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Characterization of water-soluble esters of nitrobenzoxadiazole-based GSTP1-1 inhibitors for cancer treatment.
Biochem Pharmacol. 2020 Aug;178:114060. doi: 10.1016/j.bcp.2020.114060. Epub 2020 May 29.
Biochem Pharmacol. 2020.
PMID: 32473836
A new nitrobenzoxadiazole-based GSTP1-1 inhibitor with a previously unheard of mechanism of action and high stability.
Fulci C, Rotili D, De Luca A, Stella L, Morozzo Della Rocca B, Forgione M, Di Paolo V, Mai A, Falconi M, Quintieri L, Caccuri AM.
Fulci C, et al.
J Enzyme Inhib Med Chem. 2017 Dec;32(1):240-247. doi: 10.1080/14756366.2016.1247059.
J Enzyme Inhib Med Chem. 2017.
PMID: 28097896
Free PMC article.
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Synthesis and characterisation of a new benzamide-containing nitrobenzoxadiazole as a GSTP1-1 inhibitor endowed with high stability to metabolic hydrolysis.
Di Paolo V, Fulci C, Rotili D, Sciarretta F, Lucidi A, Morozzo Della Rocca B, De Luca A, Rosato A, Quintieri L, Caccuri AM.
Di Paolo V, et al. Among authors: fulci c.
J Enzyme Inhib Med Chem. 2019 Dec;34(1):1131-1139. doi: 10.1080/14756366.2019.1617287.
J Enzyme Inhib Med Chem. 2019.
PMID: 31169043
Free PMC article.
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Effects of Glutathione Transferase-Targeting Nitrobenzoxadiazole Compounds in Relation to PD-L1 Status in Human Melanoma Cells.
Sciarretta F, Fulci C, Palumbo C, Rotili D, Tentori L, Graziani G, Caccuri AM.
Sciarretta F, et al. Among authors: fulci c.
Chemotherapy. 2019;64(3):138-145. doi: 10.1159/000503339. Epub 2019 Oct 22.
Chemotherapy. 2019.
PMID: 31639786
Free article.
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The nitrobenzoxadiazole derivative MC3181 blocks melanoma invasion and metastasis.
De Luca A, Carpanese D, Rapanotti MC, Viguria TM, Forgione MA, Rotili D, Fulci C, Iorio E, Quintieri L, Chimenti S, Bianchi L, Rosato A, Caccuri AM.
De Luca A, et al. Among authors: fulci c.
Oncotarget. 2017 Feb 28;8(9):15520-15538. doi: 10.18632/oncotarget.14690.
Oncotarget. 2017.
PMID: 28107182
Free PMC article.
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Activation of retinal Müller cells in response to glucose variability.
Picconi F, Parravano M, Sciarretta F, Fulci C, Nali M, Frontoni S, Varano M, Caccuri AM.
Picconi F, et al. Among authors: fulci c.
Endocrine. 2019 Sep;65(3):542-549. doi: 10.1007/s12020-019-02017-5. Epub 2019 Jul 20.
Endocrine. 2019.
PMID: 31327157
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Glutathione transferase P silencing promotes neuronal differentiation of retinal R28 cells.
Sciarretta F, Fulci C, Palumbo C, Aquilano K, Pastore A, Iorio E, Lettieri-Barbato D, Cicconi R, Minutolo A, Parravano M, Gilardi M, Varano M, Caccuri AM.
Sciarretta F, et al. Among authors: fulci c.
J Cell Physiol. 2019 Sep;234(9):15885-15897. doi: 10.1002/jcp.28246. Epub 2019 Feb 11.
J Cell Physiol. 2019.
PMID: 30741416
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Molecular and cellular evidence of a direct interaction between the TRAF2 C-terminal domain and ganglioside GM1.
De Luca A, Faienza F, Fulci C, Nicolai E, Calligari P, Palumbo C, Caccuri AM.
De Luca A, et al. Among authors: fulci c.
Int J Biochem Cell Biol. 2024 Feb;167:106508. doi: 10.1016/j.biocel.2023.106508. Epub 2023 Dec 22.
Int J Biochem Cell Biol. 2024.
PMID: 38142771
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