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Design, synthesis, computational and biological evaluation of new anxiolytics.
Geronikaki A, Babaev E, Dearden J, Dehaen W, Filimonov D, Galaeva I, Krajneva V, Lagunin A, Macaev F, Molodavkin G, Poroikov V, Pogrebnoi S, Saloutin V, Stepanchikova A, Stingaci E, Tkach N, Vlad L, Voronina T. Geronikaki A, et al. Among authors: dehaen w. Bioorg Med Chem. 2004 Dec 15;12(24):6559-68. doi: 10.1016/j.bmc.2004.09.016. Bioorg Med Chem. 2004. PMID: 15556772
Novel D2/5-HT receptor modulators related to cariprazine with potential implication to schizophrenia treatment.
Juza R, Vojtechova I, Stefkova-Mazochova K, Dehaen W, Petrasek T, Prchal L, Kobrlova T, Janousek J, Vlcek P, Mezeiova E, Svozil D, Karasova JZ, Pejchal J, Stark H, Satala G, Bojarski AJ, Kubacka M, Mogilski S, Randakova A, Musilek K, Soukup O, Korabecny J. Juza R, et al. Among authors: dehaen w. Eur J Med Chem. 2022 Mar 15;232:114193. doi: 10.1016/j.ejmech.2022.114193. Epub 2022 Feb 9. Eur J Med Chem. 2022. PMID: 35176563
Synthesis and In Vitro Evaluation of Novel Dopamine Receptor D2 3,4-dihydroquinolin-2(1H)-one Derivatives Related to Aripiprazole.
Juza R, Stefkova K, Dehaen W, Randakova A, Petrasek T, Vojtechova I, Kobrlova T, Pulkrabkova L, Muckova L, Mecava M, Prchal L, Mezeiova E, Musilek K, Soukup O, Korabecny J. Juza R, et al. Among authors: dehaen w. Biomolecules. 2021 Aug 24;11(9):1262. doi: 10.3390/biom11091262. Biomolecules. 2021. PMID: 34572475 Free PMC article.
Pharmacokinetic, pharmacodynamic, and behavioural studies of deschloroketamine in Wistar rats.
Štefková-Mazochová K, Danda H, Dehaen W, Jurásek B, Šíchová K, Pinterová-Leca N, Mazoch V, Krausová BH, Kysilov B, Smejkalová T, Vyklický L, Kohout M, Hájková K, Svozil D, Horsley RR, Kuchař M, Páleníček T. Štefková-Mazochová K, et al. Among authors: dehaen w. Br J Pharmacol. 2022 Jan;179(1):65-83. doi: 10.1111/bph.15680. Epub 2021 Oct 31. Br J Pharmacol. 2022. PMID: 34519023 Free article.
291 results