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N'-Phenylacetohydrazide Derivatives as Potent Ebola Virus Entry Inhibitors with an Improved Pharmacokinetic Profile.
Garcia-Rubia A, Lasala F, Ginex T, Morales-Tenorio M, Olal C, Heung M, Oquist P, Galindo I, Cuesta-Geijo MÁ, Casasnovas JM, Campillo NE, Canales Á, Alonso C, Martínez A, Muñoz-Fontela C, Delgado R, Gil C. Garcia-Rubia A, et al. J Med Chem. 2023 Apr 27;66(8):5465-5483. doi: 10.1021/acs.jmedchem.2c01785. Epub 2023 Apr 6. J Med Chem. 2023. PMID: 37021830 Free PMC article.
Deciphering the enzymatic target of a new family of antischistosomal agents bearing a quinazoline scaffold using complementary computational tools.
Sebastian-Perez V, García-Rubia A, Seif El-Din SH, Sabra AA, El-Lakkany NM, William S, Blundell TL, Maes L, Martinez A, Campillo NE, Botros SS, Gil C. Sebastian-Perez V, et al. Among authors: garcia rubia a. J Enzyme Inhib Med Chem. 2020 Dec;35(1):511-523. doi: 10.1080/14756366.2020.1712595. J Enzyme Inhib Med Chem. 2020. PMID: 31939312 Free PMC article.
Identification of potential inhibitors of protein-protein interaction useful to fight against Ebola and other highly pathogenic viruses.
Lasala F, García-Rubia A, Requena C, Galindo I, Cuesta-Geijo MA, García-Dorival I, Bueno P, Labiod N, Luczkowiak J, Martinez A, Campillo NE, Alonso C, Delgado R, Gil C. Lasala F, et al. Among authors: garcia rubia a. Antiviral Res. 2021 Feb;186:105011. doi: 10.1016/j.antiviral.2021.105011. Epub 2021 Jan 8. Antiviral Res. 2021. PMID: 33428961 Free PMC article.
The inhibition of NCS-1 binding to Ric8a rescues fragile X syndrome mice model phenotypes.
Cogram P, Fernández-Beltrán LC, Casarejos MJ, Sánchez-Yepes S, Rodríguez-Martín E, García-Rubia A, Sánchez-Barrena MJ, Gil C, Martínez A, Mansilla A. Cogram P, et al. Among authors: garcia rubia a. Front Neurosci. 2022 Nov 16;16:1007531. doi: 10.3389/fnins.2022.1007531. eCollection 2022. Front Neurosci. 2022. PMID: 36466176 Free PMC article.
Imidazole Derivatives as Promising Agents for the Treatment of Chagas Disease.
de Araújo JS, García-Rubia A, Sebastián-Pérez V, Kalejaiye TD, Bernardino da Silva P, Fonseca-Berzal CR, Maes L, De Koning HP, Soeiro MNC, Gil C. de Araújo JS, et al. Among authors: garcia rubia a. Antimicrob Agents Chemother. 2019 Mar 27;63(4):e02156-18. doi: 10.1128/AAC.02156-18. Print 2019 Apr. Antimicrob Agents Chemother. 2019. PMID: 30670432 Free PMC article.
From Kinase Inhibitors to Multitarget Ligands as Powerful Drug Leads for Alzheimer's Disease using Protein-Templated Synthesis.
Nozal V, García-Rubia A, Cuevas EP, Pérez C, Tosat-Bitrián C, Bartolomé F, Carro E, Ramírez D, Palomo V, Martínez A. Nozal V, et al. Among authors: garcia rubia a. Angew Chem Int Ed Engl. 2021 Aug 23;60(35):19344-19354. doi: 10.1002/anie.202106295. Epub 2021 Jul 26. Angew Chem Int Ed Engl. 2021. PMID: 34169618 Free PMC article.
Screening of a PDE-focused library identifies imidazoles with in vitro and in vivo antischistosomal activity.
Botros SS, William S, Sabra AA, El-Lakkany NM, Seif El-Din SH, García-Rubia A, Sebastián-Pérez V, Blaazer AR, de Heuvel E, Sijm M, Zheng Y, Salado IG, Munday JC, Maes L, de Esch IJP, Sterk GJ, Augustyns K, Leurs R, Gil C, De Koning HP. Botros SS, et al. Among authors: garcia rubia a. Int J Parasitol Drugs Drug Resist. 2019 Apr;9:35-43. doi: 10.1016/j.ijpddr.2019.01.001. Epub 2019 Jan 14. Int J Parasitol Drugs Drug Resist. 2019. PMID: 30669086 Free PMC article.
17 results