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Identification and activity of a series of azole-based compounds with lactate dehydrogenase-directed anti-malarial activity.
Cameron A, Read J, Tranter R, Winter VJ, Sessions RB, Brady RL, Vivas L, Easton A, Kendrick H, Croft SL, Barros D, Lavandera JL, Martin JJ, Risco F, García-Ochoa S, Gamo FJ, Sanz L, Leon L, Ruiz JR, Gabarró R, Mallo A, Gómez de las Heras F. Cameron A, et al. Among authors: gabarro r. J Biol Chem. 2004 Jul 23;279(30):31429-39. doi: 10.1074/jbc.M402433200. Epub 2004 Apr 26. J Biol Chem. 2004. PMID: 15117937 Free article.
Tres Cantos Open Lab: celebrating a decade of innovation in collaboration to combat endemic infectious diseases.
Calderón F, Ballell L, Barros D, Bilbe G, Cammack N, Gabarró R, Halsey A, Heaton PM, Kang G, Mizrahi V, Nathan C, Strange ME, Williams PM, Winzeler EA, Fairlamb AH. Calderón F, et al. Among authors: gabarro r. Nat Rev Drug Discov. 2021 Nov;20(11):799-800. doi: 10.1038/d41573-021-00143-2. Nat Rev Drug Discov. 2021. PMID: 34471283 No abstract available.
Expanding Bromodomain Targeting into Neglected Parasitic Diseases.
Tallant C, Bamborough P, Chung CW, Gamo FJ, Kirkpatrick R, Larminie C, Martín J, Prinjha R, Rioja I, Simola DF, Gabarró R, Calderón F. Tallant C, et al. Among authors: gabarro r. ACS Infect Dis. 2021 Nov 12;7(11):2953-2958. doi: 10.1021/acsinfecdis.1c00387. Epub 2021 Oct 6. ACS Infect Dis. 2021. PMID: 34612618
Bromodomain factor 5 is an essential regulator of transcription in Leishmania.
Jones NG, Geoghegan V, Moore G, Carnielli JBT, Newling K, Calderón F, Gabarró R, Martín J, Prinjha RK, Rioja I, Wilkinson AJ, Mottram JC. Jones NG, et al. Among authors: gabarro r. Nat Commun. 2022 Jul 13;13(1):4071. doi: 10.1038/s41467-022-31742-1. Nat Commun. 2022. PMID: 35831302 Free PMC article.
Case Study of Small Molecules As Antimalarials: 2-Amino-1-phenylethanol (APE) Derivatives.
Chaparro MJ, Vidal J, Angulo-Barturen I, Bueno JM, Burrows J, Cammack N, Castañeda P, Colmenarejo G, Coterón JM, de Las Heras L, Fernández E, Ferrer S, Gabarró R, Gamo FJ, García M, Jiménez-Díaz MB, Lafuente MJ, León ML, Martínez MS, Minick D, Prats S, Puente M, Rueda L, Sandoval E, Santos-Villarejo A, Witty M, Calderón F. Chaparro MJ, et al. Among authors: gabarro r. ACS Med Chem Lett. 2014 Mar 26;5(6):657-61. doi: 10.1021/ml500015r. eCollection 2014 Jun 12. ACS Med Chem Lett. 2014. PMID: 24944739 Free PMC article.
A Focused Screen Identifies Antifolates with Activity on Mycobacterium tuberculosis.
Kumar A, Guardia A, Colmenarejo G, Pérez E, Gonzalez RR, Torres P, Calvo D, Gómez RM, Ortega F, Jiménez E, Gabarro RC, Rullás J, Ballell L, Sherman DR. Kumar A, et al. Among authors: gabarro rc. ACS Infect Dis. 2015 Dec 11;1(12):604-14. doi: 10.1021/acsinfecdis.5b00063. Epub 2015 Aug 12. ACS Infect Dis. 2015. PMID: 26771003 Free PMC article.
Essential Bromodomain TcBDF2 as a Drug Target against Chagas Disease.
Pezza A, Tavernelli LE, Alonso VL, Perdomo V, Gabarro R, Prinjha R, Rodríguez Araya E, Rioja I, Docampo R, Calderón F, Martin J, Serra E. Pezza A, et al. Among authors: gabarro r. ACS Infect Dis. 2022 May 13;8(5):1062-1074. doi: 10.1021/acsinfecdis.2c00057. Epub 2022 Apr 28. ACS Infect Dis. 2022. PMID: 35482332
Complex Interplay between Sphingolipid and Sterol Metabolism Revealed by Perturbations to the Leishmania Metabolome Caused by Miltefosine.
Armitage EG, Alqaisi AQI, Godzien J, Peña I, Mbekeani AJ, Alonso-Herranz V, López-Gonzálvez Á, Martín J, Gabarro R, Denny PW, Barrett MP, Barbas C. Armitage EG, et al. Among authors: gabarro r. Antimicrob Agents Chemother. 2018 Apr 26;62(5):e02095-17. doi: 10.1128/AAC.02095-17. Print 2018 May. Antimicrob Agents Chemother. 2018. PMID: 29463533 Free PMC article.
Metabolic Clustering Analysis as a Strategy for Compound Selection in the Drug Discovery Pipeline for Leishmaniasis.
Armitage EG, Godzien J, Peña I, López-Gonzálvez Á, Angulo S, Gradillas A, Alonso-Herranz V, Martín J, Fiandor JM, Barrett MP, Gabarro R, Barbas C. Armitage EG, et al. Among authors: gabarro r. ACS Chem Biol. 2018 May 18;13(5):1361-1369. doi: 10.1021/acschembio.8b00204. Epub 2018 Apr 24. ACS Chem Biol. 2018. PMID: 29671577 Free article.
11 results