Di Marzo V - Search Results

1

Rational drug design paradigms: the odyssey for designing better drugs.

Kellici T, Ntountaniotis D, Vrontaki E, Liapakis G, Moutevelis-Minakakis P, Kokotos G, Hadjikakou S, Tzakos AG, Afantitis A, Melagraki G, Bryant S, Langer T, Di Marzo V, Mavromoustakos T. Kellici T, et al. Among authors: di marzo v. Comb Chem High Throughput Screen. 2015;18(3):238-56. doi: 10.2174/1386207318666150305125638. Comb Chem High Throughput Screen. 2015. PMID: 25747445 Review.

2

Synthesis and binding study of certain 6-arylalkanamides as molecular probes for cannabinoid receptor subtypes.

Taher AT, Kadry HH, Allarà M, Di Marzo V, Abadi AH, Abouzid KA. Taher AT, et al. Among authors: di marzo v. J Enzyme Inhib Med Chem. 2013 Jun;28(3):436-9. doi: 10.3109/14756366.2011.645241. Epub 2012 Jan 3. J Enzyme Inhib Med Chem. 2013. PMID: 22214210

3

Discovery of glycine sulfonamides as dual inhibitors of sn-1-diacylglycerol lipase α and α/β-hydrolase domain 6.

Janssen FJ, Deng H, Baggelaar MP, Allarà M, van der Wel T, den Dulk H, Ligresti A, van Esbroeck AC, McGuire R, Di Marzo V, Overkleeft HS, van der Stelt M. Janssen FJ, et al. Among authors: di marzo v. J Med Chem. 2014 Aug 14;57(15):6610-22. doi: 10.1021/jm500681z. Epub 2014 Jul 23. J Med Chem. 2014. PMID: 24988361

4

Three-dimensional quantitative structure-selectivity relationships analysis guided rational design of a highly selective ligand for the cannabinoid receptor 2.

Brogi S, Corelli F, Di Marzo V, Ligresti A, Mugnaini C, Pasquini S, Tafi A. Brogi S, et al. Among authors: di marzo v. Eur J Med Chem. 2011 Feb;46(2):547-55. doi: 10.1016/j.ejmech.2010.11.034. Epub 2010 Nov 27. Eur J Med Chem. 2011. PMID: 21183257

5

Rational design, synthesis, and pharmacological properties of new 1,8-naphthyridin-2(1H)-on-3-carboxamide derivatives as highly selective cannabinoid-2 receptor agonists.

Manera C, Saccomanni G, Adinolfi B, Benetti V, Ligresti A, Cascio MG, Tuccinardi T, Lucchesi V, Martinelli A, Nieri P, Masini E, Di Marzo V, Ferrarini PL. Manera C, et al. Among authors: di marzo v. J Med Chem. 2009 Jun 25;52(12):3644-51. doi: 10.1021/jm801563d. J Med Chem. 2009. PMID: 19435366

6

Synthesis, binding studies and molecular modeling of novel cannabinoid receptor ligands.

Osman NA, Mahmoud AH, Allarà M, Niess R, Abouzid KA, Di Marzo V, Abadi AH. Osman NA, et al. Among authors: di marzo v. Bioorg Med Chem. 2010 Dec 15;18(24):8463-77. doi: 10.1016/j.bmc.2010.10.050. Epub 2010 Oct 27. Bioorg Med Chem. 2010. PMID: 21074998

7

Discovery of novel Tetrahydrobenzo[b]thiophene and pyrrole based scaffolds as potent and selective CB2 receptor ligands: The structural elements controlling binding affinity, selectivity and functionality.

Osman NA, Ligresti A, Klein CD, Allarà M, Rabbito A, Di Marzo V, Abouzid KA, Abadi AH. Osman NA, et al. Among authors: di marzo v. Eur J Med Chem. 2016 Oct 21;122:619-634. doi: 10.1016/j.ejmech.2016.07.012. Epub 2016 Jul 9. Eur J Med Chem. 2016. PMID: 27448919

8

Synthesis, binding assays, cytotoxic activity and docking studies of benzimidazole and benzothiophene derivatives with selective affinity for the CB2 cannabinoid receptor.

Romero-Parra J, Mella-Raipán J, Palmieri V, Allarà M, Torres MJ, Pessoa-Mahana H, Iturriaga-Vásquez P, Escobar R, Faúndez M, Di Marzo V, Pessoa-Mahana CD. Romero-Parra J, et al. Among authors: di marzo v. Eur J Med Chem. 2016 Nov 29;124:17-35. doi: 10.1016/j.ejmech.2016.08.005. Epub 2016 Aug 5. Eur J Med Chem. 2016. PMID: 27560280

9

Structure-activity relationships of thiazole and benzothiazole derivatives as selective cannabinoid CB2 agonists with in vivo anti-inflammatory properties.

Ghonim AE, Ligresti A, Rabbito A, Mahmoud AM, Di Marzo V, Osman NA, Abadi AH. Ghonim AE, et al. Among authors: di marzo v. Eur J Med Chem. 2019 Oct 15;180:154-170. doi: 10.1016/j.ejmech.2019.07.002. Epub 2019 Jul 2. Eur J Med Chem. 2019. PMID: 31302448

10

Conformationally constrained fatty acid ethanolamides as cannabinoid and vanilloid receptor probes.

Appendino G, Ligresti A, Minassi A, Cascio MG, Allarà M, Taglialatela-Scafati O, Pertwee RG, De Petrocellis L, Di Marzo V. Appendino G, et al. Among authors: di marzo v. J Med Chem. 2009 May 14;52(9):3001-9. doi: 10.1021/jm900130m. J Med Chem. 2009. PMID: 19361197

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