Federico S - Search Results

1

Riluzole-Rasagiline Hybrids: Toward the Development of Multi-Target-Directed Ligands for Amyotrophic Lateral Sclerosis.

Albertini C, Salerno A, Atzeni S, Uliassi E, Massenzio F, Maruca A, Rocca R, Mecava M, Silva FSG, Mena D, Valente P, Duarte AI, Chavarria D, Bissaro M, Moro S, Federico S, Spalluto G, Soukup O, Borges F, Alcaro S, Monti B, Oliveira PJ, Menéndez JC, Bolognesi ML. Albertini C, et al. Among authors: federico s. ACS Chem Neurosci. 2022 Aug 3;13(15):2252-2260. doi: 10.1021/acschemneuro.2c00261. Epub 2022 Jul 22. ACS Chem Neurosci. 2022. PMID: 35868251 Free PMC article.

2

Combining selectivity and affinity predictions using an integrated Support Vector Machine (SVM) approach: An alternative tool to discriminate between the human adenosine A(2A) and A(3) receptor pyrazolo-triazolo-pyrimidine antagonists binding sites.

Michielan L, Bolcato C, Federico S, Cacciari B, Bacilieri M, Klotz KN, Kachler S, Pastorin G, Cardin R, Sperduti A, Spalluto G, Moro S. Michielan L, et al. Among authors: federico s. Bioorg Med Chem. 2009 Jul 15;17(14):5259-74. doi: 10.1016/j.bmc.2009.05.038. Epub 2009 May 21. Bioorg Med Chem. 2009. PMID: 19501513

3

Human A3 adenosine receptor as versatile G protein-coupled receptor example to validate the receptor homology modeling technology.

Morizzo E, Federico S, Spalluto G, Moro S. Morizzo E, et al. Among authors: federico s. Curr Pharm Des. 2009;15(35):4069-84. doi: 10.2174/138161209789824777. Curr Pharm Des. 2009. PMID: 20028322 Review.

4

Receptor-driven identification of novel human A₃ adenosine receptor antagonists as potential therapeutic agents.

Paoletta S, Federico S, Spalluto G, Moro S. Paoletta S, et al. Among authors: federico s. Methods Enzymol. 2010;485:225-44. doi: 10.1016/B978-0-12-381296-4.00013-0. Methods Enzymol. 2010. PMID: 21050920

5

Synthesis and biological evaluation of a new series of 1,2,4-triazolo[1,5-a]-1,3,5-triazines as human A(2A) adenosine receptor antagonists with improved water solubility.

Federico S, Paoletta S, Cheong SL, Pastorin G, Cacciari B, Stragliotto S, Klotz KN, Siegel J, Gao ZG, Jacobson KA, Moro S, Spalluto G. Federico S, et al. J Med Chem. 2011 Feb 10;54(3):877-89. doi: 10.1021/jm101349u. Epub 2011 Jan 7. J Med Chem. 2011. PMID: 21214204 Free PMC article.

6

The A3 adenosine receptor as multifaceted therapeutic target: pharmacology, medicinal chemistry, and in silico approaches.

Cheong SL, Federico S, Venkatesan G, Mandel AL, Shao YM, Moro S, Spalluto G, Pastorin G. Cheong SL, et al. Among authors: federico s. Med Res Rev. 2013 Mar;33(2):235-335. doi: 10.1002/med.20254. Epub 2011 Nov 16. Med Res Rev. 2013. PMID: 22095687 Review.

7

A novel conjugated agent between dopamine and an A2A adenosine receptor antagonist as a potential anti-Parkinson multitarget approach.

Dalpiaz A, Cacciari B, Vicentini CB, Bortolotti F, Spalluto G, Federico S, Pavan B, Vincenzi F, Borea PA, Varani K. Dalpiaz A, et al. Among authors: federico s. Mol Pharm. 2012 Mar 5;9(3):591-604. doi: 10.1021/mp200489d. Epub 2012 Feb 9. Mol Pharm. 2012. PMID: 22292533

8

Therapeutic potential of A2 and A3 adenosine receptor: a review of novel patented ligands.

Federico S, Spalluto G. Federico S, et al. Expert Opin Ther Pat. 2012 Apr;22(4):369-90. doi: 10.1517/13543776.2012.669375. Epub 2012 Mar 22. Expert Opin Ther Pat. 2012. PMID: 22435652 Review.

9

Exploring the directionality of 5-substitutions in a new series of 5-alkylaminopyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine as a strategy to design novel human a(3) adenosine receptor antagonists.

Federico S, Ciancetta A, Sabbadin D, Paoletta S, Pastorin G, Cacciari B, Klotz KN, Moro S, Spalluto G. Federico S, et al. J Med Chem. 2012 Nov 26;55(22):9654-68. doi: 10.1021/jm300899q. Epub 2012 Nov 9. J Med Chem. 2012. PMID: 23098605

10

Fluorescent ligands for adenosine receptors.

Kozma E, Jayasekara PS, Squarcialupi L, Paoletta S, Moro S, Federico S, Spalluto G, Jacobson KA. Kozma E, et al. Among authors: federico s. Bioorg Med Chem Lett. 2013 Jan 1;23(1):26-36. doi: 10.1016/j.bmcl.2012.10.112. Epub 2012 Nov 5. Bioorg Med Chem Lett. 2013. PMID: 23200243 Free PMC article. Review.

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