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Open and rearranged norbornane derived polycyclic cage molecules as potential neuroprotective agents through attenuation of MPP+- and calcium overload-induced excitotoxicity in neuroblastoma SH-SY5Y cells.
Eur J Med Chem. 2020 Oct 15;204:112617. doi: 10.1016/j.ejmech.2020.112617. Epub 2020 Jul 17.
Eur J Med Chem. 2020.
PMID: 32717484
Tricycloundecane Derivatives as Potential N-Methyl-D-aspartate (NMDA) Receptor and Voltage-Gated Calcium Channel Modulators.
Egunlusi AO, Malan SF, Joubert J.
Egunlusi AO, et al.
ChemMedChem. 2015 Jul;10(7):1259-66. doi: 10.1002/cmdc.201500072. Epub 2015 May 26.
ChemMedChem. 2015.
PMID: 26012541
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4-Oxatricyclo[5.2.1.02,6]dec-8-ene-3,5-dione Derivatives as NMDA Receptor- and VGCC Blockers with Neuroprotective Potential.
Egunlusi AO, Malan SF, Omoruyi SI, Ekpo OE, Joubert J.
Egunlusi AO, et al.
Molecules. 2020 Oct 5;25(19):4552. doi: 10.3390/molecules25194552.
Molecules. 2020.
PMID: 33027964
Free PMC article.
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Ever-expanding landscape: Alzheimer's - new targets and new patents.
Egunlusi AO, Joubert J.
Egunlusi AO, et al.
Pharm Pat Anal. 2022 Sep;11(5):135-138. doi: 10.4155/ppa-2022-0031. Epub 2022 Sep 2.
Pharm Pat Anal. 2022.
PMID: 36052611
No abstract available.
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Calcium Modulating Effect of Polycyclic Cages: A Suitable Therapeutic Approach Against Excitotoxic-induced Neurodegeneration.
Egunlusi AO, Malan SF, Palchykov VA, Joubert J.
Egunlusi AO, et al.
Mini Rev Med Chem. 2024 Jan 24. doi: 10.2174/0113895575273868231128104121. Online ahead of print.
Mini Rev Med Chem. 2024.
PMID: 38275027
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