Frédérick R - Search Results

1

Interrogating the Lactate Dehydrogenase Tetramerization Site Using (Stapled) Peptides.

Thabault L, Brisson L, Brustenga C, Martinez Gache SA, Prévost JRC, Kozlova A, Spillier Q, Liberelle M, Benyahia Z, Messens J, Copetti T, Sonveaux P, Frédérick R. Thabault L, et al. Among authors: frederick r. J Med Chem. 2020 May 14;63(9):4628-4643. doi: 10.1021/acs.jmedchem.9b01955. Epub 2020 Apr 15. J Med Chem. 2020. PMID: 32250117

2

Tryptophan 2,3-dioxygenase (TDO) inhibitors. 3-(2-(pyridyl)ethenyl)indoles as potential anticancer immunomodulators.

Dolusić E, Larrieu P, Moineaux L, Stroobant V, Pilotte L, Colau D, Pochet L, Van den Eynde B, Masereel B, Wouters J, Frédérick R. Dolusić E, et al. Among authors: frederick r. J Med Chem. 2011 Aug 11;54(15):5320-34. doi: 10.1021/jm2006782. Epub 2011 Jul 18. J Med Chem. 2011. PMID: 21726069

3

Thiosemicarbazide, a fragment with promising indolamine-2,3-dioxygenase (IDO) inhibition properties.

Serra S, Moineaux L, Vancraeynest C, Masereel B, Wouters J, Pochet L, Frédérick R. Serra S, et al. Among authors: frederick r. Eur J Med Chem. 2014 Jul 23;82:96-105. doi: 10.1016/j.ejmech.2014.05.044. Epub 2014 May 15. Eur J Med Chem. 2014. PMID: 24878638

4

3D-QSAR, design, synthesis and characterization of trisubstituted harmine derivatives with in vitro antiproliferative properties.

Meinguet C, Bruyère C, Frédérick R, Mathieu V, Vancraeynest C, Pochet L, Laloy J, Mortier J, Wolber G, Kiss R, Masereel B, Wouters J. Meinguet C, et al. Among authors: frederick r. Eur J Med Chem. 2015 Apr 13;94:45-55. doi: 10.1016/j.ejmech.2015.02.044. Epub 2015 Feb 24. Eur J Med Chem. 2015. PMID: 25747498 Free article.

5

Synthesis and biological evaluation of di-aryl urea derivatives as c-Kit inhibitors.

Ravez S, Arsenlis S, Barczyk A, Dupont A, Frédérick R, Hesse S, Kirsch G, Depreux P, Goossens L. Ravez S, et al. Among authors: frederick r. Bioorg Med Chem. 2015 Nov 15;23(22):7340-7. doi: 10.1016/j.bmc.2015.10.035. Epub 2015 Oct 24. Bioorg Med Chem. 2015. PMID: 26526740

6

Synthesis, evaluation and structure-activity relationship of new 3-carboxamide coumarins as FXIIa inhibitors.

Bouckaert C, Serra S, Rondelet G, Dolušić E, Wouters J, Dogné JM, Frédérick R, Pochet L. Bouckaert C, et al. Among authors: frederick r. Eur J Med Chem. 2016 Mar 3;110:181-94. doi: 10.1016/j.ejmech.2016.01.023. Epub 2016 Jan 16. Eur J Med Chem. 2016. PMID: 26827162

7

Lactate Dehydrogenase B Controls Lysosome Activity and Autophagy in Cancer.

Brisson L, Bański P, Sboarina M, Dethier C, Danhier P, Fontenille MJ, Van Hée VF, Vazeille T, Tardy M, Falces J, Bouzin C, Porporato PE, Frédérick R, Michiels C, Copetti T, Sonveaux P. Brisson L, et al. Among authors: frederick r. Cancer Cell. 2016 Sep 12;30(3):418-431. doi: 10.1016/j.ccell.2016.08.005. Cancer Cell. 2016. PMID: 27622334 Free article.

8

Challenges and Opportunities in the Development of Serine Synthetic Pathway Inhibitors for Cancer Therapy.

Ravez S, Spillier Q, Marteau R, Feron O, Frédérick R. Ravez S, et al. Among authors: frederick r. J Med Chem. 2017 Feb 23;60(4):1227-1237. doi: 10.1021/acs.jmedchem.6b01167. Epub 2016 Dec 22. J Med Chem. 2017. PMID: 27959531 Review.

9

α-Ketothioamide Derivatives: A Promising Tool to Interrogate Phosphoglycerate Dehydrogenase (PHGDH).

Ravez S, Corbet C, Spillier Q, Dutu A, Robin AD, Mullarky E, Cantley LC, Feron O, Frédérick R. Ravez S, et al. Among authors: frederick r. J Med Chem. 2017 Feb 23;60(4):1591-1597. doi: 10.1021/acs.jmedchem.6b01166. Epub 2017 Jan 27. J Med Chem. 2017. PMID: 28085281 Free PMC article.

10

Radiosynthesis and validation of (±)-[18F]-3-fluoro-2-hydroxypropionate ([18F]-FLac) as a PET tracer of lactate to monitor MCT1-dependent lactate uptake in tumors.

Van Hée VF, Labar D, Dehon G, Grasso D, Grégoire V, Muccioli GG, Frédérick R, Sonveaux P. Van Hée VF, et al. Among authors: frederick r. Oncotarget. 2017 Apr 11;8(15):24415-24428. doi: 10.18632/oncotarget.14705. Oncotarget. 2017. PMID: 28107190 Free PMC article.

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