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Mild and Efficient Palladium-Mediated C-N Cross-Coupling Reaction between DNA-Conjugated Aryl Bromides and Aromatic Amines.
ACS Comb Sci. 2019 Feb 11;21(2):69-74. doi: 10.1021/acscombsci.8b00142. Epub 2019 Jan 10.
ACS Comb Sci. 2019.
PMID: 30615417
On-DNA Palladium-Catalyzed Hydrogenation-like Reaction Suitable for DNA-Encoded Library Synthesis.
Priego J, de Pedro Beato E, Benavides J, Gironda-Martínez A, González F, Blas J, Martín-Ortega MD, Rama-Garda R, Ezquerra J, Toledo MA, Torrado A.
Priego J, et al. Among authors: gironda martinez a.
Bioconjug Chem. 2021 Jan 20;32(1):88-93. doi: 10.1021/acs.bioconjchem.0c00566. Epub 2020 Dec 24.
Bioconjug Chem. 2021.
PMID: 33356163
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Critical Evaluation of Photo-cross-linking Parameters for the Implementation of Efficient DNA-Encoded Chemical Library Selections.
Sannino A, Gironda-Martínez A, Gorre ÉMD, Prati L, Piazzi J, Scheuermann J, Neri D, Donckele EJ, Samain F.
Sannino A, et al. Among authors: gironda martinez a.
ACS Comb Sci. 2020 Apr 13;22(4):204-212. doi: 10.1021/acscombsci.0c00023. Epub 2020 Mar 6.
ACS Comb Sci. 2020.
PMID: 32109359
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DNA-Compatible Diazo-Transfer Reaction in Aqueous Media Suitable for DNA-Encoded Chemical Library Synthesis.
Gironda-Martínez A, Neri D, Samain F, Donckele EJ.
Gironda-Martínez A, et al.
Org Lett. 2019 Dec 6;21(23):9555-9558. doi: 10.1021/acs.orglett.9b03726. Epub 2019 Nov 20.
Org Lett. 2019.
PMID: 31747292
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DNA-Encoded Chemical Libraries: A Comprehensive Review with Succesful Stories and Future Challenges.
Gironda-Martínez A, Donckele EJ, Samain F, Neri D.
Gironda-Martínez A, et al.
ACS Pharmacol Transl Sci. 2021 Jun 14;4(4):1265-1279. doi: 10.1021/acsptsci.1c00118. eCollection 2021 Aug 13.
ACS Pharmacol Transl Sci. 2021.
PMID: 34423264
Free PMC article.
Review.
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Identification and Validation of New Interleukin-2 Ligands Using DNA-Encoded Libraries.
Gironda-Martínez A, Gorre ÉMD, Prati L, Gosalbes JF, Dakhel S, Cazzamalli S, Samain F, Donckele EJ, Neri D.
Gironda-Martínez A, et al.
J Med Chem. 2021 Dec 9;64(23):17496-17510. doi: 10.1021/acs.jmedchem.1c01693. Epub 2021 Nov 25.
J Med Chem. 2021.
PMID: 34821503
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Multitarget drugs as potential therapeutic agents for alzheimer's disease. A new family of 5-substituted indazole derivatives as cholinergic and BACE1 inhibitors.
González-Naranjo P, Pérez C, González-Sánchez M, Gironda-Martínez A, Ulzurrun E, Bartolomé F, Rubio-Fernández M, Martin-Requero A, Campillo NE, Páez JA.
González-Naranjo P, et al. Among authors: gironda martinez a.
J Enzyme Inhib Med Chem. 2022 Dec;37(1):2348-2356. doi: 10.1080/14756366.2022.2117315.
J Enzyme Inhib Med Chem. 2022.
PMID: 36050834
Free PMC article.
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