Gerhard Gruber - Search Results

Year	Number of Results
2002	4
2003	4
2004	5
2005	2
2006	3
2007	6
2008	8
2009	9
2010	14
2011	12
2012	10
2013	9
2014	8
2015	12
2016	9
2017	15
2018	13
2019	16
2020	15
2021	8
2022	8
2023	7
2024	2

1

High efficacy of the F-ATP synthase inhibitor TBAJ-5307 against nontuberculous mycobacteria in vitro and in vivo.

Ragunathan P, Sae-Lao P, Hamela C, Alcaraz M, Krah A, Poh WH, Ern Pee CJ, Hou Lim AY, Rice SA, Pethe K, Bond PJ, Dick T, Kremer L, Bates RW, Grüber G. Ragunathan P, et al. Among authors: gruber g. J Biol Chem. 2024 Feb;300(2):105618. doi: 10.1016/j.jbc.2023.105618. Epub 2024 Jan 3. J Biol Chem. 2024. PMID: 38176652 Free PMC article.

2

Variations of the Mycobacterium abscessus F-ATP synthase subunit a-c interface alter binding and potency of the anti-TB drug bedaquiline.

Krah A, Ragunathan P, Bond PJ, Grüber G. Krah A, et al. Among authors: gruber g. Biochem Biophys Res Commun. 2024 Jan 1;690:149249. doi: 10.1016/j.bbrc.2023.149249. Epub 2023 Nov 20. Biochem Biophys Res Commun. 2024. PMID: 38000294

3

GaMF1.39's antibiotic efficacy and its enhanced antitubercular activity in combination with clofazimine, Telacebec, ND-011992, or TBAJ-876.

Ragunathan P, Shuyi Ng P, Singh S, Poh WH, Litty D, Kalia NP, Larsson S, Harikishore A, Rice SA, Ingham PW, Müller V, Moraski G, Miller MJ, Dick T, Pethe K, Grüber G. Ragunathan P, et al. Among authors: gruber g. Microbiol Spectr. 2023 Dec 12;11(6):e0228223. doi: 10.1128/spectrum.02282-23. Epub 2023 Nov 20. Microbiol Spectr. 2023. PMID: 37982630 Free PMC article.

4

Novel targets and inhibitors of the Mycobacterium tuberculosis cytochrome bd oxidase to foster anti-tuberculosis drug discovery.

Harikishore A, Mathiyazakan V, Pethe K, Grüber G. Harikishore A, et al. Among authors: gruber g. Expert Opin Drug Discov. 2023 Jul-Dec;18(8):917-927. doi: 10.1080/17460441.2023.2224553. Epub 2023 Jun 18. Expert Opin Drug Discov. 2023. PMID: 37332221 Review.

5

Atomic insights of an up and down conformation of the Acinetobacter baumannii F₁ -ATPase subunit ε and deciphering the residues critical for ATP hydrolysis inhibition and ATP synthesis.

Saw WG, Le KCM, Shin J, Kwek JHM, Wong CF, Ragunathan P, Fong TC, Müller V, Grüber G. Saw WG, et al. Among authors: gruber g. FASEB J. 2023 Jul;37(7):e23040. doi: 10.1096/fj.202300175RR. FASEB J. 2023. PMID: 37318822

6

Cryo-EM structure of the Mycobacterium abscessus F₁-ATPase.

Wong CF, Leow CY, Grüber G. Wong CF, et al. Among authors: gruber g. Biochem Biophys Res Commun. 2023 Sep 3;671:140-145. doi: 10.1016/j.bbrc.2023.05.095. Epub 2023 Jun 5. Biochem Biophys Res Commun. 2023. PMID: 37302287

7

The FGFR inhibitor PD173074 binds to the C-terminus of oncofetal HMGA2 and modulates its DNA-binding and transcriptional activation functions.

Ahmed SM, Ragunathan P, Shin J, Peter S, Kleissle S, Neuenschwander M, Schäfer R, Kries JPV, Grüber G, Dröge P. Ahmed SM, et al. Among authors: gruber g. FEBS Lett. 2023 Aug;597(15):1977-1988. doi: 10.1002/1873-3468.14675. Epub 2023 Jun 8. FEBS Lett. 2023. PMID: 37259564

8

Cryo-Electron Microscopy Structure of the Mycobacterium tuberculosis Cytochrome bcc:aa₃ Supercomplex and a Novel Inhibitor Targeting Subunit Cytochrome cI.

Mathiyazakan V, Wong CF, Harikishore A, Pethe K, Grüber G. Mathiyazakan V, et al. Among authors: gruber g. Antimicrob Agents Chemother. 2023 Jun 15;67(6):e0153122. doi: 10.1128/aac.01531-22. Epub 2023 May 9. Antimicrob Agents Chemother. 2023. PMID: 37158740 Free PMC article.

9

Structural Elements Involved in ATP Hydrolysis Inhibition and ATP Synthesis of Tuberculosis and Nontuberculous Mycobacterial F-ATP Synthase Decipher New Targets for Inhibitors.

Wong CF, Saw WG, Basak S, Sano M, Ueno H, Kerk HW, Litty D, Ragunathan P, Dick T, Müller V, Noji H, Grüber G. Wong CF, et al. Among authors: gruber g. Antimicrob Agents Chemother. 2022 Dec 20;66(12):e0105622. doi: 10.1128/aac.01056-22. Epub 2022 Nov 29. Antimicrob Agents Chemother. 2022. PMID: 36445139 Free PMC article.

10

Structure activity relationship of pyrazinoic acid analogs as potential antimycobacterial agents.

Hegde PV, Aragaw WW, Cole MS, Jachak G, Ragunathan P, Sharma S, Harikishore A, Grüber G, Dick T, Aldrich CC. Hegde PV, et al. Among authors: gruber g. Bioorg Med Chem. 2022 Nov 15;74:117046. doi: 10.1016/j.bmc.2022.117046. Epub 2022 Oct 7. Bioorg Med Chem. 2022. PMID: 36228522 Free PMC article.

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