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Repositioning of Small Molecules through the Inverse Virtual Screening in silico Tool: Case of Benzothiazole-Based Inhibitors of Soluble Epoxide Hydrolase (sEH).
Chempluschem. 2024 May 16:e202400234. doi: 10.1002/cplu.202400234. Online ahead of print.
Chempluschem. 2024.
PMID: 38753468
Prodrug Approach to Exploit (S) Alanine as Arginine Mimic Moiety in the Development of Protein Arginine Methyltransferase 4 Inhibitors.
Milite C, Sarno G, Pacilio I, Cianciulli A, Viviano M, Iannelli G, Gazzillo E, Feoli A, Cipriano A, Chini MG, Castellano S, Bifulco G, Sbardella G.
Milite C, et al. Among authors: gazzillo e.
ChemMedChem. 2024 May 16:e202400139. doi: 10.1002/cmdc.202400139. Online ahead of print.
ChemMedChem. 2024.
PMID: 38752332
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Exploring the Anticancer Potential of Premna resinosa (Hochst.) Leaf Surface Extract: Discovering New Diterpenes as Heat Shock Protein 70 (Hsp70) Binding Agents.
Parisi V, Donadio G, Bellone ML, Belaabed S, Bader A, Bisio A, Iobbi V, Gazzillo E, Chini MG, Bifulco G, Faraone I, Vassallo A.
Parisi V, et al. Among authors: gazzillo e.
Plants (Basel). 2023 Jun 22;12(13):2421. doi: 10.3390/plants12132421.
Plants (Basel). 2023.
PMID: 37446982
Free PMC article.
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Exploring the chemical space of functionalized [1,2,4]triazolo[4,3-a]quinoxaline-based compounds targeting the bromodomain of BRD9.
Gazzillo E, Pierri M, Colarusso E, Chini MG, Ferraro MG, Piccolo M, Irace C, Bruno I, Bifulco G, Terracciano S, Lauro G.
Gazzillo E, et al.
Bioorg Chem. 2023 Oct;139:106677. doi: 10.1016/j.bioorg.2023.106677. Epub 2023 Jun 12.
Bioorg Chem. 2023.
PMID: 37352721
Free article.
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Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders.
Colarusso E, Ceccacci S, Monti MC, Gazzillo E, Giordano A, Chini MG, Ferraro MG, Piccolo M, Ruggiero D, Irace C, Terracciano S, Bruno I, Bifulco G, Lauro G.
Colarusso E, et al. Among authors: gazzillo e.
Eur J Med Chem. 2023 Feb 5;247:115018. doi: 10.1016/j.ejmech.2022.115018. Epub 2022 Dec 17.
Eur J Med Chem. 2023.
PMID: 36577218
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Repositioning of Quinazolinedione-Based Compounds on Soluble Epoxide Hydrolase (sEH) through 3D Structure-Based Pharmacophore Model-Driven Investigation.
Gazzillo E, Terracciano S, Ruggiero D, Potenza M, Chini MG, Lauro G, Fischer K, Hofstetter RK, Giordano A, Werz O, Bruno I, Bifulco G.
Gazzillo E, et al.
Molecules. 2022 Jun 16;27(12):3866. doi: 10.3390/molecules27123866.
Molecules. 2022.
PMID: 35744994
Free PMC article.
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Introducing structure-based three-dimensional pharmacophore models for accelerating the discovery of selective BRD9 binders.
Pierri M, Gazzillo E, Chini MG, Ferraro MG, Piccolo M, Maione F, Irace C, Bifulco G, Bruno I, Terracciano S, Lauro G.
Pierri M, et al. Among authors: gazzillo e.
Bioorg Chem. 2022 Jan;118:105480. doi: 10.1016/j.bioorg.2021.105480. Epub 2021 Nov 15.
Bioorg Chem. 2022.
PMID: 34823196
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