021 Mar 31. Nanoscale. 2021. PMID: 33885535
43 results