Gago F - Search Results

1

TSAO compounds: the comprehensive story of a unique family of HIV-1 specific inhibitors of reverse transcriptase.

Camarasa MJ, San-Félix A, Velázquez S, Pérez-Pérez MJ, Gago F, Balzarini J. Camarasa MJ, et al. Among authors: gago f. Curr Top Med Chem. 2004;4(9):945-63. doi: 10.2174/1568026043388600. Curr Top Med Chem. 2004. PMID: 15134550 Free article. Review.

2

Comparative binding energy analysis of HIV-1 protease inhibitors: incorporation of solvent effects and validation as a powerful tool in receptor-based drug design.

Pérez C, Pastor M, Ortiz AR, Gago F. Pérez C, et al. Among authors: gago f. J Med Chem. 1998 Mar 12;41(6):836-52. doi: 10.1021/jm970535b. J Med Chem. 1998. PMID: 9526559

3

Abasic analogues of TSAO-T as the first sugar derivatives that specifically inhibit HIV-1 reverse transcriptase.

Velázquez S, Chamorro C, Pérez-Pérez MJ, Alvarez R, Jimeno ML, Martín-Domenech A, Pérez C, Gago F, De Clercq E, Balzarini J, San-Félix A, Camarasa MJ. Velázquez S, et al. Among authors: gago f. J Med Chem. 1998 Nov 5;41(23):4636-47. doi: 10.1021/jm980370m. J Med Chem. 1998. PMID: 9804703 Free article.

4

Regiospecific synthesis and anti-human immunodeficiency virus activity of novel 5-substituted N-alkylcarbamoyl and N,N-dialkylcarbamoyl 1,2,3-triazole-TSAO analogues.

Velázquez S, Alvarez R, Pérez C, Gago F, De Clercq E, Balzarini J, Camarasa MJ. Velázquez S, et al. Among authors: gago f. Antivir Chem Chemother. 1998 Nov;9(6):481-9. doi: 10.1177/095632029800900604. Antivir Chem Chemother. 1998. PMID: 9865386

5

Novel 3'-spiro nucleoside analogues of TSAO-T. Part II. A comparative study based on NMR conformational analysis in solution and theoretical calculations.

Alvarez R, Jimeno ML, Gago F, Balzarini J, Pérez-Pérez MJ, Camarasa MJ. Alvarez R, et al. Among authors: gago f. Antivir Chem Chemother. 1998 Jul;9(4):333-40. Antivir Chem Chemother. 1998. PMID: 9875412

6

Identification of a putative binding site for [2',5'-bis-O-(tert-butyldimethylsilyl)-beta-D-ribofuranosyl]-3'-spiro-5''-(4''-amino-1'',2''-oxathiole-2'',2''-dioxide)thymine (TSAO) derivatives at the p51-p66 interface of HIV-1 reverse transcriptase.

Rodríguez-Barrios F, Pérez C, Lobatón E, Velázquez S, Chamorro C, San-Félix A, Pérez-Pérez MJ, Camarasa MJ, Pelemans H, Balzarini J, Gago F. Rodríguez-Barrios F, et al. Among authors: gago f. J Med Chem. 2001 Jun 7;44(12):1853-65. doi: 10.1021/jm001095i. J Med Chem. 2001. PMID: 11384232

7

Exploring the role of the 5'-position of TSAO-T. Synthesis and anti-HIV evaluation of novel TSAO-T derivatives.

Chamorro C, Pérez-Pérez MJ, Rodríguez-Barrios F, Gago F, De Clercq E, Balzarini J, San-Félix A, Camarasa MJ. Chamorro C, et al. Among authors: gago f. Antiviral Res. 2001 Jun;50(3):207-22. doi: 10.1016/s0166-3542(01)00145-0. Antiviral Res. 2001. PMID: 11397508

8

Synthesis of 3' '-substituted TSAO derivatives with anti-HIV-1 and anti-HIV-2 activity through an efficient palladium-catalyzed cross-coupling approach.

Lobatón E, Rodríguez-Barrios F, Gago F, Pérez-Pérez MJ, De Clercq E, Balzarini J, Camarasa MJ, Velázquez S. Lobatón E, et al. Among authors: gago f. J Med Chem. 2002 Aug 29;45(18):3934-45. doi: 10.1021/jm020820h. J Med Chem. 2002. PMID: 12190315

9

Synthesis and structural characterization of pyrimidine bi- and tricyclic nucleosides with sugar puckers conformationally locked into the eastern region of the pseudorotational cycle.

Chamorro C, Luengo SM, Bonache MC, Velázquez S, Pérez-Pérez MJ, Camarasa MJ, Gago F, Jimeno ML, San-Félix A. Chamorro C, et al. Among authors: gago f. J Org Chem. 2003 Aug 22;68(17):6695-704. doi: 10.1021/jo034088l. J Org Chem. 2003. PMID: 12919035

10

Improving the selectivity of acyclic nucleoside analogues as inhibitors of human mitochondrial thymidine kinase: replacement of a triphenylmethoxy moiety with substituted amines and carboxamides.

Hernández AI, Balzarini J, Rodríguez-Barrios F, San-Félix A, Karlsson A, Gago F, Camarasa MJ, Pérez-Pérez MJ. Hernández AI, et al. Among authors: gago f. Bioorg Med Chem Lett. 2003 Sep 15;13(18):3027-30. doi: 10.1016/s0960-894x(03)00639-5. Bioorg Med Chem Lett. 2003. PMID: 12941326

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