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In Vivo Performance and Properties of Tamoxifen Metabolites for CreERT2 Control.
PLoS One. 2016 Apr 14;11(4):e0152989. doi: 10.1371/journal.pone.0152989. eCollection 2016.
PLoS One. 2016.
PMID: 27077909
Free PMC article.
The "Gatekeeper" Residue Influences the Mode of Binding of Acetyl Indoles to Bromodomains.
Unzue A, Zhao H, Lolli G, Dong J, Zhu J, Zechner M, Dolbois A, Caflisch A, Nevado C.
Unzue A, et al. Among authors: dolbois a.
J Med Chem. 2016 Apr 14;59(7):3087-97. doi: 10.1021/acs.jmedchem.5b01757. Epub 2016 Mar 30.
J Med Chem. 2016.
PMID: 26982797
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Chemical Space Expansion of Bromodomain Ligands Guided by in Silico Virtual Couplings (AutoCouple).
Batiste L, Unzue A, Dolbois A, Hassler F, Wang X, Deerain N, Zhu J, Spiliotopoulos D, Nevado C, Caflisch A.
Batiste L, et al. Among authors: dolbois a.
ACS Cent Sci. 2018 Feb 28;4(2):180-188. doi: 10.1021/acscentsci.7b00401. Epub 2018 Feb 7.
ACS Cent Sci. 2018.
PMID: 29532017
Free PMC article.
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Binding Motifs in the CBP Bromodomain: An Analysis of 20 Crystal Structures of Complexes with Small Molecules.
Zhu J, Dong J, Batiste L, Unzue A, Dolbois A, Pascanu V, Śledź P, Nevado C, Caflisch A.
Zhu J, et al. Among authors: dolbois a.
ACS Med Chem Lett. 2018 Aug 8;9(9):929-934. doi: 10.1021/acsmedchemlett.8b00286. eCollection 2018 Sep 13.
ACS Med Chem Lett. 2018.
PMID: 30258543
Free PMC article.
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Hitting a Moving Target: Simulation and Crystallography Study of ATAD2 Bromodomain Blockers.
Dolbois A, Batiste L, Wiedmer L, Dong J, Brütsch M, Huang D, Deerain NM, Spiliotopoulos D, Cheng-Sánchez I, Laul E, Nevado C, Śledź P, Caflisch A.
Dolbois A, et al.
ACS Med Chem Lett. 2020 Jun 30;11(8):1573-1580. doi: 10.1021/acsmedchemlett.0c00080. eCollection 2020 Aug 13.
ACS Med Chem Lett. 2020.
PMID: 32832026
Free PMC article.
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1,4,9-Triazaspiro[5.5]undecan-2-one Derivatives as Potent and Selective METTL3 Inhibitors.
Dolbois A, Bedi RK, Bochenkova E, Müller A, Moroz-Omori EV, Huang D, Caflisch A.
Dolbois A, et al.
J Med Chem. 2021 Sep 9;64(17):12738-12760. doi: 10.1021/acs.jmedchem.1c00773. Epub 2021 Aug 25.
J Med Chem. 2021.
PMID: 34431664
Free article.
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Selectively Disrupting m6A-Dependent Protein-RNA Interactions with Fragments.
Bedi RK, Huang D, Wiedmer L, Li Y, Dolbois A, Wojdyla JA, Sharpe ME, Caflisch A, Sledz P.
Bedi RK, et al. Among authors: dolbois a.
ACS Chem Biol. 2020 Mar 20;15(3):618-625. doi: 10.1021/acschembio.9b00894. Epub 2020 Mar 2.
ACS Chem Biol. 2020.
PMID: 32101404
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METTL3 Inhibitors for Epitranscriptomic Modulation of Cellular Processes.
Moroz-Omori EV, Huang D, Kumar Bedi R, Cheriyamkunnel SJ, Bochenkova E, Dolbois A, Rzeczkowski MD, Li Y, Wiedmer L, Caflisch A.
Moroz-Omori EV, et al. Among authors: dolbois a.
ChemMedChem. 2021 Oct 6;16(19):3035-3043. doi: 10.1002/cmdc.202100291. Epub 2021 Jul 29.
ChemMedChem. 2021.
PMID: 34237194
Free PMC article.
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