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Page 1
X-ray screening identifies active site and allosteric inhibitors of SARS-CoV-2 main protease.
Günther S, Reinke PYA, Fernández-García Y, Lieske J, Lane TJ, Ginn HM, Koua FHM, Ehrt C, Ewert W, Oberthuer D, Yefanov O, Meier S, Lorenzen K, Krichel B, Kopicki JD, Gelisio L, Brehm W, Dunkel I, Seychell B, Gieseler H, Norton-Baker B, Escudero-Pérez B, Domaracky M, Saouane S, Tolstikova A, White TA, Hänle A, Groessler M, Fleckenstein H, Trost F, Galchenkova M, Gevorkov Y, Li C, Awel S, Peck A, Barthelmess M, Schlünzen F, Lourdu Xavier P, Werner N, Andaleeb H, Ullah N, Falke S, Srinivasan V, França BA, Schwinzer M, Brognaro H, Rogers C, Melo D, Zaitseva-Doyle JJ, Knoska J, Peña-Murillo GE, Mashhour AR, Hennicke V, Fischer P, Hakanpää J, Meyer J, Gribbon P, Ellinger B, Kuzikov M, Wolf M, Beccari AR, Bourenkov G, von Stetten D, Pompidor G, Bento I, Panneerselvam S, Karpics I, Schneider TR, Garcia-Alai MM, Niebling S, Günther C, Schmidt C, Schubert R, Han H, Boger J, Monteiro DCF, Zhang L, Sun X, Pletzer-Zelgert J, Wollenhaupt J, Feiler CG, Weiss MS, Schulz EC, Mehrabi P, Karničar K, Usenik A, Loboda J, Tidow H, Chari A, Hilgenfeld R, Uetrecht C, Cox R, Zaliani A, Beck T, Rarey M, Günther S, Turk D, Hinrichs W, Chapman HN, Pearson AR, Betzel C, Meents A. Günther S, et al. Among authors: fleckenstein h. Science. 2021 May 7;372(6542):642-646. doi: 10.1126/science.abf7945. Epub 2021 Apr 2. Science. 2021. PMID: 33811162 Free PMC article.
Natively inhibited Trypanosoma brucei cathepsin B structure determined by using an X-ray laser.
Redecke L, Nass K, DePonte DP, White TA, Rehders D, Barty A, Stellato F, Liang M, Barends TRM, Boutet S, Williams GJ, Messerschmidt M, Seibert MM, Aquila A, Arnlund D, Bajt S, Barth T, Bogan MJ, Caleman C, Chao TC, Doak RB, Fleckenstein H, Frank M, Fromme R, Galli L, Grotjohann I, Hunter MS, Johansson LC, Kassemeyer S, Katona G, Kirian RA, Koopmann R, Kupitz C, Lomb L, Martin AV, Mogk S, Neutze R, Shoeman RL, Steinbrener J, Timneanu N, Wang D, Weierstall U, Zatsepin NA, Spence JCH, Fromme P, Schlichting I, Duszenko M, Betzel C, Chapman HN. Redecke L, et al. Among authors: fleckenstein h. Science. 2013 Jan 11;339(6116):227-230. doi: 10.1126/science.1229663. Epub 2012 Nov 29. Science. 2013. PMID: 23196907 Free PMC article.
Electronic damage in S atoms in a native protein crystal induced by an intense X-ray free-electron laser pulse.
Galli L, Son SK, Klinge M, Bajt S, Barty A, Bean R, Betzel C, Beyerlein KR, Caleman C, Doak RB, Duszenko M, Fleckenstein H, Gati C, Hunt B, Kirian RA, Liang M, Nanao MH, Nass K, Oberthür D, Redecke L, Shoeman R, Stellato F, Yoon CH, White TA, Yefanov O, Spence J, Chapman HN. Galli L, et al. Among authors: fleckenstein h. Struct Dyn. 2015 Apr 29;2(4):041703. doi: 10.1063/1.4919398. eCollection 2015 Jul. Struct Dyn. 2015. PMID: 26798803 Free PMC article.
Simple convergent-nozzle aerosol injector for single-particle diffractive imaging with X-ray free-electron lasers.
Kirian RA, Awel S, Eckerskorn N, Fleckenstein H, Wiedorn M, Adriano L, Bajt S, Barthelmess M, Bean R, Beyerlein KR, Chavas LM, Domaracky M, Heymann M, Horke DA, Knoska J, Metz M, Morgan A, Oberthuer D, Roth N, Sato T, Xavier PL, Yefanov O, Rode AV, Küpper J, Chapman HN. Kirian RA, et al. Among authors: fleckenstein h. Struct Dyn. 2015 Jun 19;2(4):041717. doi: 10.1063/1.4922648. eCollection 2015 Jul. Struct Dyn. 2015. PMID: 26798816 Free PMC article.
Post-sample aperture for low background diffraction experiments at X-ray free-electron lasers.
Wiedorn MO, Awel S, Morgan AJ, Barthelmess M, Bean R, Beyerlein KR, Chavas LMG, Eckerskorn N, Fleckenstein H, Heymann M, Horke DA, Knoška J, Mariani V, Oberthür D, Roth N, Yefanov O, Barty A, Bajt S, Küpper J, Rode AV, Kirian RA, Chapman HN. Wiedorn MO, et al. Among authors: fleckenstein h. J Synchrotron Radiat. 2017 Nov 1;24(Pt 6):1296-1298. doi: 10.1107/S1600577517011961. Epub 2017 Oct 16. J Synchrotron Radiat. 2017. PMID: 29091073 Free PMC article.
Analysis of XFEL serial diffraction data from individual crystalline fibrils.
