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Table representation of search results timeline featuring number of search results per year.
Year | Number of Results |
---|---|
2018 | 1 |
2019 | 1 |
2021 | 1 |
2022 | 3 |
2023 | 1 |
2024 | 1 |
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7 results
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Page 1
Groebke Blackburn Bienaymé-mediated multi-component synthesis of selective HDAC6 inhibitors with anti-inflammatory properties.
Bioorg Chem. 2024 Feb;143:107072. doi: 10.1016/j.bioorg.2023.107072. Epub 2024 Jan 2.
Bioorg Chem. 2024.
PMID: 38185013
Photocaged Histone Deacetylase Inhibitors as Prodrugs in Targeted Cancer Therapy.
Kraft FB, Hanl M, Feller F, Schäker-Hübner L, Hansen FK.
Kraft FB, et al.
Pharmaceuticals (Basel). 2023 Feb 25;16(3):356. doi: 10.3390/ph16030356.
Pharmaceuticals (Basel). 2023.
PMID: 36986455
Free PMC article.
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Development of the first non-hydroxamate selective HDAC6 degraders.
Keuler T, König B, Bückreiß N, Kraft FB, König P, Schäker-Hübner L, Steinebach C, Bendas G, Gütschow M, Hansen FK.
Keuler T, et al. Among authors: kraft fb.
Chem Commun (Camb). 2022 Oct 4;58(79):11087-11090. doi: 10.1039/d2cc03712b.
Chem Commun (Camb). 2022.
PMID: 36098075
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Synthesis, Antiplasmodial, and Antileukemia Activity of Dihydroartemisinin-HDAC Inhibitor Hybrids as Multitarget Drugs.
von Bredow L, Schäfer TM, Hogenkamp J, Tretbar M, Stopper D, Kraft FB, Schliehe-Diecks J, Schöler A, Borkhardt A, Bhatia S, Held J, Hansen FK.
von Bredow L, et al. Among authors: kraft fb.
Pharmaceuticals (Basel). 2022 Mar 9;15(3):333. doi: 10.3390/ph15030333.
Pharmaceuticals (Basel). 2022.
PMID: 35337131
Free PMC article.
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Balancing Histone Deacetylase (HDAC) Inhibition and Drug-likeness: Biological and Physicochemical Evaluation of Class I Selective HDAC Inhibitors.
Schäker-Hübner L, Haschemi R, Büch T, Kraft FB, Brumme B, Schöler A, Jenke R, Meiler J, Aigner A, Bendas G, Hansen FK.
Schäker-Hübner L, et al. Among authors: kraft fb.
ChemMedChem. 2022 May 4;17(9):e202100755. doi: 10.1002/cmdc.202100755. Epub 2022 Feb 18.
ChemMedChem. 2022.
PMID: 35073610
Free PMC article.
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4-Acyl Pyrrole Capped HDAC Inhibitors: A New Scaffold for Hybrid Inhibitors of BET Proteins and Histone Deacetylases as Antileukemia Drug Leads.
Schäker-Hübner L, Warstat R, Ahlert H, Mishra P, Kraft FB, Schliehe-Diecks J, Schöler A, Borkhardt A, Breit B, Bhatia S, Hügle M, Günther S, Hansen FK.
Schäker-Hübner L, et al. Among authors: kraft fb.
J Med Chem. 2021 Oct 14;64(19):14620-14646. doi: 10.1021/acs.jmedchem.1c01119. Epub 2021 Sep 28.
J Med Chem. 2021.
PMID: 34582215
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Access to 1-Phospha-2-azanorbornenes by Phospha-aza-Diels-Alder Reactions.
Wonneberger P, König N, Kraft FB, Sárosi MB, Hey-Hawkins E.
Wonneberger P, et al. Among authors: kraft fb.
Angew Chem Int Ed Engl. 2019 Mar 4;58(10):3208-3211. doi: 10.1002/anie.201811673. Epub 2018 Dec 6.
Angew Chem Int Ed Engl. 2019.
PMID: 30375151
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