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Donepezil Derivatives Targeting Amyloid-β Cascade in Alzheimer's Disease.
Mezeiova E, Chalupova K, Nepovimova E, Gorecki L, Prchal L, Malinak D, Kuca K, Soukup O, Korabecny J. Mezeiova E, et al. Among authors: gorecki l. Curr Alzheimer Res. 2019;16(9):772-800. doi: 10.2174/1567205016666190228122956. Curr Alzheimer Res. 2019. PMID: 30819078 Review.
Profiling donepezil template into multipotent hybrids with antioxidant properties.
Mezeiova E, Spilovska K, Nepovimova E, Gorecki L, Soukup O, Dolezal R, Malinak D, Janockova J, Jun D, Kuca K, Korabecny J. Mezeiova E, et al. Among authors: gorecki l. J Enzyme Inhib Med Chem. 2018 Dec;33(1):583-606. doi: 10.1080/14756366.2018.1443326. J Enzyme Inhib Med Chem. 2018. PMID: 29529892 Free PMC article. Review.
Phenothiazine-Tacrine Heterodimers: Pursuing Multitarget Directed Approach in Alzheimer's Disease.
Gorecki L, Uliassi E, Bartolini M, Janockova J, Hrabinova M, Hepnarova V, Prchal L, Muckova L, Pejchal J, Karasova JZ, Mezeiova E, Benkova M, Kobrlova T, Soukup O, Petralla S, Monti B, Korabecny J, Bolognesi ML. Gorecki L, et al. ACS Chem Neurosci. 2021 May 5;12(9):1698-1715. doi: 10.1021/acschemneuro.1c00184. Epub 2021 Apr 14. ACS Chem Neurosci. 2021. PMID: 33852284
Huprine Y - Tryptophan heterodimers with potential implication to Alzheimer's disease treatment.
Mezeiova E, Hrabinova M, Hepnarova V, Jun D, Janockova J, Muckova L, Prchal L, Kristofikova Z, Kucera T, Gorecki L, Chalupova K, Kunes J, Hroudova J, Soukup O, Korabecny J. Mezeiova E, et al. Among authors: gorecki l. Bioorg Med Chem Lett. 2021 Jul 1;43:128100. doi: 10.1016/j.bmcl.2021.128100. Epub 2021 May 10. Bioorg Med Chem Lett. 2021. PMID: 33984470
A 7-methoxytacrine-4-pyridinealdoxime hybrid as a novel prophylactic agent with reactivation properties in organophosphate intoxication.
Nepovimova E, Korabecny J, Dolezal R, Nguyen TD, Jun D, Soukup O, Pasdiorova M, Jost P, Muckova L, Malinak D, Gorecki L, Musilek K, Kuca K. Nepovimova E, et al. Among authors: gorecki l. Toxicol Res (Camb). 2016 May 25;5(4):1012-1016. doi: 10.1039/c6tx00130k. eCollection 2016 Jul 1. Toxicol Res (Camb). 2016. PMID: 30090408 Free PMC article.
In vitro and in silico Evaluation of Non-Quaternary Reactivators of AChE as Antidotes of Organophosphorus Poisoning - a New Hope or a Blind Alley?
Soukup O, Korabecny J, Malinak D, Nepovimova E, Pham NL, Musilek K, Hrabinova M, Hepnarova V, Dolezal R, Pavek P, Jost P, Kobrlova T, Jankockova J, Gorecki L, Psotka M, Nguyen TD, Box K, Outhwaite B, Ceckova M, Sorf A, Jun D, Kuca K. Soukup O, et al. Among authors: gorecki l. Med Chem. 2018;14(3):281-292. doi: 10.2174/1573406414666180112105657. Med Chem. 2018. PMID: 29332594
Synthesis, in vitro screening and molecular docking of isoquinolinium-5-carbaldoximes as acetylcholinesterase and butyrylcholinesterase reactivators.
Malinak D, Dolezal R, Hepnarova V, Hozova M, Andrys R, Bzonek P, Racakova V, Korabecny J, Gorecki L, Mezeiova E, Psotka M, Jun D, Kuca K, Musilek K. Malinak D, et al. Among authors: gorecki l. J Enzyme Inhib Med Chem. 2020 Dec;35(1):478-488. doi: 10.1080/14756366.2019.1710501. J Enzyme Inhib Med Chem. 2020. PMID: 31910701 Free PMC article.
33 results