Wojtas DH, Ayyer K, Liang M, Mossou E, Romoli F, Seuring C, Beyerlein KR, Bean RJ, Morgan AJ, Oberthuer D, Fleckenstein H, Heymann M, Gati C, Yefanov O, Barthelmess M, Ornithopoulou E, Galli L, Xavier PL, Ling WL, Frank M, Yoon CH, White TA, Bajt S, Mitraki A, Boutet S, Aquila A, Barty A, Forsyth VT, Chapman HN, Millane RP. Wojtas DH, et al. Among authors: fleckenstein h. IUCrJ. 2017 Oct 20;4(Pt 6):795-811. doi: 10.1107/S2052252517014324. eCollection 2017 Nov 1. IUCrJ. 2017. PMID: 29123682 Free PMC article.
Rapid sample delivery for megahertz serial crystallography at X-ray FELs.
Wiedorn MO, Awel S, Morgan AJ, Ayyer K, Gevorkov Y, Fleckenstein H, Roth N, Adriano L, Bean R, Beyerlein KR, Chen J, Coe J, Cruz-Mazo F, Ekeberg T, Graceffa R, Heymann M, Horke DA, Knoška J, Mariani V, Nazari R, Oberthür D, Samanta AK, Sierra RG, Stan CA, Yefanov O, Rompotis D, Correa J, Erk B, Treusch R, Schulz J, Hogue BG, Gañán-Calvo AM, Fromme P, Küpper J, Rode AV, Bajt S, Kirian RA, Chapman HN. Wiedorn MO, et al. Among authors: fleckenstein h. IUCrJ. 2018 Jul 27;5(Pt 5):574-584. doi: 10.1107/S2052252518008369. eCollection 2018 Sep 1. IUCrJ. 2018. PMID: 30224961 Free PMC article.
Megahertz serial crystallography.
Wiedorn MO, Oberthür D, Bean R, Schubert R, Werner N, Abbey B, Aepfelbacher M, Adriano L, Allahgholi A, Al-Qudami N, Andreasson J, Aplin S, Awel S, Ayyer K, Bajt S, Barák I, Bari S, Bielecki J, Botha S, Boukhelef D, Brehm W, Brockhauser S, Cheviakov I, Coleman MA, Cruz-Mazo F, Danilevski C, Darmanin C, Doak RB, Domaracky M, Dörner K, Du Y, Fangohr H, Fleckenstein H, Frank M, Fromme P, Gañán-Calvo AM, Gevorkov Y, Giewekemeyer K, Ginn HM, Graafsma H, Graceffa R, Greiffenberg D, Gumprecht L, Göttlicher P, Hajdu J, Hauf S, Heymann M, Holmes S, Horke DA, Hunter MS, Imlau S, Kaukher A, Kim Y, Klyuev A, Knoška J, Kobe B, Kuhn M, Kupitz C, Küpper J, Lahey-Rudolph JM, Laurus T, Le Cong K, Letrun R, Xavier PL, Maia L, Maia FRNC, Mariani V, Messerschmidt M, Metz M, Mezza D, Michelat T, Mills G, Monteiro DCF, Morgan A, Mühlig K, Munke A, Münnich A, Nette J, Nugent KA, Nuguid T, Orville AM, Pandey S, Pena G, Villanueva-Perez P, Poehlsen J, Previtali G, Redecke L, Riekehr WM, Rohde H, Round A, Safenreiter T, Sarrou I, Sato T, Schmidt M, Schmitt B, Schönherr R, Schulz J, Sellberg JA, Seibert MM, Seuring C, Shelby ML, Shoeman RL, Sikorski M, Silenzi A, Stan CA, Shi X, Stern S, Sztuk-Dambie… See abstract for full author list ➔ Wiedorn MO, et al. Among authors: fleckenstein h. Nat Commun. 2018 Oct 2;9(1):4025. doi: 10.1038/s41467-018-06156-7. Nat Commun. 2018. PMID: 30279492 Free PMC article.
X-ray focusing with efficient high-NA multilayer Laue lenses.
Bajt S, Prasciolu M, Fleckenstein H, Domaracký M, Chapman HN, Morgan AJ, Yefanov O, Messerschmidt M, Du Y, Murray KT, Mariani V, Kuhn M, Aplin S, Pande K, Villanueva-Perez P, Stachnik K, Chen JP, Andrejczuk A, Meents A, Burkhardt A, Pennicard D, Huang X, Yan H, Nazaretski E, Chu YS, Hamm CE. Bajt S, et al. Among authors: fleckenstein h. Light Sci Appl. 2018 Mar 23;7:17162. doi: 10.1038/lsa.2017.162. eCollection 2018. Light Sci Appl. 2018. PMID: 30839543 Free PMC article.
Coherent diffractive imaging of microtubules using an X-ray laser.
Brändén G, Hammarin G, Harimoorthy R, Johansson A, Arnlund D, Malmerberg E, Barty A, Tångefjord S, Berntsen P, DePonte DP, Seuring C, White TA, Stellato F, Bean R, Beyerlein KR, Chavas LMG, Fleckenstein H, Gati C, Ghoshdastider U, Gumprecht L, Oberthür D, Popp D, Seibert M, Tilp T, Messerschmidt M, Williams GJ, Loh ND, Chapman HN, Zwart P, Liang M, Boutet S, Robinson RC, Neutze R. Brändén G, et al. Among authors: fleckenstein h. Nat Commun. 2019 Jun 13;10(1):2589. doi: 10.1038/s41467-019-10448-x. Nat Commun. 2019. PMID: 31197138 Free PMC article.
46 results