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Dipeptidyl-peptidase IV (DPP IV/CD26)-activated prodrugs: a successful strategy for improving water solubility and oral bioavailability.
Curr Med Chem. 2015;22(8):1041-54. doi: 10.2174/0929867322666150114163449.
Curr Med Chem. 2015.
PMID: 25620096
Review.
Efficient conversion of tetrapeptide-based TSAO prodrugs to the parent drug by dipeptidyl-peptidase IV (DPPIV/CD26).
García-Aparicio C, Diez-Torrubia A, Balzarini J, Lambeir AM, Velázquez S, Camarasa MJ.
García-Aparicio C, et al. Among authors: diez torrubia a.
Antiviral Res. 2007 Nov;76(2):130-9. doi: 10.1016/j.antiviral.2007.06.009. Epub 2007 Aug 1.
Antiviral Res. 2007.
PMID: 17675255
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Application of the dipeptidyl peptidase IV (DPPIV/CD26) based prodrug approach to different amine-containing drugs.
Diez-Torrubia A, García-Aparicio C, Cabrera S, De Meester I, Balzarini J, Camarasa MJ, Velázquez S.
Diez-Torrubia A, et al.
J Med Chem. 2010 Jan 28;53(2):559-72. doi: 10.1021/jm901590f.
J Med Chem. 2010.
PMID: 20000418
Free article.
Item in Clipboard
Dipeptidyl peptidase IV dependent water-soluble prodrugs of highly lipophilic bicyclic nucleoside analogues.
Diez-Torrubia A, Balzarini J, Andrei G, Snoeck R, De Meester I, Camarasa MJ, Velázquez S.
Diez-Torrubia A, et al.
J Med Chem. 2011 Mar 24;54(6):1927-42. doi: 10.1021/jm101624e. Epub 2011 Feb 18.
J Med Chem. 2011.
PMID: 21332170
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Dipeptidyl peptidase IV (DPPIV/CD26)-based prodrugs of hydroxy-containing drugs.
Diez-Torrubia A, Cabrera S, Lambeir AM, Balzarini J, Camarasa MJ, Velázquez S.
Diez-Torrubia A, et al.
ChemMedChem. 2012 Apr;7(4):618-28. doi: 10.1002/cmdc.201100504. Epub 2012 Feb 3.
ChemMedChem. 2012.
PMID: 22307932
Free article.
Item in Clipboard
Dipeptidyl peptidase IV-activated prodrugs of anti-varicella zoster virus bicyclic nucleoside analogues containing different self-cleavage spacer systems.
Diez-Torrubia A, Cabrera S, De Meester I, Camarasa MJ, Balzarini J, Velázquez S.
Diez-Torrubia A, et al.
ChemMedChem. 2012 Sep;7(9):1612-22. doi: 10.1002/cmdc.201200295. Epub 2012 Aug 6.
ChemMedChem. 2012.
PMID: 22887971
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Novel water-soluble prodrugs of acyclovir cleavable by the dipeptidyl-peptidase IV (DPP IV/CD26) enzyme.
Diez-Torrubia A, Cabrera S, de Castro S, García-Aparicio C, Mulder G, De Meester I, Camarasa MJ, Balzarini J, Velázquez S.
Diez-Torrubia A, et al.
Eur J Med Chem. 2013;70:456-68. doi: 10.1016/j.ejmech.2013.10.001. Epub 2013 Oct 9.
Eur J Med Chem. 2013.
PMID: 24185376
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Preclinical development of bicyclic nucleoside analogues as potent and selective inhibitors of varicella zoster virus.
McGuigan C, Pathirana RN, Migliore M, Adak R, Luoni G, Jones AT, Díez-Torrubia A, Camarasa MJ, Velázquez S, Henson G, Verbeken E, Sienaert R, Naesens L, Snoeck R, Andrei G, Balzarini J.
McGuigan C, et al. Among authors: diez torrubia a.
J Antimicrob Chemother. 2007 Dec;60(6):1316-30. doi: 10.1093/jac/dkm376. Epub 2007 Oct 22.
J Antimicrob Chemother. 2007.
PMID: 17956908
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