Docsa T - Search Results

1

Dual-Target Compounds against Type 2 Diabetes Mellitus: Proof of Concept for Sodium Dependent Glucose Transporter (SGLT) and Glycogen Phosphorylase (GP) Inhibitors.

Sipos Á, Szennyes E, Hajnal NÉ, Kun S, Szabó KE, Uray K, Somsák L, Docsa T, Bokor É. Sipos Á, et al. Among authors: docsa t. Pharmaceuticals (Basel). 2021 Apr 15;14(4):364. doi: 10.3390/ph14040364. Pharmaceuticals (Basel). 2021. PMID: 33920838 Free PMC article.

2

Efficient inhibition of muscle and liver glycogen phosphorylases by a new glucopyranosylidene-spiro-thiohydantoin.

Osz E, Somsák L, Szilágyi L, Kovács L, Docsa T, Tóth B, Gergely P. Osz E, et al. Among authors: docsa t. Bioorg Med Chem Lett. 1999 May 17;9(10):1385-90. doi: 10.1016/s0960-894x(99)00192-4. Bioorg Med Chem Lett. 1999. PMID: 10360741

3

Synthesis of and a comparative study on the inhibition of muscle and liver glycogen phosphorylases by epimeric pairs of d-gluco- and d-xylopyranosylidene-spiro-(thio)hydantoins and N-(d-glucopyranosyl) amides.

Somsák L, Kovács L, Tóth M, Osz E, Szilágyi L, Györgydeák Z, Dinya Z, Docsa T, Tóth B, Gergely P. Somsák L, et al. Among authors: docsa t. J Med Chem. 2001 Aug 16;44(17):2843-8. doi: 10.1021/jm010892t. J Med Chem. 2001. PMID: 11495595

4

Glucose analog inhibitors of glycogen phosphorylases as potential antidiabetic agents: recent developments.

Somsák L, Nagya V, Hadady Z, Docsa T, Gergely P. Somsák L, et al. Among authors: docsa t. Curr Pharm Des. 2003;9(15):1177-89. doi: 10.2174/1381612033454919. Curr Pharm Des. 2003. PMID: 12769745 Review.

5

Synthesis of N-(beta-D-glucopyranosyl)- and N-(2-acetamido-2-deoxy-beta-D-glucopyranosyl) amides as inhibitors of glycogen phosphorylase.

Györgydeák Z, Hadady Z, Felföldi N, Krakomperger A, Nagy V, Tóth M, Brunyánszki A, Docsa T, Gergely P, Somsák L. Györgydeák Z, et al. Among authors: docsa t. Bioorg Med Chem. 2004 Sep 15;12(18):4861-70. doi: 10.1016/j.bmc.2004.07.013. Bioorg Med Chem. 2004. PMID: 15336265

6

Kinetic and crystallographic studies on 2-(beta-D-glucopyranosyl)-5-methyl-1, 3, 4-oxadiazole, -benzothiazole, and -benzimidazole, inhibitors of muscle glycogen phosphorylase b. Evidence for a new binding site.

Chrysina ED, Kosmopoulou MN, Tiraidis C, Kardakaris R, Bischler N, Leonidas DD, Hadady Z, Somsak L, Docsa T, Gergely P, Oikonomakos NG. Chrysina ED, et al. Among authors: docsa t. Protein Sci. 2005 Apr;14(4):873-88. doi: 10.1110/ps.041216105. Epub 2005 Mar 1. Protein Sci. 2005. PMID: 15741340 Free PMC article.

7

Crystallographic studies on two bioisosteric analogues, N-acetyl-beta-D-glucopyranosylamine and N-trifluoroacetyl-beta-D-glucopyranosylamine, potent inhibitors of muscle glycogen phosphorylase.

Anagnostou E, Kosmopoulou MN, Chrysina ED, Leonidas DD, Hadjiloi T, Tiraidis C, Zographos SE, Györgydeák Z, Somsák L, Docsa T, Gergely P, Kolisis FN, Oikonomakos NG. Anagnostou E, et al. Among authors: docsa t. Bioorg Med Chem. 2006 Jan 1;14(1):181-9. doi: 10.1016/j.bmc.2005.08.010. Epub 2005 Oct 4. Bioorg Med Chem. 2006. PMID: 16213146

8

Synthesis of N-(beta-D-glucopyranosyl) monoamides of dicarboxylic acids as potential inhibitors of glycogen phosphorylase.

Czifrák K, Hadady Z, Docsa T, Gergely P, Schmidt J, Wessjohann L, Somsák L. Czifrák K, et al. Among authors: docsa t. Carbohydr Res. 2006 Jun 12;341(8):947-56. doi: 10.1016/j.carres.2006.03.002. Epub 2006 Mar 29. Carbohydr Res. 2006. PMID: 16564511

9

Synthesis and structure-activity relationships of C-glycosylated oxadiazoles as inhibitors of glycogen phosphorylase.

Tóth M, Kun S, Bokor E, Benltifa M, Tallec G, Vidal S, Docsa T, Gergely P, Somsák L, Praly JP. Tóth M, et al. Among authors: docsa t. Bioorg Med Chem. 2009 Jul 1;17(13):4773-85. doi: 10.1016/j.bmc.2009.04.036. Epub 2009 Apr 23. Bioorg Med Chem. 2009. PMID: 19450985 Free article.

10

Glucose-based spiro-heterocycles as potent inhibitors of glycogen phosphorylase.

Nagy V, Benltifa M, Vidal S, Berzsényi E, Teilhet C, Czifrák K, Batta G, Docsa T, Gergely P, Somsák L, Praly JP. Nagy V, et al. Among authors: docsa t. Bioorg Med Chem. 2009 Aug 1;17(15):5696-707. doi: 10.1016/j.bmc.2009.05.080. Epub 2009 Jun 6. Bioorg Med Chem. 2009. PMID: 19574053

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